DK653089A - 4,5,6,7-tetrahydrobenzimidazolderivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser - Google Patents

4,5,6,7-tetrahydrobenzimidazolderivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser Download PDF

Info

Publication number
DK653089A
DK653089A DK653089A DK653089A DK653089A DK 653089 A DK653089 A DK 653089A DK 653089 A DK653089 A DK 653089A DK 653089 A DK653089 A DK 653089A DK 653089 A DK653089 A DK 653089A
Authority
DK
Denmark
Prior art keywords
group
derivatives
tetrahydrobenzimidazold
procedures
preparing
Prior art date
Application number
DK653089A
Other languages
English (en)
Other versions
DK653089D0 (da
Inventor
Mitsuaki Ohta
Tokuo Koide
Takeshi Suzuki
Akira Matsuhisa
Isao Yanagisawa
Keiji Miyata
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26389240&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK653089(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of DK653089D0 publication Critical patent/DK653089D0/da
Publication of DK653089A publication Critical patent/DK653089A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08Radicals containing only hydrogen and carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Reinforced Plastic Materials (AREA)
  • Adhesive Tapes (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
  • Steroid Compounds (AREA)
DK653089A 1988-12-22 1989-12-21 4,5,6,7-tetrahydrobenzimidazolderivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser DK653089A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP32532788 1988-12-22
JP4889689 1989-02-28

Publications (2)

Publication Number Publication Date
DK653089D0 DK653089D0 (da) 1989-12-21
DK653089A true DK653089A (da) 1990-06-23

Family

ID=26389240

Family Applications (1)

Application Number Title Priority Date Filing Date
DK653089A DK653089A (da) 1988-12-22 1989-12-21 4,5,6,7-tetrahydrobenzimidazolderivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser

Country Status (15)

Country Link
US (1) US4977175A (da)
EP (1) EP0376624B1 (da)
KR (1) KR900009608A (da)
CN (1) CN1027536C (da)
AT (1) ATE111454T1 (da)
AU (1) AU630397B2 (da)
CA (1) CA2004911A1 (da)
DE (1) DE68918257T2 (da)
DK (1) DK653089A (da)
ES (1) ES2063831T3 (da)
FI (1) FI896075A7 (da)
IE (1) IE65639B1 (da)
NO (1) NO178188C (da)
PT (1) PT92609B (da)
YU (1) YU47216B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0381422B1 (en) * 1989-02-02 1996-10-23 Yamanouchi Pharmaceutical Co. Ltd. Tetrahydrobenzimidazole derivatives
GB8928837D0 (en) * 1989-12-21 1990-02-28 Beecham Group Plc Pharmaceuticals
GB9214184D0 (en) * 1992-07-03 1992-08-12 Smithkline Beecham Plc Pharmaceuticals
GB9225141D0 (en) * 1992-12-01 1993-01-20 Smithkline Beecham Corp Chemical compounds
US5262537A (en) * 1993-03-19 1993-11-16 Anaquest, Inc. Derivatives of 4,5,6,7-tetrahydroimidazo-[4,5-c]pyridinyl-6-carboxylic acid
WO1997024334A1 (en) 1995-12-28 1997-07-10 Fujisawa Pharmaceutical Co., Ltd. Benzimidazole derivatives
TW453999B (en) 1997-06-27 2001-09-11 Fujisawa Pharmaceutical Co Benzimidazole derivatives
JP2003527395A (ja) * 2000-03-17 2003-09-16 ノボ ノルディスク アクティーゼルスカブ ヒスタミンh3受容体リガンドとしての縮環イミダゾール
US6437147B1 (en) 2000-03-17 2002-08-20 Novo Nordisk Imidazole compounds
AU2003237881A1 (en) 2002-05-17 2003-12-02 Neurogen Corporation Substituted ring-fused imidazole derivates: gabaa receptor ligands
ES2833251T3 (es) * 2016-08-16 2021-06-14 Bayer Cropscience Ag Procedimiento para producir derivados de 2-(3,6-dihalopiridin-2-il)-3h-imidazol[4,5-c]piridina y compuestos relacionados por reacción del derivado de piridina 3h-imidazol[4,5-c] con una base organometálica de zinc-amina

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1260294A (en) * 1968-03-15 1972-01-12 Rhein Chemie Holding G M B H 4,5,6,7-tetrahydrobenzimidazoles, process for their production and their use as corrosion inhibitors and antioxidants
DE1948795A1 (de) * 1969-09-26 1971-04-08 Rhein Chemie Rheinau Gmbh 4,5,6,7-Tetrahydrobenzimidazole,Verfahren zu ihrer Herstellung und ihre Verwendung als Korrosionsinhibitoren und Alterungsschutzmittel
US3987054A (en) * 1970-09-23 1976-10-19 Pliva Pharmaceutical And Chemical Works 4,5,6,7-tetrahydrobenzimidazoles
FR2531083B1 (fr) * 1982-06-29 1986-11-28 Sandoz Sa Nouveaux derives de la piperidine, leur preparation et leur utilisation comme medicaments
SE460359B (sv) * 1984-01-25 1989-10-02 Glaxo Group Ltd 3-imidazolylmetyltetrahydrokarbazoloner, foerfarande foer framstaellning av dessa och en farmaceutisk komposition
DE3650772T2 (de) * 1985-04-27 2003-04-03 F. Hoffmann-La Roche Ag, Basel Derivate von Indazole-3-carboxamide und -3-carboxylsäure
US4826990A (en) * 1987-09-30 1989-05-02 American Home Products Corporation 2-aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents

Also Published As

Publication number Publication date
EP0376624B1 (en) 1994-09-14
AU630397B2 (en) 1992-10-29
ES2063831T3 (es) 1995-01-16
IE894185L (en) 1990-06-22
DK653089D0 (da) 1989-12-21
DE68918257D1 (de) 1994-10-20
YU243989A (en) 1991-02-28
YU47216B (sh) 1995-01-31
FI896075A0 (fi) 1989-12-19
PT92609B (pt) 1995-09-12
CA2004911A1 (en) 1990-06-22
NO178188C (no) 1996-02-07
NO895198L (no) 1990-06-25
ATE111454T1 (de) 1994-09-15
NO178188B (no) 1995-10-30
PT92609A (pt) 1990-06-29
CN1027536C (zh) 1995-02-01
US4977175A (en) 1990-12-11
EP0376624A1 (en) 1990-07-04
DE68918257T2 (de) 1995-02-02
FI896075A7 (fi) 1990-06-23
IE65639B1 (en) 1995-11-15
KR900009608A (ko) 1990-07-05
CN1043706A (zh) 1990-07-11
AU4714589A (en) 1990-06-28
NO895198D0 (no) 1989-12-21

Similar Documents

Publication Publication Date Title
DK0427549T3 (da) Heterocykliske oxy-phenoxyeddikesyrederivater og deres anvendelse som herbicider
DK0673937T3 (da) Bicyclisk heterocyclisk sulfonamid og sulfonsyreesterderivater
DK426289D0 (da) Spiroforbindelser og farmaceutisk praeparat indeholdende en saadan forbindelse
EP0225739A3 (en) 2-2-dimethyl-3-hydroxy-3-propargyl-4-(1,2,4-triazole-1-yl -butane derivatives as plant growth regulators
DK653089D0 (da) 4,5,6,7-tetrahydrobenzimidazolderivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser
DK519985D0 (da) Quinoloncarboxylsyrederivater, fremgangsmaade til fremstilling deraf og antibakterielt middel indeholdende saadanne derivater
IS3828A (is) Hliðstæð aðferð til tilreiðslu á nýjum afleiðum thiazolidinone og oxazolidinone sem gagnlegar eru til æðaútvíkkunar
EP0417790A3 (en) S-triazolo(3,4-i)purine derivatives
SU1568881A3 (ru) Cпocoб бopьбы c гpибhыmи зaбoлebahияmи pactehий
CS275480B2 (en) Fungicide and method of active substances production
AU1586588A (en) Fungicidal derivatives of propenoic acid and processes for their preparation
ES540288A0 (es) Un procedimiento de preparar un derivado de n-acil-amino- acido
EP0307226B1 (en) Process for the preparation of a macrolide compound

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment