ECSP003403A - PROTEASE INHIBITORS XI - Google Patents

PROTEASE INHIBITORS XI

Info

Publication number
ECSP003403A
ECSP003403A ECSP003403A ECSP003403A EC SP003403 A ECSP003403 A EC SP003403A EC SP003403 A ECSP003403 A EC SP003403A EC SP003403 A ECSP003403 A EC SP003403A
Authority
EC
Ecuador
Prior art keywords
excessive
disease
cartilage
matrix
proteases
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Yamashita Dennis Shinji
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP003403 priority Critical patent/ECSP003403A/en
Publication of ECSP003403A publication Critical patent/ECSP003403A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención proporciona inhibidores de proteasas de 4-amino-4,5-dihidro-benzo [b] [1,4] dioxocin-3-ona, y sus sales, hidratos y solvatos farmacéuticamente aceptables que inhiben las proteasas, con inclusión de la captesina K, composiciones farmacéuticas de tales compuestos y métodos para tratar enfermedades de pérdida ósea excesiva o degradación excesiva de cartílago o matriz, que incluyen osteoporosis, enfermedad gingival con inclusión de gingivitis y periodontitis, artritis, más especificamente osteoartritis y artritis reumatoide; enfermedad de Paget; hipercalcemia de carácter maligno; y enfermedad metabólica osea, que comprenden inhibir dicha pérdida ósea o degradación excesiva de cartílago o matriz por administración a un paciente que se encuentra en necesidad de ello de un compuesto de la presente invención.The present invention provides inhibitors of 4-amino-4,5-dihydro-benzo [b] [1,4] dioxocin-3-one proteases, and their pharmaceutically acceptable salts, hydrates and solvates that inhibit proteases, including captesin K, pharmaceutical compositions of such compounds, and methods of treating diseases of excessive bone loss or excessive degradation of cartilage or matrix, including osteoporosis, gingival disease including gingivitis and periodontitis, arthritis, more specifically osteoarthritis and rheumatoid arthritis; Paget's disease; malignant hypercalcemia; and bone metabolic disease, which comprises inhibiting said bone loss or excessive cartilage or matrix degradation by administration to a patient in need thereof of a compound of the present invention.

ECSP003403 2000-03-28 2000-03-28 PROTEASE INHIBITORS XI ECSP003403A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP003403 ECSP003403A (en) 2000-03-28 2000-03-28 PROTEASE INHIBITORS XI

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP003403 ECSP003403A (en) 2000-03-28 2000-03-28 PROTEASE INHIBITORS XI

Publications (1)

Publication Number Publication Date
ECSP003403A true ECSP003403A (en) 2000-05-25

Family

ID=42041033

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP003403 ECSP003403A (en) 2000-03-28 2000-03-28 PROTEASE INHIBITORS XI

Country Status (1)

Country Link
EC (1) ECSP003403A (en)

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