ECSP11011433A - Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides - Google Patents
Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloidesInfo
- Publication number
- ECSP11011433A ECSP11011433A EC2011011433A ECSP11011433A ECSP11011433A EC SP11011433 A ECSP11011433 A EC SP11011433A EC 2011011433 A EC2011011433 A EC 2011011433A EC SP11011433 A ECSP11011433 A EC SP11011433A EC SP11011433 A ECSP11011433 A EC SP11011433A
- Authority
- EC
- Ecuador
- Prior art keywords
- phenilamids
- fenilures
- vanilloid
- ligands
- receiver
- Prior art date
Links
- 239000003446 ligand Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- PAYRUJLWNCNPSJ-UHFFFAOYSA-N Aniline Chemical class NC1=CC=CC=C1 PAYRUJLWNCNPSJ-UHFFFAOYSA-N 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000002483 medication Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
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- Virology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
- Cardiology (AREA)
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Abstract
La invención se refiere a derivados de fenilureas y fenilamidas sustituidas, a un procedimiento para su obtención, a medicamentos que contienen estos compuestos así como al uso de estos compuestos para la fabricación de medicamentos.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17628409P | 2009-05-07 | 2009-05-07 | |
| EP09006237 | 2009-05-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP11011433A true ECSP11011433A (es) | 2011-12-30 |
Family
ID=40908456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2011011433A ECSP11011433A (es) | 2009-05-07 | 2011-11-01 | Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US8592471B2 (es) |
| EP (1) | EP2427435B1 (es) |
| JP (1) | JP5745505B2 (es) |
| KR (1) | KR101746016B1 (es) |
| CN (2) | CN106243037A (es) |
| AR (1) | AR076752A1 (es) |
| AU (1) | AU2010244685B2 (es) |
| BR (1) | BRPI1011043B8 (es) |
| CA (1) | CA2759951C (es) |
| CO (1) | CO6440569A2 (es) |
| EC (1) | ECSP11011433A (es) |
| ES (1) | ES2640257T3 (es) |
| IL (1) | IL215661A (es) |
| MX (1) | MX2011011797A (es) |
| NZ (1) | NZ595759A (es) |
| PE (1) | PE20120374A1 (es) |
| RU (1) | RU2553392C2 (es) |
| TW (1) | TWI491595B (es) |
| WO (1) | WO2010127856A1 (es) |
| ZA (1) | ZA201107706B (es) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009067493A2 (en) * | 2007-11-19 | 2009-05-28 | Envivo Pharmaceuticals, Inc. | 1,3,5 tri-subtituted benzenes for treatment of alzheimer's disease and other disorders |
| RU2527177C2 (ru) | 2007-12-20 | 2014-08-27 | Энвиво Фармасьютикалз, Инк. | Четырехзамещенные бензолы |
| US8946204B2 (en) * | 2009-05-07 | 2015-02-03 | Gruenenthal Gmbh | Substituted phenylureas and phenylamides as vanilloid receptor ligands |
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