ECSP10010625A - Derivados de iminopiridina y uso de los mismos - Google Patents
Derivados de iminopiridina y uso de los mismosInfo
- Publication number
- ECSP10010625A ECSP10010625A EC2010010625A ECSP10010625A ECSP10010625A EC SP10010625 A ECSP10010625 A EC SP10010625A EC 2010010625 A EC2010010625 A EC 2010010625A EC SP10010625 A ECSP10010625 A EC SP10010625A EC SP10010625 A ECSP10010625 A EC SP10010625A
- Authority
- EC
- Ecuador
- Prior art keywords
- iminopiridine
- derivatives
- same
- compound
- prophylactic
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000026723 Urinary tract disease Diseases 0.000 abstract 1
- 208000012931 Urologic disease Diseases 0.000 abstract 1
- 239000000674 adrenergic antagonist Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000000069 prophylactic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
- 208000014001 urinary system disease Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Se describe un compuesto el cual tiene una excelente actividad selectiva superior como antagonista del receptor adrenérgico 1D y por lo tanto es útil como un agente profiláctico/terapéutico para el tratamiento de una enfermedad del tracto urinario inferior y similares. Se describe específicamente un compuesto representado por la fórmula (I) [en donde cada símbolo es como se definió en la descripción] o una de sus sales.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2008113130 | 2008-04-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP10010625A true ECSP10010625A (es) | 2011-03-31 |
Family
ID=41216865
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2010010625A ECSP10010625A (es) | 2008-04-23 | 2010-11-23 | Derivados de iminopiridina y uso de los mismos |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20110039892A1 (es) |
| EP (1) | EP2269989A4 (es) |
| JP (1) | JPWO2009131135A1 (es) |
| KR (1) | KR20110005277A (es) |
| CN (1) | CN102066328A (es) |
| AU (1) | AU2009238999A1 (es) |
| BR (1) | BRPI0911464A2 (es) |
| CA (1) | CA2722031A1 (es) |
| CO (1) | CO6260133A2 (es) |
| CR (1) | CR11766A (es) |
| DO (1) | DOP2010000322A (es) |
| EA (1) | EA201071228A1 (es) |
| EC (1) | ECSP10010625A (es) |
| IL (1) | IL208824A0 (es) |
| MX (1) | MX2010011651A (es) |
| WO (1) | WO2009131135A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2535330A3 (en) * | 2006-10-23 | 2012-12-26 | Takeda Pharmaceutical Company Limited | Iminopyridine derivative and use thereof |
| US8481569B2 (en) * | 2008-04-23 | 2013-07-09 | Takeda Pharmaceutical Company Limited | Iminopyridine derivatives and use thereof |
| MY184642A (en) * | 2011-08-26 | 2021-04-13 | Meiji Seika Pharma Co Ltd | Method for producing pest control agent |
| AU2022388884A1 (en) * | 2021-11-15 | 2024-05-30 | Pi Industries Ltd. | Bicyclic heteroaromatic compounds and their use as pest control agents |
Family Cites Families (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4840544B1 (es) | 1970-04-24 | 1973-12-01 | ||
| DD106377A1 (es) | 1973-06-18 | 1974-06-12 | ||
| NL175059C (nl) * | 1974-02-23 | Boehringer Mannheim Gmbh | Bereiding van bloeddrukverlagende stoffen en van preparaten die ze bevatten. | |
| GR78245B (es) | 1980-09-12 | 1984-09-26 | Ciba Geigy Ag | |
| FR2540109B1 (fr) * | 1983-01-28 | 1985-08-30 | Logeais Labor Jacques | Imino-2 pyrrolidines, leur procede de preparation et leurs applications en therapeutique |
| DD263759A1 (de) | 1986-04-01 | 1989-01-11 | Akad Wissenschaften Ddr | Verfahren zur herstellung von 1-substituierten 2-imino-5-(pyrid-4-yl)-1,2-dihydro-pyridin-3-carbonsaeure-derivaten |
| US5252498A (en) * | 1989-08-28 | 1993-10-12 | Semiconductor Energy Laboratory Co., Ltd. | Method of forming electronic devices utilizing diamond |
| DE4021439A1 (de) * | 1989-12-14 | 1991-06-20 | Bayer Ag | 2-iminopyridin-derivate |
| US5688795A (en) * | 1994-11-08 | 1997-11-18 | Syntex (U.S.A.) Inc. | 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy!-pyridine, pyrimidine and benzene derivatives as α1 -adrenoceptor antagonists |
| JP2992677B2 (ja) | 1995-06-05 | 1999-12-20 | 武田薬品工業株式会社 | 骨形成促進医薬組成物 |
| US6218396B1 (en) * | 1998-02-20 | 2001-04-17 | Orth-Mcneil Pharmaceutical, Inc. | Substituted pyridino arylpiperazines useful in the treatment of benign prostatic hyperplasia |
| US6153614A (en) * | 1998-07-16 | 2000-11-28 | Abbott Laboratories | Piperazinyl pyrimidine dione compounds selective for adrenoceptors |
| CA2338037A1 (en) * | 1998-07-17 | 2000-01-27 | Synaptic Pharmaceutical Corporation | Compounds specific for the human .alpha.1d adrenergic receptor and uses thereof |
| DE19845202A1 (de) * | 1998-10-01 | 2000-04-06 | Wella Ag | Haarwuchsmittel |
| AU9598601A (en) * | 2000-10-20 | 2002-04-29 | Eisai Co Ltd | Nitrogenous aromatic ring compounds |
| FR2825705B1 (fr) * | 2001-06-08 | 2005-05-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
| US7375100B2 (en) * | 2003-06-04 | 2008-05-20 | Pfizer Inc | 2-amino-pyridine derivatives useful for the treatment of diseases |
| ES2241496B1 (es) * | 2004-04-15 | 2006-12-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de piridina. |
| US20050288270A1 (en) * | 2004-05-27 | 2005-12-29 | Pfizer Inc | New aminopyridine derivatives and their use as pharmaceuticals |
| TW200700392A (en) * | 2005-03-16 | 2007-01-01 | Astrazeneca Ab | Novel compounds |
| ES2303758B1 (es) * | 2006-02-20 | 2009-08-13 | Laboratorios Almirall S.A. | Nuevos derivados de piridin-3-amina. |
| EP2535330A3 (en) * | 2006-10-23 | 2012-12-26 | Takeda Pharmaceutical Company Limited | Iminopyridine derivative and use thereof |
| JP4117008B2 (ja) | 2006-10-30 | 2008-07-09 | シャープ株式会社 | 暗号化装置 |
| MY150032A (en) * | 2007-07-19 | 2013-11-29 | Merck Sharp & Dohme | Heterocyclic amide compounds as protein kinase inhibitors |
| WO2009115572A2 (en) * | 2008-03-21 | 2009-09-24 | Novartis Ag | Novel heterocyclic compounds and uses therof |
| US8481569B2 (en) * | 2008-04-23 | 2013-07-09 | Takeda Pharmaceutical Company Limited | Iminopyridine derivatives and use thereof |
| AR071392A1 (es) * | 2008-04-23 | 2010-06-16 | Takeda Pharmaceutical | Derivados de iminopiridina y su uso |
-
2009
- 2009-04-21 US US12/989,379 patent/US20110039892A1/en not_active Abandoned
- 2009-04-22 EP EP09734611A patent/EP2269989A4/en not_active Withdrawn
- 2009-04-22 BR BRPI0911464A patent/BRPI0911464A2/pt not_active IP Right Cessation
- 2009-04-22 AU AU2009238999A patent/AU2009238999A1/en not_active Abandoned
- 2009-04-22 CN CN2009801239040A patent/CN102066328A/zh active Pending
- 2009-04-22 CA CA2722031A patent/CA2722031A1/en not_active Abandoned
- 2009-04-22 WO PCT/JP2009/057961 patent/WO2009131135A1/ja not_active Ceased
- 2009-04-22 EA EA201071228A patent/EA201071228A1/ru unknown
- 2009-04-22 JP JP2010509193A patent/JPWO2009131135A1/ja not_active Withdrawn
- 2009-04-22 MX MX2010011651A patent/MX2010011651A/es not_active Application Discontinuation
- 2009-04-22 KR KR1020107025981A patent/KR20110005277A/ko not_active Withdrawn
-
2010
- 2010-10-19 IL IL208824A patent/IL208824A0/en unknown
- 2010-10-22 DO DO2010000322A patent/DOP2010000322A/es unknown
- 2010-10-27 CR CR11766A patent/CR11766A/es not_active Application Discontinuation
- 2010-11-23 EC EC2010010625A patent/ECSP10010625A/es unknown
- 2010-11-23 CO CO10146698A patent/CO6260133A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0911464A2 (pt) | 2016-07-12 |
| AU2009238999A1 (en) | 2009-10-29 |
| US20110039892A1 (en) | 2011-02-17 |
| MX2010011651A (es) | 2010-12-06 |
| KR20110005277A (ko) | 2011-01-17 |
| CA2722031A1 (en) | 2009-10-29 |
| EA201071228A1 (ru) | 2011-06-30 |
| CR11766A (es) | 2010-12-15 |
| IL208824A0 (en) | 2011-01-31 |
| CO6260133A2 (es) | 2011-03-22 |
| DOP2010000322A (es) | 2011-01-31 |
| EP2269989A4 (en) | 2011-05-25 |
| CN102066328A (zh) | 2011-05-18 |
| EP2269989A1 (en) | 2011-01-05 |
| WO2009131135A1 (ja) | 2009-10-29 |
| JPWO2009131135A1 (ja) | 2011-08-18 |
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