EA200602017A1 - КОМПОЗИЦИЯ ДЛЯ АЭРОЗОЛЬНОЙ ИНГАЛЯЦИИ β-АГОНИСТОВ - Google Patents

КОМПОЗИЦИЯ ДЛЯ АЭРОЗОЛЬНОЙ ИНГАЛЯЦИИ β-АГОНИСТОВ

Info

Publication number
EA200602017A1
EA200602017A1 EA200602017A EA200602017A EA200602017A1 EA 200602017 A1 EA200602017 A1 EA 200602017A1 EA 200602017 A EA200602017 A EA 200602017A EA 200602017 A EA200602017 A EA 200602017A EA 200602017 A1 EA200602017 A1 EA 200602017A1
Authority
EA
Eurasian Patent Office
Prior art keywords
aerosol inhalation
agonists
composition
propellant
residues
Prior art date
Application number
EA200602017A
Other languages
English (en)
Other versions
EA012583B1 (ru
Inventor
Майкл Эйвен
Original Assignee
Бёрингер Ингельхайм Интернациональ Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34979667&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200602017(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of EA200602017A1 publication Critical patent/EA200602017A1/ru
Publication of EA012583B1 publication Critical patent/EA012583B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/04Amoebicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Dispersion Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

В заявке описана не содержащая пропеллент лекарственная композиция для аэрозольной ингаляции, содержащая одно или несколько соединений общей формулы ()в которой остатки R, R, Rи Хмогут иметь указанные в формуле изобретения и описании значения.
EA200602017A 2004-05-14 2005-05-10 КОМПОЗИЦИЯ ДЛЯ АЭРОЗОЛЬНОЙ ИНГАЛЯЦИИ β-АГОНИСТОВ EA012583B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004024452A DE102004024452A1 (de) 2004-05-14 2004-05-14 Aerosolformulierung für die Inhalation von Betaagonisten
PCT/EP2005/005028 WO2005110421A2 (de) 2004-05-14 2005-05-10 Aerosolformulierung für die inhalation von betaagonisten

Publications (2)

Publication Number Publication Date
EA200602017A1 true EA200602017A1 (ru) 2007-06-29
EA012583B1 EA012583B1 (ru) 2009-10-30

Family

ID=34979667

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200602017A EA012583B1 (ru) 2004-05-14 2005-05-10 КОМПОЗИЦИЯ ДЛЯ АЭРОЗОЛЬНОЙ ИНГАЛЯЦИИ β-АГОНИСТОВ

Country Status (26)

Country Link
EP (1) EP1809293B1 (ru)
JP (1) JP4620730B2 (ru)
KR (1) KR101288791B1 (ru)
CN (1) CN101056640A (ru)
AR (1) AR049096A1 (ru)
AU (1) AU2005244414B2 (ru)
BR (1) BRPI0511135B8 (ru)
CA (1) CA2564379C (ru)
DE (1) DE102004024452A1 (ru)
DK (1) DK1809293T3 (ru)
EA (1) EA012583B1 (ru)
EC (1) ECSP067004A (ru)
ES (1) ES2575925T3 (ru)
HU (1) HUE027780T2 (ru)
IL (1) IL179218A (ru)
MX (1) MXPA06013216A (ru)
MY (1) MY148403A (ru)
NO (1) NO20065030L (ru)
PE (1) PE20060311A1 (ru)
PL (1) PL1809293T3 (ru)
SG (1) SG152265A1 (ru)
TW (1) TWI356703B (ru)
UA (1) UA87312C2 (ru)
UY (1) UY28891A1 (ru)
WO (1) WO2005110421A2 (ru)
ZA (1) ZA200607462B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
KR101360803B1 (ko) 2005-08-15 2014-02-11 베링거 인겔하임 인터내셔날 게엠베하 베타모방제의 제조방법
BRPI0618370A2 (pt) * 2005-11-09 2011-08-30 Boehringer Ingelheim Int formulação aerossol de medicamento, uso do mesmo e kit de inalação
UY30543A1 (es) * 2006-08-18 2008-03-31 Boehringer Ingelheim Int Formulacion de aerosol para la inhalacion de beta- agonistas
CA2738616A1 (en) * 2008-11-21 2010-05-27 Boehringer Ingelheim International Gmbh Aerosol formulation for the inhalation of beta agonists
US20110281858A1 (en) * 2008-11-21 2011-11-17 Boehringer Ingelheim International Gmbh Aerosol formulation for the inhalation of beta agonists
EP2906218B1 (en) 2012-10-09 2016-12-14 Boehringer Ingelheim International GmbH Beta-2-adrenoceptor agonist for the treatment of cough
JP2019536812A (ja) 2016-12-12 2019-12-19 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング オロダテロールとの同時投与による間質性肺疾患の処置方法に使用するためのニンテダニブ
EP4069669A1 (en) * 2019-12-05 2022-10-12 Syngenta Crop Protection AG One step process for the preparation of phenyl ethyl amine derivatives

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3134590A1 (de) * 1981-09-01 1983-03-10 Boehringer Ingelheim KG, 6507 Ingelheim Neue benzo-heterocyclen
US4460581A (en) * 1982-10-12 1984-07-17 Boehringer Ingelheim Kg (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones
JPH0637388B2 (ja) * 1986-02-17 1994-05-18 千寿製薬株式会社 水性液剤
GB9405019D0 (en) * 1994-03-15 1994-04-27 Smithkline Beecham Plc Novel compounds
DE10253282A1 (de) * 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung
WO2005102349A1 (de) * 2004-04-22 2005-11-03 Boehringer Ingelheim International Gmbh Arzneinmittelkombinationen enthaltend benzoxazine zur behandlung von atemwegserkrankungen
DE102004019539A1 (de) * 2004-04-22 2005-11-10 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von Atemwegserkrankungen
DE102004024454A1 (de) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
DE102004024451A1 (de) * 2004-05-14 2005-12-22 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pulverformulierungen für die Inhalation, die Enantiomerenreine Betaagonisten enthalten

Also Published As

Publication number Publication date
DE102004024452A1 (de) 2005-12-08
PL1809293T3 (pl) 2016-09-30
BRPI0511135A (pt) 2007-11-27
IL179218A0 (en) 2007-03-08
NO20065030L (no) 2006-11-30
ZA200607462B (en) 2008-06-25
KR20070022084A (ko) 2007-02-23
IL179218A (en) 2012-10-31
CN101056640A (zh) 2007-10-17
AU2005244414A1 (en) 2005-11-24
TW200608981A (en) 2006-03-16
DK1809293T3 (en) 2016-06-20
EA012583B1 (ru) 2009-10-30
EP1809293A2 (de) 2007-07-25
WO2005110421A2 (de) 2005-11-24
HUE027780T2 (en) 2016-11-28
BRPI0511135B1 (pt) 2019-11-12
TWI356703B (en) 2012-01-21
UY28891A1 (es) 2005-12-30
WO2005110421A3 (de) 2006-03-16
ECSP067004A (es) 2007-02-28
ES2575925T3 (es) 2016-07-04
KR101288791B1 (ko) 2013-07-29
AR049096A1 (es) 2006-06-28
AU2005244414B2 (en) 2010-12-09
EP1809293B1 (de) 2016-03-16
CA2564379A1 (en) 2005-11-24
JP2007537188A (ja) 2007-12-20
MXPA06013216A (es) 2007-02-08
MY148403A (en) 2013-04-30
CA2564379C (en) 2013-07-30
BRPI0511135B8 (pt) 2021-05-25
UA87312C2 (ru) 2009-07-10
PE20060311A1 (es) 2006-05-08
JP4620730B2 (ja) 2011-01-26
SG152265A1 (en) 2009-05-29

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Legal Events

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KZ KG MD TJ TM

ND4A Extension of term of a eurasian patent
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): BY