DK3512846T3 - Ketonhæmmere af lysin-gingipain - Google Patents

Ketonhæmmere af lysin-gingipain Download PDF

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DK3512846T3
DK3512846T3 DK17851664.7T DK17851664T DK3512846T3 DK 3512846 T3 DK3512846 T3 DK 3512846T3 DK 17851664 T DK17851664 T DK 17851664T DK 3512846 T3 DK3512846 T3 DK 3512846T3
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gingipain
lysine
ketone inhibitors
inhibitors
ketone
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DK17851664.7T
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English (en)
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Robert A Galemmo Jr
Stephen S Dominy
Casey C Lynch
Leslie J Holsinger
Andrei W Konradi
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Lighthouse Pharmaceuticals Inc
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    • C07C237/24—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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