ATE79637T1 - Substituierte alkylamide von teicoplaninverbindungen. - Google Patents

Substituierte alkylamide von teicoplaninverbindungen.

Info

Publication number: ATE79637T1
Authority: AT; Austria
Prior art keywords: alkylamides; substitute; teicoplanin compounds; teicoplanin; compounds
Prior art date: 1987-03-02

Application number

AT88902122T

Other languages

English (en)

Inventor

Adriano Malabarba

Giorgio Tarzia

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-03-02

Filing date

1988-02-23

Publication date

1992-09-15

1988-02-23 Application filed by Lepetit Spa filed Critical Lepetit Spa

1992-09-15 Application granted granted Critical

1992-09-15 Publication of ATE79637T1 publication Critical patent/ATE79637T1/de

Links

YMWQIYMUNZBOOV-AQQDCCNYSA-N hms2094o05 Chemical class CCCCC\C=C\CCC(=O)N[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1OC(C(=C1)OC=2C(=CC(=CC=2)[C@@H](O[C@H]2[C@@H]([C@@H](O)[C@H](O)[C@@H](CO)O2)NC(C)=O)[C@H]2C(N[C@@H](C3=CC(O)=CC(OC4[C@H]([C@@H](O)[C@H](O)[C@@H](CO)O4)O)=C3C=3C(O)=CC=C(C=3)[C@@H](NC3=O)C(=O)N2)C(O)=O)=O)Cl)=C(OC=2C(=CC(CC(C(N4)=O)NC(=O)[C@H](N)C=5C=C(O6)C(O)=CC=5)=CC=2)Cl)C=C1[C@H]3NC(=O)[C@@H]4C1=CC6=CC(O)=C1 YMWQIYMUNZBOOV-AQQDCCNYSA-N 0.000 title 1
DQJCDTNMLBYVAY-ZXXIYAEKSA-N (2S,5R,10R,13R)-16-{[(2R,3S,4R,5R)-3-{[(2S,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-5-(ethylamino)-6-hydroxy-2-(hydroxymethyl)oxan-4-yl]oxy}-5-(4-aminobutyl)-10-carbamoyl-2,13-dimethyl-4,7,12,15-tetraoxo-3,6,11,14-tetraazaheptadecan-1-oic acid Chemical group NCCCC[C@H](C(=O)N[C@@H](C)C(O)=O)NC(=O)CC[C@H](C(N)=O)NC(=O)[C@@H](C)NC(=O)C(C)O[C@@H]1[C@@H](NCC)C(O)O[C@H](CO)[C@H]1O[C@H]1[C@H](NC(C)=O)[C@@H](O)[C@H](O)[C@@H](CO)O1 DQJCDTNMLBYVAY-ZXXIYAEKSA-N 0.000 abstract 1
DDTDNCYHLGRFBM-YZEKDTGTSA-N chembl2367892 Chemical class CC(=O)N[C@H]1[C@@H](O)[C@H](O)[C@H](CO)O[C@H]1O[C@@H]([C@H]1C(N[C@@H](C2=CC(O)=CC(O[C@@H]3[C@H]([C@H](O)[C@H](O)[C@@H](CO)O3)O)=C2C=2C(O)=CC=C(C=2)[C@@H](NC(=O)[C@@H]2NC(=O)[C@@H]3C=4C=C(O)C=C(C=4)OC=4C(O)=CC=C(C=4)[C@@H](N)C(=O)N[C@H](CC=4C=C(Cl)C(O5)=CC=4)C(=O)N3)C(=O)N1)C(O)=O)=O)C(C=C1Cl)=CC=C1OC1=C(O[C@H]3[C@H]([C@@H](O)[C@H](O)[C@H](CO)O3)NC(C)=O)C5=CC2=C1 DDTDNCYHLGRFBM-YZEKDTGTSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Luminescent Compositions (AREA)
Peptides Or Proteins (AREA)
Polyamides (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)

AT88902122T 1987-03-02 1988-02-23 Substituierte alkylamide von teicoplaninverbindungen. ATE79637T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB878704847A GB8704847D0 (en)	1987-03-02	1987-03-02	Substituted alkylamides of teicoplanin compounds
PCT/EP1988/000129 WO1988006600A1 (en)	1987-03-02	1988-02-23	Substituted alkylamides of teicoplanin compounds
EP88902122A EP0340245B1 (de)	1987-03-02	1988-02-23	Substituierte alkylamide von teicoplanin-verbindungen

Publications (1)

Publication Number	Publication Date
ATE79637T1 true ATE79637T1 (de)	1992-09-15

Family

ID=10613186

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT88902122T ATE79637T1 (de)	1987-03-02	1988-02-23	Substituierte alkylamide von teicoplaninverbindungen.

Country Status (22)

Country	Link
US (1)	US5198418A (de)
EP (1)	EP0340245B1 (de)
JP (1)	JPH0776234B2 (de)
KR (1)	KR960014104B1 (de)
CN (1)	CN88101000A (de)
AT (1)	ATE79637T1 (de)
AU (1)	AU619460B2 (de)
DE (1)	DE3873907T2 (de)
DK (1)	DK543088A (de)
ES (1)	ES2009555A6 (de)
FI (1)	FI91765C (de)
GB (1)	GB8704847D0 (de)
GR (1)	GR1001625B (de)
HU (1)	HU205371B (de)
IE (1)	IE62860B1 (de)
IL (1)	IL85493A0 (de)
NO (1)	NO176568C (de)
NZ (1)	NZ223669A (de)
PH (1)	PH27406A (de)
PT (1)	PT86827B (de)
WO (1)	WO1988006600A1 (de)
ZA (1)	ZA881445B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds
GB8827202D0 (en) *	1988-11-22	1988-12-29	Lepetit Spa	Process for preparing 63-carboxyamides of teicoplanin antibiotics
EP0376041B1 (de) *	1988-12-27	1996-02-28	GRUPPO LEPETIT S.p.A.	C63-Amidderivate von 34-de(acetylglucosaminyl)-34-deoxy-teicoplaninen
IE64155B1 (en) *	1989-03-29	1995-07-12	Lepetit Spa	New substituted alkylamide derivatives of teicoplanin
US5500410A (en) *	1989-03-29	1996-03-19	Gruppo Lepetit S.P.A.	Substituted alkylamide derivatives of teicoplanin
EP0391077A1 (de) *	1989-04-03	1990-10-10	GRUPPO LEPETIT S.p.A.	O56-Alkyl-Derivate von Aglycon und Pseudoaglycone von Teicoplanin
US5185320A (en) *	1989-04-03	1993-02-09	Gruppo Lepetit S.P.A.	O56 -alkyl derivatives of aglycone and pseudo aglycones of teicoplanin
AU647122B2 (en) *	1990-05-28	1994-03-17	Gruppo Lepetit S.P.A.	C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy- teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
WO1992010516A1 (en) *	1990-12-05	1992-06-25	Gruppo Lepetit S.P.A.	38-decarboxy-38-hydroxymethyl derivatives of teicoplanin antibiotics, and a process for preparing them
WO1993002697A1 (en) *	1991-08-08	1993-02-18	Amylin Pharmaceuticals, Inc.	Production of peptide amides
GB2278540A (en) *	1993-09-24	1994-12-07	Nick Andrew Lewis	Extendible garment hanger
US5679769A (en) *	1994-03-15	1997-10-21	Sloan-Kettering Institute For Cancer Research	Synthesis of asparagine-linked glycopeptides on a polymeric solid support
EP0912604B1 (de)	1996-04-23	2001-11-14	Biosearch Italia S.p.A.	Chemisches Verfahren zur Herstellung von Amidderivaten von A 40926 Antibiotikum
PT1140993E (pt)	1998-12-23	2003-10-31	Theravance Inc	Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos
SG87877A1 (en) *	1998-12-23	2002-04-16	Advanced Medicine Inc	Glycopeptide derivatives and pharmaceutical compositions containing the same
AU2001259298A1 (en)	2000-05-02	2001-11-12	Advanced Medicine, Inc.	Polyacid glycopeptide derivatives

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3981303A (en) *	1971-09-09	1976-09-21	Alza Corporation	Bioerodible ocular device
GB1496386A (en) *	1975-03-05	1977-12-30	Lepetit Spa	Antibiotics
US4604239A (en) *	1982-03-24	1986-08-05	Eli Lilly And Company	Antibiotics
GB8307847D0 (en) *	1983-03-22	1983-04-27	Lepetit Spa	Antibiotics l 17054 and l 17046
US4534969A (en) *	1983-09-19	1985-08-13	The Dow Chemical Company	Method for improving lactation in ruminant animals
AU579120B2 (en) *	1983-12-16	1988-11-17	Gruppo Lepetit S.P.A.	Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
IT1173329B (it) *	1984-02-21	1987-06-24	Lepetit Spa	Procedimento per la trasformazione quantitativa di teicoplanina a2 fattore 1 in teicoplanina a2 fattore 3
GB8415092D0 (en) *	1984-06-13	1984-07-18	Lepetit Spa	Ester derivatives
GB8420405D0 (en) *	1984-08-10	1984-09-12	Lepetit Spa	Preparing antibiotic l 17046
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds

1987
- 1987-03-02 GB GB878704847A patent/GB8704847D0/en active Pending
1988
- 1988-02-22 IL IL85493A patent/IL85493A0/xx not_active IP Right Cessation
- 1988-02-23 AT AT88902122T patent/ATE79637T1/de not_active IP Right Cessation
- 1988-02-23 JP JP63501993A patent/JPH0776234B2/ja not_active Expired - Lifetime
- 1988-02-23 HU HU881742A patent/HU205371B/hu not_active IP Right Cessation
- 1988-02-23 EP EP88902122A patent/EP0340245B1/de not_active Expired - Lifetime
- 1988-02-23 WO PCT/EP1988/000129 patent/WO1988006600A1/en not_active Ceased
- 1988-02-23 KR KR1019880701400A patent/KR960014104B1/ko not_active Expired - Lifetime
- 1988-02-23 AU AU13632/88A patent/AU619460B2/en not_active Ceased
- 1988-02-23 DE DE8888902122T patent/DE3873907T2/de not_active Expired - Fee Related
- 1988-02-25 PT PT86827A patent/PT86827B/pt not_active IP Right Cessation
- 1988-02-25 IE IE51388A patent/IE62860B1/en not_active IP Right Cessation
- 1988-02-26 NZ NZ223669A patent/NZ223669A/en unknown
- 1988-02-29 CN CN198888101000A patent/CN88101000A/zh active Pending
- 1988-03-01 ES ES8800594A patent/ES2009555A6/es not_active Expired
- 1988-03-01 GR GR880100118A patent/GR1001625B/el unknown
- 1988-03-01 ZA ZA881445A patent/ZA881445B/xx unknown
- 1988-03-02 PH PH36578A patent/PH27406A/en unknown
- 1988-09-29 DK DK543088A patent/DK543088A/da not_active Application Discontinuation
- 1988-10-28 NO NO884821A patent/NO176568C/no unknown
1989
- 1989-08-31 FI FI894078A patent/FI91765C/fi not_active IP Right Cessation
1992
- 1992-01-21 US US07/826,198 patent/US5198418A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU1363288A (en)	1988-09-26
GR880100118A (en)	1989-01-31
NO176568B (no)	1995-01-16
KR890700607A (ko)	1989-04-26
DE3873907T2 (de)	1993-01-14
KR960014104B1 (ko)	1996-10-14
NO884821L (no)	1988-10-28
HU205371B (en)	1992-04-28
JPH0776234B2 (ja)	1995-08-16
FI894078L (fi)	1989-08-31
DK543088D0 (da)	1988-09-29
US5198418A (en)	1993-03-30
DK543088A (da)	1988-09-29
IL85493A0 (en)	1988-07-31
GR1001625B (el)	1994-07-29
PH27406A (en)	1993-06-21
IE62860B1 (en)	1995-03-08
FI894078A0 (fi)	1989-08-31
IE880513L (en)	1988-09-02
WO1988006600A1 (en)	1988-09-07
FI91765B (fi)	1994-04-29
HUT51300A (en)	1990-04-28
FI91765C (fi)	1994-08-10
PT86827A (pt)	1988-03-01
NO176568C (no)	1995-04-26
PT86827B (pt)	1992-05-29
GB8704847D0 (en)	1987-04-08
AU619460B2 (en)	1992-01-30
ZA881445B (en)	1989-01-25
JPH02502456A (ja)	1990-08-09
DE3873907D1 (de)	1992-09-24
NZ223669A (en)	1990-12-21
CN88101000A (zh)	1988-09-14
EP0340245B1 (de)	1992-08-19
ES2009555A6 (es)	1989-10-01
EP0340245A1 (de)	1989-11-08
NO884821D0 (no)	1988-10-28

Legal Events

Date	Code	Title	Description
1993-02-15	UEP	Publication of translation of european patent specification
1999-11-15	REN	Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
ATE79637T1 (de)	1992-09-15	Substituierte alkylamide von teicoplaninverbindungen.
LV10614A (lv)	1995-04-20	2-anilinopirimidina atvasinajumi
FI904851A0 (fi)	1990-10-02	Radiomaerkta antikoagulantpeptider.
BR8801609A (pt)	1989-02-08	Conjunto de farol substituivel
DE69004685D1 (de)	1993-12-23	Substituierte alkylamidderivate von teicoplanin.
DE69230224D1 (de)	1999-12-02	Potenzierung von nmda-antagonisten
DE68916850D1 (de)	1994-08-25	Antikoagulierende Peptid-Alkohole.
DE58902491D1 (de)	1992-11-26	Neue difluormethyl-thiadiazolyl-oxyessigsaeureamiden.
TR23694A (tr)	1990-07-01	G i z l i
KR890701553A (ko)	1989-12-20	시스테인의 신규 유도체
PT87378A (pt)	1989-05-31	Neue 2-aminoalkyl-4-benzyl-1-(2h)-phthalazinon-derivate
DE3881991D1 (de)	1993-07-29	Zusammensetzung von gleitgliedern.
ATE136884T1 (de)	1996-05-15	Neue 2-mercaptomethylen-tetrahydronaphthalin- und -indan-2-carboxamide als enkephalinaseinhibitoren
KR890010740U (ko)	1989-07-11	공업용 재봉틀의 다리
GR1000471B (el)	1992-07-30	Μεθοδος παρασκευης κινολινοθειοαιθερων.
ATA903787A (de)	1990-12-15	Neue xanthinderivate
DE3855595D1 (de)	1996-11-07	Absoluter Kodierer des Multiumlaufstyps
BR8706170A (pt)	1989-06-06	Amplicador de linha al 4000
SE8700758D0 (sv)	1987-02-24	Motverkar vevning hos hestar
ATA265587A (de)	1992-02-15	Neue 9-deazaguanine
ATA53487A (de)	1991-08-15	Gliederkessel
DE3855592D1 (de)	1996-11-07	Absoluter Kodierer des Multiumlauftyps
DE3855594D1 (de)	1996-11-07	Absoluter Kodierer des Multiumlaufstyps
BR6802719U (pt)	1990-08-07	Disposicao construtiva de quadros
SE8701209D0 (sv)	1987-03-24	Hopfestningsanordning for kledesplagg