ECSP067091A - Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina - Google Patents

Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina

Info

Publication number
ECSP067091A
ECSP067091A EC2006007091A ECSP067091A ECSP067091A EC SP067091 A ECSP067091 A EC SP067091A EC 2006007091 A EC2006007091 A EC 2006007091A EC SP067091 A ECSP067091 A EC SP067091A EC SP067091 A ECSP067091 A EC SP067091A
Authority
EC
Ecuador
Prior art keywords
receptor antagonists
gonadotropine
processes
preparation
free
Prior art date
Application number
EC2006007091A
Other languages
English (en)
Inventor
Alexander V Gontcharov
Gulnaz Khafizova
John R Potoski
Donna Mary Huryn
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP067091A publication Critical patent/ECSP067091A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08Radicals containing only hydrogen and carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención se relaciona a métodos de producción de antagonistas de receptor de Hormona que Libera Gonadotropina ("GnRH") (también conocida como Hormona que Libera Hormona de Luteinización).
EC2006007091A 2004-06-17 2006-12-18 Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina ECSP067091A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58066504P 2004-06-17 2004-06-17

Publications (1)

Publication Number Publication Date
ECSP067091A true ECSP067091A (es) 2007-01-26

Family

ID=34972567

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006007091A ECSP067091A (es) 2004-06-17 2006-12-18 Procesos para preparacion de antagonistas de receptor de hormona que libera gonadotropina

Country Status (16)

Country Link
US (1) US7714130B2 (es)
EP (1) EP1756093A1 (es)
JP (1) JP2008503470A (es)
CN (1) CN1968948A (es)
AU (1) AU2005264998A1 (es)
BR (1) BRPI0512239A (es)
CA (1) CA2570693A1 (es)
CR (1) CR8786A (es)
EC (1) ECSP067091A (es)
IL (1) IL179993A0 (es)
MX (1) MXPA06014797A (es)
NO (1) NO20070248L (es)
NZ (1) NZ552093A (es)
RU (1) RU2007101509A (es)
WO (1) WO2006009736A1 (es)
ZA (1) ZA200610594B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006009734A1 (en) * 2004-06-17 2006-01-26 Wyeth Gonadotropin releasing hormone receptor antagonists
WO2006009736A1 (en) 2004-06-17 2006-01-26 Wyeth Processes for preparing gonadotropin releasing hormone receptor antagonists
CN101048383A (zh) * 2004-11-23 2007-10-03 惠氏公司 促性腺激素释放激素受体拮抗剂
US7538113B2 (en) * 2005-02-18 2009-05-26 Wyeth 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7534796B2 (en) * 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor
US7582634B2 (en) * 2005-02-18 2009-09-01 Wyeth 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US20060189619A1 (en) * 2005-02-24 2006-08-24 Wyeth 3-({4-[2-(4-Tert-butylphenyl)-1h-benzimidazol-4-yl]piperazin-1-yl}methyl)pyrido[2,3-b]]pyrazi ne compounds
CA2601978A1 (en) * 2005-03-07 2006-09-14 Wyeth Quinoxaline dihydrohalide dihydrates and synthetic methods therefor
US7531542B2 (en) * 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) * 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor
US10272070B2 (en) 2014-10-14 2019-04-30 The Board of Trustees of the Leland Stanford Junio r University Method for treating neurodegenerative diseases
CN105879033B (zh) * 2015-04-01 2019-03-26 北京大学人民医院 GnRH Ⅱ型拮抗剂在抑制孕激素耐药子宫内膜癌细胞增殖中的应用
EP3390367B1 (en) 2015-12-15 2020-09-09 The Board of Trustees of the Leland Stanford Junior University Method for preventing and/or treating aging-associated cognitive impairment and neuroinflammation
MX2021001456A (es) 2018-08-06 2021-05-27 Univ Leland Stanford Junior 2-arilbenzimidazoles como activadores de ppargc1a para tratar enfermedades neurodegenerativas.

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Also Published As

Publication number Publication date
CN1968948A (zh) 2007-05-23
RU2007101509A (ru) 2008-07-27
WO2006009736A1 (en) 2006-01-26
NO20070248L (no) 2007-01-15
CR8786A (es) 2007-08-28
MXPA06014797A (es) 2007-02-16
JP2008503470A (ja) 2008-02-07
ZA200610594B (en) 2008-07-30
US20050282820A1 (en) 2005-12-22
BRPI0512239A (pt) 2008-02-19
IL179993A0 (en) 2007-05-15
NZ552093A (en) 2009-06-26
CA2570693A1 (en) 2006-01-26
EP1756093A1 (en) 2007-02-28
AU2005264998A1 (en) 2006-01-26
US7714130B2 (en) 2010-05-11

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