DK543088D0 - Substituerede alkylamider af teicoplaninforbindelser - Google Patents

Substituerede alkylamider af teicoplaninforbindelser

Info

Publication number: DK543088D0
Authority: DK; Denmark
Prior art keywords: teicoplane; compounds; substituted alkylamides; substituted; alkylamides
Prior art date: 1987-03-02

Application number

DK543088A

Other languages

English (en)

Other versions

DK543088A (da

Inventor

Adriano Malabarba

Giorgio Tarzia

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-03-02

Filing date

1988-09-29

Publication date

1988-09-29

1988-09-29 Application filed by Lepetit Spa filed Critical Lepetit Spa

1988-09-29 Publication of DK543088A publication Critical patent/DK543088A/da

1988-09-29 Publication of DK543088D0 publication Critical patent/DK543088D0/da

Links

150000001875 compounds Chemical class 0.000 title 1
DQJCDTNMLBYVAY-ZXXIYAEKSA-N (2S,5R,10R,13R)-16-{[(2R,3S,4R,5R)-3-{[(2S,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-5-(ethylamino)-6-hydroxy-2-(hydroxymethyl)oxan-4-yl]oxy}-5-(4-aminobutyl)-10-carbamoyl-2,13-dimethyl-4,7,12,15-tetraoxo-3,6,11,14-tetraazaheptadecan-1-oic acid Chemical group NCCCC[C@H](C(=O)N[C@@H](C)C(O)=O)NC(=O)CC[C@H](C(N)=O)NC(=O)[C@@H](C)NC(=O)C(C)O[C@@H]1[C@@H](NCC)C(O)O[C@H](CO)[C@H]1O[C@H]1[C@H](NC(C)=O)[C@@H](O)[C@H](O)[C@@H](CO)O1 DQJCDTNMLBYVAY-ZXXIYAEKSA-N 0.000 abstract 1
DDTDNCYHLGRFBM-YZEKDTGTSA-N chembl2367892 Chemical class CC(=O)N[C@H]1[C@@H](O)[C@H](O)[C@H](CO)O[C@H]1O[C@@H]([C@H]1C(N[C@@H](C2=CC(O)=CC(O[C@@H]3[C@H]([C@H](O)[C@H](O)[C@@H](CO)O3)O)=C2C=2C(O)=CC=C(C=2)[C@@H](NC(=O)[C@@H]2NC(=O)[C@@H]3C=4C=C(O)C=C(C=4)OC=4C(O)=CC=C(C=4)[C@@H](N)C(=O)N[C@H](CC=4C=C(Cl)C(O5)=CC=4)C(=O)N3)C(=O)N1)C(O)=O)=O)C(C=C1Cl)=CC=C1OC1=C(O[C@H]3[C@H]([C@@H](O)[C@H](O)[C@H](CO)O3)NC(C)=O)C5=CC2=C1 DDTDNCYHLGRFBM-YZEKDTGTSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Peptides Or Proteins (AREA)
Luminescent Compositions (AREA)
Polyamides (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)

DK543088A 1987-03-02 1988-09-29 Substituerede alkylamider af teicoplaninforbindelser DK543088D0 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB878704847A GB8704847D0 (en)	1987-03-02	1987-03-02	Substituted alkylamides of teicoplanin compounds
PCT/EP1988/000129 WO1988006600A1 (en)	1987-03-02	1988-02-23	Substituted alkylamides of teicoplanin compounds

Publications (2)

Publication Number	Publication Date
DK543088A DK543088A (da)	1988-09-29
DK543088D0 true DK543088D0 (da)	1988-09-29

Family

ID=10613186

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK543088A DK543088D0 (da)	1987-03-02	1988-09-29	Substituerede alkylamider af teicoplaninforbindelser

Country Status (22)

Country	Link
US (1)	US5198418A (da)
EP (1)	EP0340245B1 (da)
JP (1)	JPH0776234B2 (da)
KR (1)	KR960014104B1 (da)
CN (1)	CN88101000A (da)
AT (1)	ATE79637T1 (da)
AU (1)	AU619460B2 (da)
DE (1)	DE3873907T2 (da)
DK (1)	DK543088D0 (da)
ES (1)	ES2009555A6 (da)
FI (1)	FI91765C (da)
GB (1)	GB8704847D0 (da)
GR (1)	GR1001625B (da)
HU (1)	HU205371B (da)
IE (1)	IE62860B1 (da)
IL (1)	IL85493A0 (da)
NO (1)	NO176568C (da)
NZ (1)	NZ223669A (da)
PH (1)	PH27406A (da)
PT (1)	PT86827B (da)
WO (1)	WO1988006600A1 (da)
ZA (1)	ZA881445B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds
GB8827202D0 (en) *	1988-11-22	1988-12-29	Lepetit Spa	Process for preparing 63-carboxyamides of teicoplanin antibiotics
ATE134646T1 (de) *	1988-12-27	1996-03-15	Lepetit Spa	C63-amidderivate von 34-de(acetylglucosaminyl)-34-deoxy-teicoplanine
IE64155B1 (en) *	1989-03-29	1995-07-12	Lepetit Spa	New substituted alkylamide derivatives of teicoplanin
US5500410A (en) *	1989-03-29	1996-03-19	Gruppo Lepetit S.P.A.	Substituted alkylamide derivatives of teicoplanin
US5185320A (en) *	1989-04-03	1993-02-09	Gruppo Lepetit S.P.A.	O56 -alkyl derivatives of aglycone and pseudo aglycones of teicoplanin
EP0391077A1 (en) *	1989-04-03	1990-10-10	GRUPPO LEPETIT S.p.A.	O56-alkyl derivatives of aglycone and pseudoaglycones of teicoplanin
AU647122B2 (en) *	1990-05-28	1994-03-17	Gruppo Lepetit S.P.A.	C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy- teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
WO1992010516A1 (en) *	1990-12-05	1992-06-25	Gruppo Lepetit S.P.A.	38-decarboxy-38-hydroxymethyl derivatives of teicoplanin antibiotics, and a process for preparing them
ATE173022T1 (de) *	1991-08-08	1998-11-15	Amylin Pharmaceuticals Inc	Produktion von peptid-amiden
GB2278540A (en) *	1993-09-24	1994-12-07	Nick Andrew Lewis	Extendible garment hanger
US5679769A (en) *	1994-03-15	1997-10-21	Sloan-Kettering Institute For Cancer Research	Synthesis of asparagine-linked glycopeptides on a polymeric solid support
KR20000010589A (ko)	1996-04-23	2000-02-15	클라우디오 쿼르타	항생제a40926의아미드유도체의개선된화학적제조방법
MY123217A (en) *	1998-12-23	2006-05-31	Theravance Inc	Glycopeptide derivatives and pharmaceutical compositions containing the same
DE69908819T2 (de) *	1998-12-23	2004-05-06	Theravance, Inc., South San Francisco	Glycopeptid-derivate und pharmazeutische zusammensetzungen, die sie enthalten
US6770621B2 (en)	2000-05-02	2004-08-03	Theravance, Inc.	Polyacid glycopeptide derivatives

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3981303A (en) *	1971-09-09	1976-09-21	Alza Corporation	Bioerodible ocular device
GB1496386A (en) *	1975-03-05	1977-12-30	Lepetit Spa	Antibiotics
US4604239A (en) *	1982-03-24	1986-08-05	Eli Lilly And Company	Antibiotics
GB8307847D0 (en) *	1983-03-22	1983-04-27	Lepetit Spa	Antibiotics l 17054 and l 17046
US4534969A (en) *	1983-09-19	1985-08-13	The Dow Chemical Company	Method for improving lactation in ruminant animals
AU579120B2 (en) *	1983-12-16	1988-11-17	Gruppo Lepetit S.P.A.	Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
IT1173329B (it) *	1984-02-21	1987-06-24	Lepetit Spa	Procedimento per la trasformazione quantitativa di teicoplanina a2 fattore 1 in teicoplanina a2 fattore 3
GB8415092D0 (en) *	1984-06-13	1984-07-18	Lepetit Spa	Ester derivatives
GB8420405D0 (en) *	1984-08-10	1984-09-12	Lepetit Spa	Preparing antibiotic l 17046
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds

1987
- 1987-03-02 GB GB878704847A patent/GB8704847D0/en active Pending
1988
- 1988-02-22 IL IL85493A patent/IL85493A0/xx not_active IP Right Cessation
- 1988-02-23 AT AT88902122T patent/ATE79637T1/de not_active IP Right Cessation
- 1988-02-23 HU HU881742A patent/HU205371B/hu not_active IP Right Cessation
- 1988-02-23 WO PCT/EP1988/000129 patent/WO1988006600A1/en not_active Ceased
- 1988-02-23 AU AU13632/88A patent/AU619460B2/en not_active Ceased
- 1988-02-23 DE DE8888902122T patent/DE3873907T2/de not_active Expired - Fee Related
- 1988-02-23 KR KR1019880701400A patent/KR960014104B1/ko not_active Expired - Lifetime
- 1988-02-23 JP JP63501993A patent/JPH0776234B2/ja not_active Expired - Lifetime
- 1988-02-23 EP EP88902122A patent/EP0340245B1/en not_active Expired - Lifetime
- 1988-02-25 PT PT86827A patent/PT86827B/pt not_active IP Right Cessation
- 1988-02-25 IE IE51388A patent/IE62860B1/en not_active IP Right Cessation
- 1988-02-26 NZ NZ223669A patent/NZ223669A/en unknown
- 1988-02-29 CN CN198888101000A patent/CN88101000A/zh active Pending
- 1988-03-01 ES ES8800594A patent/ES2009555A6/es not_active Expired
- 1988-03-01 ZA ZA881445A patent/ZA881445B/xx unknown
- 1988-03-01 GR GR880100118A patent/GR1001625B/el unknown
- 1988-03-02 PH PH36578A patent/PH27406A/en unknown
- 1988-09-29 DK DK543088A patent/DK543088D0/da not_active Application Discontinuation
- 1988-10-28 NO NO884821A patent/NO176568C/no unknown
1989
- 1989-08-31 FI FI894078A patent/FI91765C/fi not_active IP Right Cessation
1992
- 1992-01-21 US US07/826,198 patent/US5198418A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
NZ223669A (en)	1990-12-21
IE880513L (en)	1988-09-02
CN88101000A (zh)	1988-09-14
DE3873907T2 (de)	1993-01-14
JPH0776234B2 (ja)	1995-08-16
FI91765C (fi)	1994-08-10
FI894078L (fi)	1989-08-31
JPH02502456A (ja)	1990-08-09
NO176568C (no)	1995-04-26
HU205371B (en)	1992-04-28
HUT51300A (en)	1990-04-28
ES2009555A6 (es)	1989-10-01
ZA881445B (en)	1989-01-25
GR880100118A (en)	1989-01-31
DE3873907D1 (de)	1992-09-24
NO884821D0 (no)	1988-10-28
FI894078A0 (fi)	1989-08-31
AU619460B2 (en)	1992-01-30
KR890700607A (ko)	1989-04-26
EP0340245A1 (en)	1989-11-08
ATE79637T1 (de)	1992-09-15
PH27406A (en)	1993-06-21
NO176568B (no)	1995-01-16
DK543088A (da)	1988-09-29
FI91765B (fi)	1994-04-29
IE62860B1 (en)	1995-03-08
IL85493A0 (en)	1988-07-31
AU1363288A (en)	1988-09-26
PT86827B (pt)	1992-05-29
KR960014104B1 (ko)	1996-10-14
GR1001625B (el)	1994-07-29
NO884821L (no)	1988-10-28
PT86827A (pt)	1988-03-01
WO1988006600A1 (en)	1988-09-07
GB8704847D0 (en)	1987-04-08
US5198418A (en)	1993-03-30
EP0340245B1 (en)	1992-08-19

Legal Events

Date	Code	Title	Description
1997-10-20	AHS	Application shelved for other reasons than non-payment

Publication	Publication Date	Title
DK543088A (da)	1988-09-29	Substituerede alkylamider af teicoplaninforbindelser
ATE219938T1 (de)	2002-07-15	Neue 4-arylpiperazine und 4-arylpiperidine
DE69227407D1 (de)	1998-12-03	Superlumineszierende optische Quelle
FI922181L (fi)	1992-12-01	Oeverdragna tuggummiprodukter polerade med faergat vax
BR8801609A (pt)	1989-02-08	Conjunto de farol substituivel
DE69221635D1 (de)	1997-09-18	Neue tabakersatzstoffe
DE69207568D1 (de)	1996-02-22	Schutzbalg
FI930962A0 (fi)	1993-03-04	Anordning foer registrering av den malbara laddningens maengd i ett visst oegonblick i en malningstrumma
NO924126D0 (no)	1992-10-23	3-indolylthioacetatderivater
DK0465481T3 (da)	1994-02-21	Substituerede alkylamidderivater af teicoplanin
FI892222A0 (fi)	1989-05-09	Peptidalkoholer med antikoagulantverkan.
IT9019323A0 (it)	1990-02-09	Procedimento di preparazione di l-a-glicerilfosforil-d-myoinositolo e suoi sali da fosfatidi grezzi o parzialmente purificati
DE69132871D1 (de)	2002-01-31	Copolyetherester-Formmassen
MX9102079A (es)	1993-01-01	Plemezcla de semduramicina
FI930411A0 (fi)	1993-01-29	Bombesin antagonister
DK316589D0 (da)	1989-06-26	Substituerede azacyclohexylderivater af rifamyciner
FI923287L (fi)	1993-01-21	Kabeldragningsanordning med aotminstone ett kabeldragningsroer
PT87378A (pt)	1989-05-31	Neue 2-aminoalkyl-4-benzyl-1-(2h)-phthalazinon-derivate
BR8807123A (pt)	1989-10-17	Lanterna de projecao catadioptrica
DE69115750D1 (de)	1996-02-08	Neue Nojirimycinderivate
ATA125290A (de)	1994-02-15	Gliederkessel
FI924327L (fi)	1993-02-13	Ett skivformat byggelement med skydds-, ventilations-, vaermeisolerings- och torkverkan
KR920013544U (ko)	1992-07-27	스위치의 고정장치
SE9003608D0 (sv)	1990-11-13	Magnetlampa
BR7001700U (pt)	1992-03-17	Controle de filas-fila livre