DK526989A - Fremgangsmaade til fremstilling af 1,4-diazabicyclo(3.2.2)nonan samt mellemprodukter ved fremgangsmaaden og fremgangsmaader til fremstilling af disse - Google Patents
Fremgangsmaade til fremstilling af 1,4-diazabicyclo(3.2.2)nonan samt mellemprodukter ved fremgangsmaaden og fremgangsmaader til fremstilling af disseInfo
- Publication number
- DK526989A DK526989A DK526989A DK526989A DK526989A DK 526989 A DK526989 A DK 526989A DK 526989 A DK526989 A DK 526989A DK 526989 A DK526989 A DK 526989A DK 526989 A DK526989 A DK 526989A
- Authority
- DK
- Denmark
- Prior art keywords
- procedure
- nonane
- diazabicyclo
- intermediates
- procedures
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 5
- 239000000543 intermediate Substances 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 2
- XJKNACDCUAFDHD-UHFFFAOYSA-N 1,4-diazabicyclo[3.2.2]nonane Chemical compound C1CC2CCN1CCN2 XJKNACDCUAFDHD-UHFFFAOYSA-N 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- BKIMMITUMNQMOS-UHFFFAOYSA-N nonane Chemical compound CCCCCCCCC BKIMMITUMNQMOS-UHFFFAOYSA-N 0.000 abstract 2
- FTTATHOUSOIFOQ-UHFFFAOYSA-N 1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazine Chemical compound C1NCCN2CCCC21 FTTATHOUSOIFOQ-UHFFFAOYSA-N 0.000 abstract 1
- -1 alkyl stannane Chemical compound 0.000 abstract 1
- XAGFODPZIPBFFR-UHFFFAOYSA-N aluminium Chemical compound [Al] XAGFODPZIPBFFR-UHFFFAOYSA-N 0.000 abstract 1
- 229910052782 aluminium Inorganic materials 0.000 abstract 1
- 229910000080 stannane Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/24—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having more than one carboxyl group bound to the carbon skeleton, e.g. aspartic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/262,542 US4895943A (en) | 1988-10-25 | 1988-10-25 | Preparation of 1,4-diazabicyclo(3.2.2)nonane |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK526989D0 DK526989D0 (da) | 1989-10-24 |
| DK526989A true DK526989A (da) | 1990-04-26 |
Family
ID=22997941
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK526989A DK526989A (da) | 1988-10-25 | 1989-10-24 | Fremgangsmaade til fremstilling af 1,4-diazabicyclo(3.2.2)nonan samt mellemprodukter ved fremgangsmaaden og fremgangsmaader til fremstilling af disse |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4895943A (da) |
| EP (1) | EP0366301B1 (da) |
| JP (1) | JPH0699408B2 (da) |
| KR (1) | KR910007887B1 (da) |
| AT (1) | ATE110724T1 (da) |
| AU (1) | AU616062B2 (da) |
| CA (1) | CA2001211A1 (da) |
| DE (1) | DE68917853T2 (da) |
| DK (1) | DK526989A (da) |
| HU (1) | HU205116B (da) |
| IE (1) | IE893416L (da) |
| IL (1) | IL92025A (da) |
| MY (1) | MY104455A (da) |
| NO (1) | NO172050C (da) |
| NZ (1) | NZ231108A (da) |
| PT (1) | PT92087A (da) |
| ZA (1) | ZA898047B (da) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1997046514A1 (en) * | 1996-05-31 | 1997-12-11 | Novartis Ag | Process for the preparation of hydrazine derivatives useful as intermediates for the preparation of peptide analogues |
| SE0202430D0 (sv) * | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | New Compounds |
| SE0202465D0 (sv) * | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | New compounds |
| CA2499128C (en) | 2002-09-25 | 2012-07-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof |
| ATE363484T1 (de) | 2003-09-26 | 2007-06-15 | Astrazeneca Ab | Nichtamidnonane |
| PL1697378T3 (pl) * | 2003-12-22 | 2008-04-30 | Memory Pharm Corp | Indole, 1h-indazole, 1,2-benzoizoksazole i 1,2-benzoizotiazole oraz ich wytwarzanie i zastosowania |
| WO2005092890A2 (en) | 2004-03-25 | 2005-10-06 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| DE602005024677D1 (de) * | 2004-04-22 | 2010-12-23 | Memory Pharm Corp | Indole, 1h-indazole, 1,2-benzisoxazole, 1,2-benzoisothiazole, deren herstellung und verwendungen |
| RU2386633C2 (ru) * | 2004-05-07 | 2010-04-20 | Мемори Фармасьютиклз Корпорейшн | 1h-индазолы, бензотиазолы, 1, 2-бензоизоксазолы, 1, 2-бензоизотиазолы и хромоны и их получение и применения |
| JP2008525464A (ja) * | 2004-12-22 | 2008-07-17 | メモリー・ファーマシューティカルズ・コーポレイション | α−７ニコチン性受容体リガンド並びにその製造及び使用 |
| US8106066B2 (en) * | 2005-09-23 | 2012-01-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
| CN103450064A (zh) * | 2013-07-30 | 2013-12-18 | 中国科学院上海微系统与信息技术研究所 | 一种芳基乙烯基丙二酰亚胺的制备及伯胺的检测方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3883533A (en) * | 1973-12-27 | 1975-05-13 | Universal Oil Prod Co | Process for preparing 1,4-diazabicyclo octane |
| EP0076089A3 (en) * | 1981-09-28 | 1983-05-25 | Beecham Group Plc | Azabicycloalkane derivatives, process for their preparation, and a pharmaceutical composition containing them |
| US4571396A (en) * | 1984-04-16 | 1986-02-18 | Warner-Lambert Company | Antibacterial agents |
| GB8518236D0 (en) * | 1985-07-19 | 1985-08-29 | Beecham Group Plc | Compounds |
| IN166416B (da) * | 1985-09-18 | 1990-05-05 | Pfizer |
-
1988
- 1988-10-25 US US07/262,542 patent/US4895943A/en not_active Expired - Fee Related
-
1989
- 1989-10-11 EP EP89310389A patent/EP0366301B1/en not_active Expired - Lifetime
- 1989-10-11 DE DE68917853T patent/DE68917853T2/de not_active Expired - Fee Related
- 1989-10-11 AT AT89310389T patent/ATE110724T1/de not_active IP Right Cessation
- 1989-10-17 IL IL9202589A patent/IL92025A/en not_active IP Right Cessation
- 1989-10-23 CA CA002001211A patent/CA2001211A1/en not_active Abandoned
- 1989-10-23 MY MYPI89001469A patent/MY104455A/en unknown
- 1989-10-24 NO NO894230A patent/NO172050C/no unknown
- 1989-10-24 HU HU895422A patent/HU205116B/hu not_active IP Right Cessation
- 1989-10-24 PT PT92087A patent/PT92087A/pt unknown
- 1989-10-24 ZA ZA898047A patent/ZA898047B/xx unknown
- 1989-10-24 IE IE893416A patent/IE893416L/xx unknown
- 1989-10-24 DK DK526989A patent/DK526989A/da not_active Application Discontinuation
- 1989-10-24 AU AU43700/89A patent/AU616062B2/en not_active Ceased
- 1989-10-24 NZ NZ231108A patent/NZ231108A/en unknown
- 1989-10-24 KR KR1019890015276A patent/KR910007887B1/ko not_active Expired
- 1989-10-25 JP JP1278301A patent/JPH0699408B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| US4895943A (en) | 1990-01-23 |
| NO172050C (no) | 1993-06-02 |
| ZA898047B (en) | 1991-06-26 |
| NO894230L (no) | 1990-04-26 |
| DE68917853T2 (de) | 1995-01-12 |
| EP0366301A3 (en) | 1991-07-31 |
| KR900006301A (ko) | 1990-05-07 |
| HUT54366A (en) | 1991-02-28 |
| EP0366301A2 (en) | 1990-05-02 |
| IL92025A (en) | 1994-10-07 |
| ATE110724T1 (de) | 1994-09-15 |
| AU616062B2 (en) | 1991-10-17 |
| DK526989D0 (da) | 1989-10-24 |
| EP0366301B1 (en) | 1994-08-31 |
| PT92087A (pt) | 1990-04-30 |
| HU895422D0 (en) | 1990-01-28 |
| MY104455A (en) | 1994-03-31 |
| HU205116B (en) | 1992-03-30 |
| IL92025A0 (en) | 1990-07-12 |
| NO172050B (no) | 1993-02-22 |
| JPH02174769A (ja) | 1990-07-06 |
| CA2001211A1 (en) | 1990-04-25 |
| IE893416L (en) | 1990-04-25 |
| AU4370089A (en) | 1990-05-03 |
| NZ231108A (en) | 1992-03-26 |
| KR910007887B1 (ko) | 1991-10-04 |
| JPH0699408B2 (ja) | 1994-12-07 |
| DE68917853D1 (de) | 1994-10-06 |
| NO894230D0 (no) | 1989-10-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |