DK540278A - Fremgangsmaade til fremstilling af cephalosporiner - Google Patents

Fremgangsmaade til fremstilling af cephalosporiner

Info

Publication number: DK540278A
Authority: DK; Denmark
Prior art keywords: cephalosporins; procedure; preparation
Prior art date: 1977-12-20

Application number

DK540278A

Other languages

Danish (da)

English (en)

Inventor

A S Katner

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-12-20

Filing date

1978-11-30

Publication date

1979-06-21

1978-11-30 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1979-06-21 Publication of DK540278A publication Critical patent/DK540278A/da

Links

229930186147 Cephalosporin Natural products 0.000 title 1
229940124587 cephalosporin Drugs 0.000 title 1
HOKIDJSKDBPKTQ-GLXFQSAKSA-N cephalosporin C Chemical compound S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)[C@@H](NC(=O)CCC[C@@H](N)C(O)=O)[C@@H]12 HOKIDJSKDBPKTQ-GLXFQSAKSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK540278A 1977-12-20 1978-11-30 Fremgangsmaade til fremstilling af cephalosporiner DK540278A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US05/862,318 US4200745A (en)	1977-12-20	1977-12-20	7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins

Publications (1)

Publication Number	Publication Date
DK540278A true DK540278A (da)	1979-06-21

Family

ID=25338200

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK540278A DK540278A (da)	1977-12-20	1978-11-30	Fremgangsmaade til fremstilling af cephalosporiner

Country Status (33)

Country	Link
US (1)	US4200745A (de)
EP (1)	EP0002605B1 (de)
JP (1)	JPS5490194A (de)
AR (1)	AR220733A1 (de)
AT (1)	AT364189B (de)
AU (1)	AU518484B2 (de)
BE (1)	BE872616A (de)
CA (1)	CA1140112A (de)
CH (1)	CH635846A5 (de)
CS (1)	CS204957B2 (de)
DD (1)	DD139857A5 (de)
DE (1)	DE2861493D1 (de)
DK (1)	DK540278A (de)
EG (1)	EG13666A (de)
ES (1)	ES476154A1 (de)
FI (1)	FI67083C (de)
FR (1)	FR2412553A1 (de)
GB (1)	GB2010256B (de)
GR (1)	GR72240B (de)
HU (1)	HU181875B (de)
IE (1)	IE47696B1 (de)
IL (1)	IL56166A0 (de)
IT (1)	IT1112300B (de)
LU (1)	LU80669A1 (de)
MX (1)	MX5586E (de)
NZ (1)	NZ189121A (de)
PH (1)	PH15368A (de)
PL (1)	PL123368B1 (de)
PT (1)	PT68888A (de)
RO (1)	RO75804A (de)
SU (1)	SU793403A3 (de)
YU (1)	YU300278A (de)
ZA (1)	ZA787110B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5760345B2 (de) *	1974-12-19	1982-12-18	Takeda Chemical Industries Ltd
CH641468A5 (de) *	1978-05-30	1984-02-29	Hoffmann La Roche	Cephemderivate.
MC1259A1 (fr) *	1978-05-30	1980-01-14	Hoffmann La Roche	Derives acyles
ZA806977B (en) *	1979-11-19	1981-10-28	Fujisawa Pharmaceutical Co	7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
FI67385C (fi) *	1979-11-21	1985-03-11	Hoffmann La Roche	Foerfarande foer framstaellning av (6r 7r)-7-(2-(2-amino-4-tiazolyl)-2-(z-metoxiimino)acetamido)-3-cefem-4-karboxylsyraderivat
US4349672A (en) *	1979-11-29	1982-09-14	Hoffmann-La Roche Inc.	Cephalosporin derivatives
US4409387A (en) *	1979-11-29	1983-10-11	Hoffmann-La Roche Inc.	Cephalosporin derivatives
NZ196552A (en) *	1980-03-25	1984-07-06	Hoffmann La Roche	Cephalosporin derivatives and pharmaceutical compositions;intermediate cephalosporins
GR75706B (de) *	1980-06-30	1984-08-02	Sanofi Sa
DK379581A (da) *	1980-10-06	1982-04-07	Hoffmann La Roche	Fremgangsmaade til fremstilling af acylderivater
FR2494278A1 (fr) *	1980-11-20	1982-05-21	Rhone Poulenc Ind	Nouveaux derives de la cephalosporine, leurs preparations et les medicaments qui les contiennent
US4698338A (en) *	1986-02-19	1987-10-06	Eli Lilly And Company	7[2-(2-aminothiazol-4-yl)-2-benzyloximino]acetamido-3[4-alkyl-5-oxo-6-hydroxy-3,4-dihydro-1,2,4-triazin-3-yl]thiomethyl cephalosporins

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RO67533B (ro)	1974-08-02	1984-03-30	Eli Lilly And Company	Procedeu pentru prepararea unor derivati de 3-triaziniltiometilcefalosporina
CA1100129A (en) *	1974-08-02	1981-04-28	William H.W. Lunn	Cephalosporin compounds
FR2345153A1 (fr)	1976-03-25	1977-10-21	Roussel Uclaf	Nouvelles alcoyloximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
DE2760484C2 (de) *	1976-04-14	1992-12-03	Takeda Chemical Industries, Ltd., Osaka, Jp
NL7805715A (nl) *	1977-06-03	1978-12-05	Hoffmann La Roche	Werkwijze voor het bereiden van acylderivaten.

1977
- 1977-12-20 US US05/862,318 patent/US4200745A/en not_active Expired - Lifetime
1978
- 1978-11-30 DK DK540278A patent/DK540278A/da not_active Application Discontinuation
- 1978-12-07 PT PT68888A patent/PT68888A/pt unknown
- 1978-12-07 AR AR274724A patent/AR220733A1/es active
- 1978-12-07 NZ NZ189121A patent/NZ189121A/en unknown
- 1978-12-07 PH PH21906A patent/PH15368A/en unknown
- 1978-12-08 AU AU42347/78A patent/AU518484B2/en not_active Expired
- 1978-12-08 FR FR7834608A patent/FR2412553A1/fr active Granted
- 1978-12-08 BE BE1009182A patent/BE872616A/xx not_active IP Right Cessation
- 1978-12-10 IL IL56166A patent/IL56166A0/xx unknown
- 1978-12-11 MX MX787582U patent/MX5586E/es unknown
- 1978-12-11 GR GR57837A patent/GR72240B/el unknown
- 1978-12-13 GB GB7848211A patent/GB2010256B/en not_active Expired
- 1978-12-13 CA CA000317875A patent/CA1140112A/en not_active Expired
- 1978-12-13 DE DE7878300801T patent/DE2861493D1/de not_active Expired
- 1978-12-13 SU SU782699098A patent/SU793403A3/ru active
- 1978-12-13 EP EP78300801A patent/EP0002605B1/de not_active Expired
- 1978-12-14 FI FI783846A patent/FI67083C/fi not_active IP Right Cessation
- 1978-12-18 JP JP15810078A patent/JPS5490194A/ja active Pending
- 1978-12-18 LU LU80669A patent/LU80669A1/xx unknown
- 1978-12-18 CS CS788518A patent/CS204957B2/cs unknown
- 1978-12-19 AT AT0908378A patent/AT364189B/de not_active IP Right Cessation
- 1978-12-19 HU HU78EI830A patent/HU181875B/hu unknown
- 1978-12-19 ZA ZA787110A patent/ZA787110B/xx unknown
- 1978-12-19 IE IE2502/78A patent/IE47696B1/en unknown
- 1978-12-19 ES ES476154A patent/ES476154A1/es not_active Expired
- 1978-12-19 RO RO7895973A patent/RO75804A/ro unknown
- 1978-12-19 CH CH1295478A patent/CH635846A5/fr not_active IP Right Cessation
- 1978-12-19 EG EG712/78A patent/EG13666A/xx active
- 1978-12-19 IT IT31016/78A patent/IT1112300B/it active
- 1978-12-20 PL PL1978211973A patent/PL123368B1/pl unknown
- 1978-12-20 DD DD78209940A patent/DD139857A5/de unknown
- 1978-12-20 YU YU03002/78A patent/YU300278A/xx unknown

Also Published As

Publication number	Publication date
AU4234778A (en)	1979-06-28
FR2412553A1 (fr)	1979-07-20
RO75804A (ro)	1981-02-28
AR220733A1 (es)	1980-11-28
MX5586E (es)	1983-10-28
PL211973A1 (de)	1980-03-10
CA1140112A (en)	1983-01-25
PT68888A (en)	1979-01-01
EG13666A (en)	1983-12-31
CS204957B2 (en)	1981-04-30
IE782502L (en)	1979-06-20
SU793403A3 (ru)	1980-12-30
FI67083B (fi)	1984-09-28
YU300278A (en)	1982-10-31
IT7831016A0 (it)	1978-12-19
US4200745A (en)	1980-04-29
ATA908378A (de)	1981-02-15
DE2861493D1 (en)	1982-02-18
PH15368A (en)	1982-12-10
IE47696B1 (en)	1984-05-30
BE872616A (fr)	1979-06-08
DD139857A5 (de)	1980-01-23
ES476154A1 (es)	1980-05-16
FI67083C (fi)	1985-01-10
FR2412553B1 (de)	1982-10-15
ZA787110B (en)	1980-08-27
GR72240B (de)	1983-10-03
FI783846A7 (fi)	1979-06-21
GB2010256A (en)	1979-06-27
NZ189121A (en)	1984-02-03
IL56166A0 (en)	1979-03-12
IT1112300B (it)	1986-01-13
AU518484B2 (en)	1981-10-01
CH635846A5 (fr)	1983-04-29
JPS5490194A (en)	1979-07-17
GB2010256B (en)	1982-09-08
LU80669A1 (fr)	1979-04-13
AT364189B (de)	1981-09-25
EP0002605B1 (de)	1981-12-30
EP0002605A1 (de)	1979-06-27
HU181875B (en)	1983-11-28
PL123368B1 (en)	1982-10-30

Legal Events

Date	Code	Title	Description
1985-10-28	ATS	Application withdrawn

Publication	Publication Date	Title
DK552180A (da)	1981-06-28	Fremgangsmaade til fremstilling af tetrapeptidsemikarbazidderivater
DK110778A (da)	1978-09-15	Fremgangsmaade til fremstilling af 4-acylamino-phenyl-ethanolaminer
DK306978A (da)	1979-01-12	Fremgangsmaade til fremstilling af 1-acyl-2-cyanaziridiner
DK484677A (da)	1979-04-04	Fremgangsmaade til fremstilling af furokumariner
DK569678A (da)	1979-06-21	Fremgangsmaade til fremstilling af 2alfa-cyano-3-oxosteroider
DK168778A (da)	1978-10-20	Fremgangsmaade til fremstilling af cephalosporiner
DK145701C (da)	1983-07-18	Fremgangsmaade til fremstilling af ergotalkaloider
DK146578A (da)	1978-10-05	Fremgangsmaade til fremstilling af interphenylen 8-aza-9-dioxothia-11%12-secoprostaglandiner
DK466878A (da)	1979-04-21	Fremgangsmaade til fremstilling af 0-methallyloxyphenol
DK398078A (da)	1979-03-09	Fremgangsmaade til fremstilling af sulfonylamidinforbindelser
DK91277A (da)	1977-09-04	Fremgangsmade til fremstilling af cephalosporiner
DK237978A (da)	1979-01-19	Fremgangsmaade til fremstilling af alfafluormethyl-alfa-aminoalkansyrer
DK154949C (da)	1989-05-29	Fremgangsmaade til fremstilling af trifluormethylphenoler
DK436978A (da)	1979-04-05	Fremgangsmaade til fremstilling af sarcosinoxidase
DK226678A (da)	1978-11-24	Fremgangsmaade til fremstilling af hexahydrogamma-carbolinforbindelser
DK5778A (da)	1978-07-12	Femgangsmaade til fremstilling af 4-diphenylmethylen-1-hydroxybenzyl-piperidiner
DK577078A (da)	1979-06-28	Fremgangsmaade til fremstilling af trans-4a-aryloctahydro-1h-2-pyridiner
DK97378A (da)	1978-09-08	Fremgangsmaade til fremstilling af cephalosporiner
DK364578A (da)	1979-02-19	Fremgangsmaade til fremstilling af hydroxyphenylhydantoin
DK248978A (da)	1978-12-05	Fremgangsmaade til fremstilling af hydroxy-alfa-aminobenzylpenicillin
DK246878A (da)	1978-12-04	Fremgangsmaade til fremstilling af acylderivater
DK383978A (da)	1979-03-02	Fremgangsmaade til fremstilling af 2-chlorsulfinylazetidin-4-oner
DK339777A (da)	1978-10-30	Fremgangsmaade til fremstilling af 2-benzylperhydroazepiner
DK158976C (da)	1990-12-31	Fremgangsmaade til fremstilling af alfa-cyanobenzyl
DK206178A (da)	1978-11-12	Fremgangsmaade til fremstilling af 3-bromphthalid