ECSP003478A - SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL - Google Patents
SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALLInfo
- Publication number
- ECSP003478A ECSP003478A ECSP003478A ECSP003478A EC SP003478 A ECSP003478 A EC SP003478A EC SP003478 A ECSP003478 A EC SP003478A EC SP003478 A ECSP003478 A EC SP003478A
- Authority
- EC
- Ecuador
- Prior art keywords
- useful
- substituted
- heteroaril
- uracils
- selective inhibition
- Prior art date
Links
- 230000015271 coagulation Effects 0.000 title abstract 2
- 238000005345 coagulation Methods 0.000 title abstract 2
- 230000005764 inhibitory process Effects 0.000 title 1
- ISAKRJDGNUQOIC-UHFFFAOYSA-N Uracil Chemical compound O=C1C=CNC(=O)N1 ISAKRJDGNUQOIC-UHFFFAOYSA-N 0.000 abstract 2
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 229940127219 anticoagulant drug Drugs 0.000 abstract 1
- 208000026106 cerebrovascular disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000029078 coronary artery disease Diseases 0.000 abstract 1
- 210000004351 coronary vessel Anatomy 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 239000003001 serine protease inhibitor Substances 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 230000001732 thrombotic effect Effects 0.000 abstract 1
- 229940035893 uracil Drugs 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
El invento se relaciona a compuestos de aril policiclico sustituido y uracilos y heteroaril útiles como inhibidores de serinas proteasas de la cascada de coagulación y sus compuestos, composiciones y métodos para la terapia anticoagulante para el tratamiento y prevención de una variedad de condiciones trombóticas incluyendo arteria coronaria y enfermedades cerebrovasculares.The invention relates to substituted polycyclic aryl and uracil and heteroaryl compounds useful as coagulation cascade serine protease inhibitors and their compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombotic conditions including coronary artery and cerebrovascular diseases.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003478 ECSP003478A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003478 ECSP003478A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003478A true ECSP003478A (en) | 2000-11-24 |
Family
ID=42041104
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003478 ECSP003478A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003478A (en) |
-
2000
- 2000-05-19 EC ECSP003478 patent/ECSP003478A/en unknown
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