DK47489A - Triazolo(-1,5-c)pyrimido(1,4)azin og mellemprodukter til brug ved fremstilling deraf - Google Patents
Triazolo(-1,5-c)pyrimido(1,4)azin og mellemprodukter til brug ved fremstilling derafInfo
- Publication number
- DK47489A DK47489A DK047489A DK47489A DK47489A DK 47489 A DK47489 A DK 47489A DK 047489 A DK047489 A DK 047489A DK 47489 A DK47489 A DK 47489A DK 47489 A DK47489 A DK 47489A
- Authority
- DK
- Denmark
- Prior art keywords
- alkyl
- pyrimido
- triazolo
- compounds
- intermediates
- Prior art date
Links
- 239000000543 intermediate Substances 0.000 title abstract 2
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical compound C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 abstract 1
- 230000007883 bronchodilation Effects 0.000 abstract 1
- 229940124630 bronchodilator Drugs 0.000 abstract 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000001939 inductive effect Effects 0.000 abstract 1
- -1 methylene, carbonyl Chemical group 0.000 abstract 1
- 125000000325 methylidene group Chemical group [H]C([H])=* 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15244388A | 1988-02-05 | 1988-02-05 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK47489D0 DK47489D0 (da) | 1989-02-02 |
| DK47489A true DK47489A (da) | 1989-09-21 |
Family
ID=22542946
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK047489A DK47489A (da) | 1988-02-05 | 1989-02-02 | Triazolo(-1,5-c)pyrimido(1,4)azin og mellemprodukter til brug ved fremstilling deraf |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0327284B1 (da) |
| JP (1) | JP2694990B2 (da) |
| KR (1) | KR890013026A (da) |
| AT (1) | ATE110079T1 (da) |
| AU (1) | AU596764B2 (da) |
| CA (1) | CA1331178C (da) |
| DE (1) | DE68917491T2 (da) |
| DK (1) | DK47489A (da) |
| IE (1) | IE64917B1 (da) |
| NZ (1) | NZ227720A (da) |
| ZA (1) | ZA89639B (da) |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS50116498A (da) * | 1974-02-27 | 1975-09-11 | ||
| US4572910A (en) * | 1983-03-03 | 1986-02-25 | Riker Laboratories, Inc. | Triazolo[1,5-c]pyrimidines substituted by nitrogen-containing heterocyclic rings |
| DK135184A (da) * | 1983-03-03 | 1984-10-10 | Riker Laboratories Inc | Triazol(4,3-c)- og triazol(1,5-c)pyrimidiner |
| EP0181282A1 (de) * | 1984-10-01 | 1986-05-14 | Ciba-Geigy Ag | Triazolochinazolinverbindungen |
| EP0217748B1 (en) * | 1985-09-30 | 1991-02-06 | Ciba-Geigy Ag | 2-Substituted-e-fused-[1,2,4,]triazolo-[1,5-c]pyrimidines pharmaceutical compositions and uses thereof |
| US4639445A (en) * | 1985-10-25 | 1987-01-27 | Riker Laboratories | Metabolites of triazolo[1,5-c]pyrimidines |
| HU195822B (en) * | 1985-12-30 | 1988-07-28 | Gyogyszerkutato Intezet | Process for producing new pyrimido/5,4-b//1,h/oxazine derivatives |
| WO1988002370A1 (en) * | 1986-09-30 | 1988-04-07 | Ciba-Geigy Ag | 2-substituted-e-fused-[1,2,4]triazolo[1,5-c]pyrimidines pharmaceutical compositions and uses thereof |
| US4734413A (en) * | 1987-03-02 | 1988-03-29 | Riker Laboratories, Inc. | Substituted 1,2,4-triazolo[1,5-A]triazines as bronchodilators |
-
1989
- 1989-01-24 IE IE21089A patent/IE64917B1/en not_active IP Right Cessation
- 1989-01-24 CA CA000589003A patent/CA1331178C/en not_active Expired - Fee Related
- 1989-01-25 NZ NZ227720A patent/NZ227720A/xx unknown
- 1989-01-26 ZA ZA89639A patent/ZA89639B/xx unknown
- 1989-01-30 EP EP89300876A patent/EP0327284B1/en not_active Expired - Lifetime
- 1989-01-30 DE DE68917491T patent/DE68917491T2/de not_active Expired - Fee Related
- 1989-01-30 AT AT89300876T patent/ATE110079T1/de active
- 1989-02-02 DK DK047489A patent/DK47489A/da not_active Application Discontinuation
- 1989-02-03 AU AU29598/89A patent/AU596764B2/en not_active Ceased
- 1989-02-04 KR KR1019890001335A patent/KR890013026A/ko not_active Abandoned
- 1989-02-06 JP JP1027333A patent/JP2694990B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| DK47489D0 (da) | 1989-02-02 |
| CA1331178C (en) | 1994-08-02 |
| ATE110079T1 (de) | 1994-09-15 |
| JPH02149584A (ja) | 1990-06-08 |
| EP0327284A3 (en) | 1991-05-02 |
| NZ227720A (en) | 1992-10-28 |
| ZA89639B (en) | 1990-09-26 |
| IE890210L (en) | 1989-08-05 |
| AU596764B2 (en) | 1990-05-10 |
| DE68917491T2 (de) | 1995-02-16 |
| EP0327284A2 (en) | 1989-08-09 |
| AU2959889A (en) | 1989-08-10 |
| EP0327284B1 (en) | 1994-08-17 |
| IE64917B1 (en) | 1995-09-20 |
| JP2694990B2 (ja) | 1997-12-24 |
| KR890013026A (ko) | 1989-09-20 |
| DE68917491D1 (de) | 1994-09-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |