ECSP14008556A - Pirimidinas y triazinas fusionadas sustituidas y su uso - Google Patents

Pirimidinas y triazinas fusionadas sustituidas y su uso

Info

Publication number
ECSP14008556A
ECSP14008556A ECIEPI20148556A ECPI201408556A ECSP14008556A EC SP14008556 A ECSP14008556 A EC SP14008556A EC IEPI20148556 A ECIEPI20148556 A EC IEPI20148556A EC PI201408556 A ECPI201408556 A EC PI201408556A EC SP14008556 A ECSP14008556 A EC SP14008556A
Authority
EC
Ecuador
Prior art keywords
triazines
substitute
prevention
treatment
fused pyrimidines
Prior art date
Application number
ECIEPI20148556A
Other languages
English (en)
Inventor
Dieter Lang
Gorden Redlich
Walter Hübsch
Nils Griebenow
Johannes-Peter Stasch
Markus Follmann
Frank Wunder
Alexandros Vakalopoulos
Adrian Tersteegen
Original Assignee
Bayer Ip Gmbh
Poli Nutri Alimentos S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47559479&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP14008556(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ip Gmbh, Poli Nutri Alimentos S A filed Critical Bayer Ip Gmbh
Publication of ECSP14008556A publication Critical patent/ECSP14008556A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente solicitud se refiere a pirimidinas y triazinas condensadas sustituidas, a procesos para su preparación, a su uso solas o en combinaciones para el tratamiento y/o la prevención de enfermedades, y a su uso para producir medicamentos para el tratamiento y/o ka prevención de enfermedades, en concreto para el tratamiento y/o la prevención de trastornos cardiovasculares.
ECIEPI20148556A 2012-01-11 2014-07-09 Pirimidinas y triazinas fusionadas sustituidas y su uso ECSP14008556A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102012200349A DE102012200349A1 (de) 2012-01-11 2012-01-11 Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung

Publications (1)

Publication Number Publication Date
ECSP14008556A true ECSP14008556A (es) 2015-12-31

Family

ID=47559479

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI20148556A ECSP14008556A (es) 2012-01-11 2014-07-09 Pirimidinas y triazinas fusionadas sustituidas y su uso

Country Status (29)

Country Link
US (2) US20140357637A1 (es)
EP (1) EP2802592A1 (es)
JP (1) JP6251183B2 (es)
KR (1) KR20140114416A (es)
CN (1) CN104812762B (es)
AP (1) AP2014007844A0 (es)
AU (1) AU2013208968A1 (es)
BR (1) BR112014016971A8 (es)
CA (1) CA2860855A1 (es)
CL (1) CL2014001779A1 (es)
CO (1) CO7000776A2 (es)
CR (1) CR20140327A (es)
CU (1) CU20140082A7 (es)
DE (1) DE102012200349A1 (es)
DO (1) DOP2014000160A (es)
EA (1) EA025837B1 (es)
EC (1) ECSP14008556A (es)
GT (1) GT201400147A (es)
HK (1) HK1211585A1 (es)
IL (1) IL233460A0 (es)
MA (1) MA35844B1 (es)
MX (1) MX2014008201A (es)
NZ (1) NZ626394A (es)
PE (1) PE20142293A1 (es)
PH (1) PH12014501595A1 (es)
SG (2) SG10201605655UA (es)
TN (1) TN2014000298A1 (es)
WO (1) WO2013104703A1 (es)
ZA (1) ZA201405042B (es)

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DE102012200360A1 (de) 2012-01-11 2013-07-11 Bayer Intellectual Property Gmbh Substituierte Triazine und ihre Verwendung
DE102012200349A1 (de) 2012-01-11 2013-07-11 Bayer Intellectual Property Gmbh Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung
ES2644781T3 (es) 2012-03-06 2017-11-30 Bayer Intellectual Property Gmbh Azabiciclos sustituidos y su uso
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HK1216890A1 (zh) 2013-03-01 2016-12-09 Bayer Pharma Aktiengesellschaft 苄基-取代的吡唑并吡啶及其用途
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AU2013208968A1 (en) 2014-07-24
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JP6251183B2 (ja) 2017-12-20
EA025837B1 (ru) 2017-02-28
US20150274754A1 (en) 2015-10-01
HK1211585A1 (en) 2016-05-27
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DE102012200349A1 (de) 2013-07-11
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AP2014007844A0 (en) 2014-07-31
CA2860855A1 (en) 2013-07-18
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KR20140114416A (ko) 2014-09-26
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US9505786B2 (en) 2016-11-29
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ZA201405042B (en) 2016-08-31
SG11201403345UA (en) 2014-09-26
BR112014016971A8 (pt) 2017-07-04
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PE20142293A1 (es) 2014-12-19
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