DK507778A - Fremgangsmaade til fremstilling af 4"-deoxy-4"-acylamidoderivater af oleandomycin, erythromycin og erythromycin-carbonat. - Google Patents

Fremgangsmaade til fremstilling af 4"-deoxy-4"-acylamidoderivater af oleandomycin, erythromycin og erythromycin-carbonat.

Info

Publication number: DK507778A
Authority: DK; Denmark
Prior art keywords: erythromycin; oleandomycin; deoxy; procedure; preparation
Prior art date: 1978-01-03

Application number

DK507778A

Other languages

English (en)

Other versions

DK147943B (da

DK147943C (da

Inventor

F C Sciavolino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-01-03

Filing date

1978-11-15

Publication date

1979-07-04

1978-11-15 Application filed by Pfizer filed Critical Pfizer

1979-07-04 Publication of DK507778A publication Critical patent/DK507778A/da

1982-06-10 Priority to DK260982A priority Critical patent/DK153761C/da

1985-01-14 Publication of DK147943B publication Critical patent/DK147943B/da

1985-08-05 Application granted granted Critical

1985-08-05 Publication of DK147943C publication Critical patent/DK147943C/da

Links

ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical compound O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 2
ZWCGOSCDWAAFKK-YZPBMOCRSA-N carbonic acid;(3r,4s,5s,6r,7r,9r,11r,12r,13s,14r)-6-[(2s,3r,4s,6r)-4-(dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-14-ethyl-7,12,13-trihydroxy-4-[(2r,4r,5s,6s)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-3,5,7,9,11,13-hexamethyl-oxacyclotetradecane-2, Chemical compound OC(O)=O.O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ZWCGOSCDWAAFKK-YZPBMOCRSA-N 0.000 title 1
229960003276 erythromycin Drugs 0.000 title 1
RZPAKFUAFGMUPI-KGIGTXTPSA-N oleandomycin Chemical class O1[C@@H](C)[C@H](O)[C@@H](OC)C[C@@H]1O[C@@H]1[C@@H](C)C(=O)O[C@H](C)[C@H](C)[C@H](O)[C@@H](C)C(=O)[C@]2(OC2)C[C@H](C)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C RZPAKFUAFGMUPI-KGIGTXTPSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Communicable Diseases (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK507778A 1978-01-03 1978-11-15 Analogifremgangsmaade til fremstilling af 4''-deoxy-4''-acylamidoderivater af oleandomycin-forbindelser, erythromycin-forbindelser eller erythromycin-6,9-hemiketal-forbindelser DK147943C (da)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK260982A DK153761C (da)	1978-01-03	1982-06-10	Analogifremgangsmaade til fremstilling af 4ae-deoxo-4ae-acylamidoderivater af erythromycylamin og erythromycyliminderivater til anvendelse som udgangsmateriale ved denne fremgangsmaade

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US86672278A	1978-01-03	1978-01-03
US86672278		1978-01-03
US93764078		1978-08-29
US05/937,640 US4180654A (en)	1978-01-03	1978-08-29	4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate

Publications (3)

Publication Number	Publication Date
DK507778A true DK507778A (da)	1979-07-04
DK147943B DK147943B (da)	1985-01-14
DK147943C DK147943C (da)	1985-08-05

Family

ID=27127966

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK507778A DK147943C (da)	1978-01-03	1978-11-15	Analogifremgangsmaade til fremstilling af 4''-deoxy-4''-acylamidoderivater af oleandomycin-forbindelser, erythromycin-forbindelser eller erythromycin-6,9-hemiketal-forbindelser

Country Status (28)

Country	Link
US (1)	US4180654A (da)
JP (1)	JPS5495585A (da)
AT (1)	AT364457B (da)
AU (1)	AU506684B2 (da)
CH (1)	CH639972A5 (da)
CS (1)	CS204042B2 (da)
DD (1)	DD141026A5 (da)
DE (2)	DE2900118A1 (da)
DK (1)	DK147943C (da)
ES (2)	ES476544A1 (da)
FI (1)	FI68058C (da)
FR (1)	FR2413403A1 (da)
GB (1)	GB2013181B (da)
GR (1)	GR72779B (da)
HU (1)	HU180276B (da)
IE (1)	IE47642B1 (da)
IL (1)	IL56363A (da)
IN (1)	IN150395B (da)
IT (1)	IT1109925B (da)
LU (1)	LU80747A1 (da)
NL (1)	NL176461C (da)
NO (2)	NO146711C (da)
NZ (1)	NZ189274A (da)
PH (4)	PH14745A (da)
PL (2)	PL118573B1 (da)
PT (1)	PT69014A (da)
SE (2)	SE447118B (da)
YU (2)	YU312278A (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5848285U (ja) *	1981-09-26	1983-04-01	コナミ工業株式会社	テ−ブル型テレビゲ−ム機
US4429116A (en) *	1982-12-27	1984-01-31	Pfizer Inc.	Alkylated oleandomycin containing compounds
US4518590A (en) *	1984-04-13	1985-05-21	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
JPS62240086A (ja) *	1986-04-12	1987-10-20	株式会社　エ−ス電研	遊技機の前面構造
US5075289A (en) *	1988-06-07	1991-12-24	Abbott Laboratories	9-r-azacyclic erythromycin antibiotics
SI9010556B (sl) *	1990-03-21	1998-10-31	Pliva	Oleandomicin oksimi in postopek za njihovo pripravo
EP1628989B1 (en) *	2003-05-13	2006-12-20	Glaxo Group Limited	Novel 14 and 15 membered-ring compounds
GB0310984D0 (en) *	2003-05-13	2003-06-18	Glaxo Group Ltd	Novel compounds
GB0310992D0 (en) *	2003-05-13	2003-06-18	Glaxo Group Ltd	Novel compounds
GB0310980D0 (en) *	2003-05-13	2003-06-18	Glaxo Group Ltd	Novel compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3869445A (en) *	1973-05-03	1975-03-04	Abbott Lab	4{41 -O-sulfonyl erythromycin-9-O-oxime derivatives
US3884902A (en) *	1973-05-04	1975-05-20	Abbott Lab	Sulfonyl derivatives of erythromycin
US3884903A (en) *	1973-06-21	1975-05-20	Abbott Lab	4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
US4063014A (en) *	1975-06-12	1977-12-13	Abbott Laboratories	4"-O-sulfonyl erythromycin-9-O-oxime derivatives
US4069379A (en) *	1976-07-08	1978-01-17	Pfizer Inc.	Semi-synthetic oleandomycins
IE44509B1 (en) *	1976-03-03	1981-12-30	Pfizer	Semi-synthetic oleandomycins
US4085119A (en) *	1977-02-04	1978-04-18	Pfizer Inc.	4-Substituted amino derivatives of oleandomycin
US4090017A (en) *	1977-02-04	1978-05-16	Pfizer Inc.	4-Deoxy-4-substituted amino derivatives of oleandomycin

1978
- 1978-08-29 US US05/937,640 patent/US4180654A/en not_active Expired - Lifetime
- 1978-11-15 DK DK507778A patent/DK147943C/da not_active IP Right Cessation
- 1978-11-20 IN IN830/DEL/78A patent/IN150395B/en unknown
- 1978-12-20 GB GB7849227A patent/GB2013181B/en not_active Expired
- 1978-12-21 CH CH1303678A patent/CH639972A5/de not_active IP Right Cessation
- 1978-12-21 NZ NZ189274A patent/NZ189274A/xx unknown
- 1978-12-28 YU YU03122/78A patent/YU312278A/xx unknown
- 1978-12-28 JP JP16447078A patent/JPS5495585A/ja active Granted
- 1978-12-29 HU HU78PI660A patent/HU180276B/hu not_active IP Right Cessation
- 1978-12-29 AU AU42985/78A patent/AU506684B2/en not_active Expired
- 1978-12-30 GR GR58008A patent/GR72779B/el unknown
1979
- 1979-01-02 IT IT19013/79A patent/IT1109925B/it active
- 1979-01-02 FR FR7900014A patent/FR2413403A1/fr active Granted
- 1979-01-02 LU LU80747A patent/LU80747A1/xx unknown
- 1979-01-02 PH PH22004A patent/PH14745A/en unknown
- 1979-01-02 ES ES476544A patent/ES476544A1/es not_active Expired
- 1979-01-02 SE SE7900028A patent/SE447118B/sv not_active IP Right Cessation
- 1979-01-02 AT AT0002979A patent/AT364457B/de not_active IP Right Cessation
- 1979-01-02 IE IE5/79A patent/IE47642B1/en not_active IP Right Cessation
- 1979-01-02 NL NLAANVRAGE7900006,A patent/NL176461C/xx not_active IP Right Cessation
- 1979-01-02 IL IL56363A patent/IL56363A/xx not_active IP Right Cessation
- 1979-01-02 PT PT69014A patent/PT69014A/pt unknown
- 1979-01-02 NO NO790006A patent/NO146711C/no unknown
- 1979-01-02 FI FI790004A patent/FI68058C/fi not_active IP Right Cessation
- 1979-01-03 DE DE19792900118 patent/DE2900118A1/de active Granted
- 1979-01-03 PL PL1979227812A patent/PL118573B1/pl unknown
- 1979-01-03 DD DD79210317A patent/DD141026A5/de unknown
- 1979-01-03 DE DE2953969A patent/DE2953969C2/de not_active Expired
- 1979-01-03 CS CS79100A patent/CS204042B2/cs unknown
- 1979-01-03 PL PL1979212593A patent/PL117603B1/pl unknown
- 1979-07-11 ES ES482420A patent/ES482420A1/es not_active Expired
- 1979-12-21 PH PH23451A patent/PH15752A/en unknown
- 1979-12-21 PH PH23449A patent/PH15439A/en unknown
- 1979-12-21 PH PH23450A patent/PH15626A/en unknown
1982
- 1982-02-26 NO NO820613A patent/NO147716C/no unknown
- 1982-09-24 YU YU02139/82A patent/YU213982A/xx unknown
1983
- 1983-08-15 SE SE8304417A patent/SE448385B/sv not_active IP Right Cessation

Also Published As

Publication number	Publication date
SE7900028L (sv)	1979-07-04
IE790005L (en)	1979-07-03
DK147943B (da)	1985-01-14
NZ189274A (en)	1982-03-23
NO146711C (no)	1982-11-24
SE448385B (sv)	1987-02-16
IT1109925B (it)	1985-12-23
JPS5495585A (en)	1979-07-28
CS204042B2 (en)	1981-03-31
SE447118B (sv)	1986-10-27
ATA2979A (de)	1981-03-15
PL212593A1 (pl)	1979-08-27
NL7900006A (nl)	1979-07-05
DE2900118A1 (de)	1979-07-05
DK147943C (da)	1985-08-05
PH15626A (en)	1983-03-11
IE47642B1 (en)	1984-05-16
LU80747A1 (fr)	1979-09-07
HU180276B (en)	1983-02-28
IL56363A (en)	1982-12-31
PT69014A (en)	1979-02-01
PH15439A (en)	1983-01-18
DE2900118C2 (da)	1987-09-17
US4180654A (en)	1979-12-25
JPS5734280B2 (da)	1982-07-22
FI68058B (fi)	1985-03-29
FI68058C (fi)	1985-07-10
FR2413403A1 (fr)	1979-07-27
CH639972A5 (de)	1983-12-15
GR72779B (da)	1983-12-05
ES482420A1 (es)	1980-09-01
PH14745A (en)	1981-11-20
GB2013181A (en)	1979-08-08
IT7919013A0 (it)	1979-01-02
IL56363A0 (en)	1979-03-12
NO790006L (no)	1979-07-04
PH15752A (en)	1983-03-18
IN150395B (da)	1982-09-25
GB2013181B (en)	1982-06-03
DE2953969C2 (da)	1987-09-03
FR2413403B1 (da)	1982-07-23
AT364457B (de)	1981-10-27
NO147716B (no)	1983-02-21
PL117603B1 (en)	1981-08-31
ES476544A1 (es)	1979-12-01
DD141026A5 (de)	1980-04-09
PL118573B1 (en)	1981-10-31
SE8304417D0 (sv)	1983-08-15
FI790004A7 (fi)	1979-07-04
AU4298578A (en)	1979-07-12
YU312278A (en)	1983-01-21
NL176461C (nl)	1985-04-16
SE8304417L (sv)	1983-08-15
NO147716C (no)	1983-06-01
NO820613L (no)	1979-07-04
YU213982A (en)	1983-02-28
AU506684B2 (en)	1980-01-17
NO146711B (no)	1982-08-16

Legal Events

Date	Code	Title	Description
1995-07-24	PBP	Patent lapsed

Publication	Publication Date	Title
MX9203151A (es)	1992-07-01	Conjugado inmunogenico.
NO160103C (no)	1989-03-08	Jodtyroninimmunogenkonjugat og jodtyroninderivat for fremstilling av jodtyroninimmunogenkonjugatet.
IT1110821B (it)	1986-01-06	Copolimeri di organopolisilosani polisequenziati,cristallini e loro procedimenti di preparazione
NL7805814A (nl)	1979-08-15	Spiro-aminederivaten, de bereiding ervan, alsmede der- gelijke derivaten bevattende farmacologische prepara- ten.
DK498080A (da)	1981-05-23	Fremgangsmaade til fremstilling af 4!-epidaunorubicin, 3!,4!-diepidaunorubicin og disses doxorubicinanaloge
DK467377A (da)	1978-08-25	Fremgangsmaade til fremstilling af 1,4,3,6-dianhydro-d-glucitol-2-nitrat.
NL7806208A (nl)	1978-12-12	7 alfa-methoxy-7 beta-(1,3-dithietan-2-carboxamide) ce- falosporanzuurderivaten en de bereiding, alsmede de toepassing ervan.
NO790934L (no)	1979-09-25	2,6-dialkoksybenzamider og fremgangsmaate til deres fremstilling
NO793192L (no)	1980-04-09	4-fenyl-1,3-benzodiazepiner og fremgangsmaate til deres fremstilling.
SE8304417L (sv)	1983-08-15	Erythromycinderivat
AR216558A1 (es)	1979-12-28	Procedimiento de preparacion de 1,3-dihidro-3-(3',4',5'-trimetoxi-estiril)-6-metil-7-hidroxi-furo-(3,4,c)-piridina
DK582578A (da)	1979-06-30	2,4-thiazolidindion-derivater og fremgangsmaade til deres fremstilling
DK270077A (da)	1977-12-22	6,7-benzomorphanderivater og fremgangsmade til deres fremstillling
DK514382A (da)	1983-05-20	Azolylvinyldithioacetaler, deres fremstilling og anvendelse
NL7804361A (nl)	1978-10-27	Leucinerijk 3,1-s-alpha2-glycoproteine, zijn berei- ding en toepassing.
FI802283A7 (fi)	1981-01-01	Menetelmä 1,2-dihydro-2-okso- 5(pyridinyyli)-nikotiininitriilien valmistamiseksi.
DK162979C (da)	1992-06-01	Polyfluoralkylestere, deres fremstilling og anvendelse
IT7829638A0 (it)	1978-11-09	2,4-diammino-5-benzil-pirimidine eprocedimento per la loro preparazione.
DK364582A (da)	1983-02-15	5(6)-phenylsulfonyloxy-benzimidazolderivater, deres fremstilling og anvendelse
ES515559A0 (es)	1983-10-16	Procedimiento para preparar 1,2-dihidropirido (3,4 6) pirazinas.
NL7800687A (nl)	1978-08-08	2,9-dioxatricyclo(4,3,1,0,3,7)decanen en werkwijze ter bereiding daarvan.
NO822200L (no)	1982-12-30	24-cyklopropylcholen-3beta,22-dioler og fremgangsmaate for deres fremstilling.
ES492747A0 (es)	1981-06-01	Procedimiento de preparacion de 2-isopropilamino-pirimidina.
DK516982A (da)	1983-06-15	P-phenylendiaminer, deres fremstilling og anvendelse
AR222647A1 (es)	1981-06-15	Procedimiento para la preparacion de derivados 4"-deoxi-4"-acilamino de oleandomicina,eritromicina,y carbonato de eritromicina