DOP2002000384A - Moduladores de receptores estrogenicos. - Google Patents
Moduladores de receptores estrogenicos.Info
- Publication number
- DOP2002000384A DOP2002000384A DO2002000384A DO2002000384A DOP2002000384A DO P2002000384 A DOP2002000384 A DO P2002000384A DO 2002000384 A DO2002000384 A DO 2002000384A DO 2002000384 A DO2002000384 A DO 2002000384A DO P2002000384 A DOP2002000384 A DO P2002000384A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- compounds
- estrogenic
- estrogen
- cancer
- modulators
- Prior art date
Links
- 102000015694 estrogen receptors Human genes 0.000 title 1
- 108010038795 estrogen receptors Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000001076 estrogenic effect Effects 0.000 abstract 2
- 208000010392 Bone Fractures Diseases 0.000 abstract 1
- 206010065687 Bone loss Diseases 0.000 abstract 1
- 208000014644 Brain disease Diseases 0.000 abstract 1
- 206010006187 Breast cancer Diseases 0.000 abstract 1
- 208000026310 Breast neoplasm Diseases 0.000 abstract 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 201000009273 Endometriosis Diseases 0.000 abstract 1
- 208000033830 Hot Flashes Diseases 0.000 abstract 1
- 206010060800 Hot flush Diseases 0.000 abstract 1
- 206010021639 Incontinence Diseases 0.000 abstract 1
- 238000008214 LDL Cholesterol Methods 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 208000031481 Pathologic Constriction Diseases 0.000 abstract 1
- 206010060862 Prostate cancer Diseases 0.000 abstract 1
- 208000000236 Prostatic Neoplasms Diseases 0.000 abstract 1
- 208000002495 Uterine Neoplasms Diseases 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 210000000481 breast Anatomy 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 210000000845 cartilage Anatomy 0.000 abstract 1
- 230000004663 cell proliferation Effects 0.000 abstract 1
- 230000003920 cognitive function Effects 0.000 abstract 1
- 230000007850 degeneration Effects 0.000 abstract 1
- 230000003412 degenerative effect Effects 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 239000002834 estrogen receptor modulator Substances 0.000 abstract 1
- 201000000079 gynecomastia Diseases 0.000 abstract 1
- 230000001771 impaired effect Effects 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 102000005962 receptors Human genes 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
- 208000037804 stenosis Diseases 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 206010046766 uterine cancer Diseases 0.000 abstract 1
- 210000004291 uterus Anatomy 0.000 abstract 1
- 210000004509 vascular smooth muscle cell Anatomy 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
El invento presente se relaciona a compuestos y derivados del mismo, su síntesis, y su uso como moduladores de receptores estrogénicos. Los compuestos del invento instante son ligandos para los receptores estrogénicos y como tales pueden ser útiles en el tratamiento o prevención de una variedad de condiciones relacionadas con el funcionamiento estrogénico incluyendo: pérdida de hueso, fracturas óseas, osteoporosis, degeneración de cartílago, endometriosis, miomatosis uterina, calores inducidos por menopausia o ausencia de estrógeno (bochornos), niveles aumentados de colesterol LDL, enfermedad cardiovascular, impedimento de la función cognoscitiva, enfermedades cerebrales degenerativas, re-estenosis, ginecomastia, proliferaciones de células de músculo liso vascular, incontinencia, y cáncer, en especial cáncer de mama, útero y próstata.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000384A DOP2002000384A (es) | 2002-04-19 | 2002-04-19 | Moduladores de receptores estrogenicos. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000384A DOP2002000384A (es) | 2002-04-19 | 2002-04-19 | Moduladores de receptores estrogenicos. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2002000384A true DOP2002000384A (es) | 2003-09-30 |
Family
ID=44261073
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2002000384A DOP2002000384A (es) | 2002-04-19 | 2002-04-19 | Moduladores de receptores estrogenicos. |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2002000384A (es) |
-
2002
- 2002-04-19 DO DO2002000384A patent/DOP2002000384A/es unknown
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