ECSP003445A - Pirazolbenzodiazepinas - Google Patents

Pirazolbenzodiazepinas

Info

Publication number
ECSP003445A
ECSP003445A ECSP003445A ECSP003445A EC SP003445 A ECSP003445 A EC SP003445A EC SP003445 A ECSP003445 A EC SP003445A EC SP003445 A ECSP003445 A EC SP003445A
Authority
EC
Ecuador
Prior art keywords
pirazolbenzodiazepinas
pyrazobenzodiazepines
antiprofilerative
cdfs
colon
Prior art date
Application number
Other languages
English (en)
Inventor
Vincent Madison
Qingjie Ding
Peter Michael Wovkulich
Chung-Chen Wei
Jin Jun Liu
Giacomo Pizzolato
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP003445 priority Critical patent/ECSP003445A/es
Publication of ECSP003445A publication Critical patent/ECSP003445A/es

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Nuevas pirazolbenzodiazepinas que presentan la fórmula (gráfico), y las sales farmacéuticamente aceptables de las mismas, en donde R1, R2, R3 y R4 son como se han definido aquí, son inhibidores de quinasas dependientes de ciclina (CDFs), en particular CDK2 y son agentes antiprofilerativos útiles en el tratamiento o control de los trastornos proliferativos celulares, en particular, tumores de mama, colon, pulmón y prostata.
ECSP003445 2000-04-27 2000-04-27 Pirazolbenzodiazepinas ECSP003445A (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP003445 ECSP003445A (es) 2000-04-27 2000-04-27 Pirazolbenzodiazepinas

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP003445 ECSP003445A (es) 2000-04-27 2000-04-27 Pirazolbenzodiazepinas

Publications (1)

Publication Number Publication Date
ECSP003445A true ECSP003445A (es) 2000-11-24

Family

ID=42041073

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP003445 ECSP003445A (es) 2000-04-27 2000-04-27 Pirazolbenzodiazepinas

Country Status (1)

Country Link
EC (1) ECSP003445A (es)

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