ECSP067091A - Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina - Google Patents

Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina

Info

Publication number
ECSP067091A
ECSP067091A EC2006007091A ECSP067091A ECSP067091A EC SP067091 A ECSP067091 A EC SP067091A EC 2006007091 A EC2006007091 A EC 2006007091A EC SP067091 A ECSP067091 A EC SP067091A EC SP067091 A ECSP067091 A EC SP067091A
Authority
EC
Ecuador
Prior art keywords
receptor antagonists
gonadotropine
processes
preparation
free
Prior art date
Application number
EC2006007091A
Other languages
English (en)
Inventor
Alexander V Gontcharov
Gulnaz Khafizova
John R Potoski
Donna Mary Huryn
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP067091A publication Critical patent/ECSP067091A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención se relaciona a métodos de producción de antagonistas de receptor de Hormona que Libera Gonadotropina ("GnRH") (también conocida como Hormona que Libera Hormona de Luteinización).
EC2006007091A 2004-06-17 2006-12-18 Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina ECSP067091A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58066504P 2004-06-17 2004-06-17

Publications (1)

Publication Number Publication Date
ECSP067091A true ECSP067091A (es) 2007-01-26

Family

ID=34972567

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006007091A ECSP067091A (es) 2004-06-17 2006-12-18 Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina

Country Status (16)

Country Link
US (1) US7714130B2 (es)
EP (1) EP1756093A1 (es)
JP (1) JP2008503470A (es)
CN (1) CN1968948A (es)
AU (1) AU2005264998A1 (es)
BR (1) BRPI0512239A (es)
CA (1) CA2570693A1 (es)
CR (1) CR8786A (es)
EC (1) ECSP067091A (es)
IL (1) IL179993A0 (es)
MX (1) MXPA06014797A (es)
NO (1) NO20070248L (es)
NZ (1) NZ552093A (es)
RU (1) RU2007101509A (es)
WO (1) WO2006009736A1 (es)
ZA (1) ZA200610594B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0512239A (pt) 2004-06-17 2008-02-19 Wyeth Corp processos para preparação de antagonistas de receptores de hormÈnios liberadores de gonatropina
EP1758895A1 (en) * 2004-06-17 2007-03-07 Wyeth a Corporation of the State of Delaware Gonadotropin releasing hormone receptor antagonists
CA2587853A1 (en) * 2004-11-23 2006-06-01 Wyeth Gonadotropin releasing hormone receptor antagonists
US7534796B2 (en) * 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor
US7538113B2 (en) * 2005-02-18 2009-05-26 Wyeth 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7582634B2 (en) * 2005-02-18 2009-09-01 Wyeth 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US20060189619A1 (en) * 2005-02-24 2006-08-24 Wyeth 3-({4-[2-(4-Tert-butylphenyl)-1h-benzimidazol-4-yl]piperazin-1-yl}methyl)pyrido[2,3-b]]pyrazi ne compounds
JP2008533025A (ja) * 2005-03-07 2008-08-21 ワイス キノキサリンジヒドロハライド二水和物およびそのための合成方法
US7531542B2 (en) * 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) * 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor
WO2016061190A1 (en) 2014-10-14 2016-04-21 The Board Of Trustees Of The Leland Stanford Junior University Method for treating neurodegenerative diseases
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BR112021002165A2 (pt) 2018-08-06 2021-05-04 The Board Of Trustees Of The Leland Stanford Junior University composto, composição farmacêutica, e, métodos para tratar uma doença neurodegenerativa e deficiência cognitiva associada ao envelhecimento e neuroinflamação

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US7531542B2 (en) * 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) * 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor

Also Published As

Publication number Publication date
JP2008503470A (ja) 2008-02-07
MXPA06014797A (es) 2007-02-16
IL179993A0 (en) 2007-05-15
ZA200610594B (en) 2008-07-30
NO20070248L (no) 2007-01-15
BRPI0512239A (pt) 2008-02-19
NZ552093A (en) 2009-06-26
CR8786A (es) 2007-08-28
CA2570693A1 (en) 2006-01-26
US7714130B2 (en) 2010-05-11
EP1756093A1 (en) 2007-02-28
US20050282820A1 (en) 2005-12-22
WO2006009736A1 (en) 2006-01-26
AU2005264998A1 (en) 2006-01-26
CN1968948A (zh) 2007-05-23
RU2007101509A (ru) 2008-07-27

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