BRPI1011043A2 - compostos de fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, sua composição farmacêutica, seu uso e seu processo de preparação. - Google Patents

compostos de fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, sua composição farmacêutica, seu uso e seu processo de preparação.

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Publication number
BRPI1011043A2
BRPI1011043A2 BRPI1011043A BRPI1011043A BRPI1011043A2 BR PI1011043 A2 BRPI1011043 A2 BR PI1011043A2 BR PI1011043 A BRPI1011043 A BR PI1011043A BR PI1011043 A BRPI1011043 A BR PI1011043A BR PI1011043 A2 BRPI1011043 A2 BR PI1011043A2
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
preparation process
receptor ligands
phenylurea compounds
phenylamides
Prior art date
Application number
BRPI1011043A
Other languages
English (en)
Inventor
Bernhard Lesch
Gregor Bahrenberg
Jean De Vry
Jeewoo Lee
Klaus Schiene
Myeong-Seop Kim
Nils Damann
Robert Frank
Sven Frormann
Thomas Christoph
Yong-Soo Kim
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40908456&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI1011043(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of BRPI1011043A2 publication Critical patent/BRPI1011043A2/pt
Publication of BRPI1011043A8 publication Critical patent/BRPI1011043A8/pt
Publication of BRPI1011043B1 publication Critical patent/BRPI1011043B1/pt
Publication of BRPI1011043B8 publication Critical patent/BRPI1011043B8/pt

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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  • Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Anesthesiology (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
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  • Molecular Biology (AREA)
  • Gynecology & Obstetrics (AREA)
BRPI1011043A 2009-05-07 2010-05-06 fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, seus usos e seu processo de preparação, e composição farmacêutica BRPI1011043B8 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US17628409P 2009-05-07 2009-05-07
EP09006237 2009-05-07
US61/176,284 2009-05-07
EP09006237.3 2009-05-07
PCT/EP2010/002786 WO2010127856A1 (en) 2009-05-07 2010-05-06 Substituted phenyllureas and phenylamides as vanilloid receptor ligands

Publications (4)

Publication Number Publication Date
BRPI1011043A2 true BRPI1011043A2 (pt) 2016-09-13
BRPI1011043A8 BRPI1011043A8 (pt) 2017-09-12
BRPI1011043B1 BRPI1011043B1 (pt) 2020-10-13
BRPI1011043B8 BRPI1011043B8 (pt) 2021-05-25

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ID=40908456

Family Applications (1)

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BRPI1011043A BRPI1011043B8 (pt) 2009-05-07 2010-05-06 fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, seus usos e seu processo de preparação, e composição farmacêutica

Country Status (20)

Country Link
US (2) US8592471B2 (pt)
EP (1) EP2427435B1 (pt)
JP (1) JP5745505B2 (pt)
KR (1) KR101746016B1 (pt)
CN (2) CN106243037A (pt)
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US20100331381A1 (en) 2010-12-30
CO6440569A2 (es) 2012-05-15
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ECSP11011433A (es) 2011-12-30
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US20150011592A9 (en) 2015-01-08
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BRPI1011043B8 (pt) 2021-05-25
CA2759951C (en) 2017-05-02
BRPI1011043A8 (pt) 2017-09-12
KR20120034641A (ko) 2012-04-12
TWI491595B (zh) 2015-07-11
IL215661A (en) 2015-09-24
US9120756B2 (en) 2015-09-01
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CN106243037A (zh) 2016-12-21
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