ECSP15032926A - Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona - Google Patents

Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Info

Publication number
ECSP15032926A
ECSP15032926A ECIEPI201532926A ECPI201532926A ECSP15032926A EC SP15032926 A ECSP15032926 A EC SP15032926A EC IEPI201532926 A ECIEPI201532926 A EC IEPI201532926A EC PI201532926 A ECPI201532926 A EC PI201532926A EC SP15032926 A ECSP15032926 A EC SP15032926A
Authority
EC
Ecuador
Prior art keywords
compounds
fungicides
dihydropyrimidin
imino
fluoro
Prior art date
Application number
ECIEPI201532926A
Other languages
English (en)
Inventor
W Owen
Beth Lorsbach
Chenglin Yao
Lindsay Stelzer
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP15032926A publication Critical patent/ECSP15032926A/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se relaciona con el campo de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1H)-onas y sus derivados y con el uso de éstos compuestos como fungicidas. Los fungicidas son compuestos, de origen natural o sintético, que actúan para proteger y/o para curar las plantas contra el daño causado por los hongos relevantes agrícolas. Generalmente, no existe un fungicida útil en todas las situaciones. Por lo tanto, la investigación está en curso para producir fungicidas que puedan tener un mejor funcionamiento, son más fáciles de usar, y cuestan menos. La presente invención se relaciona con los compuestos de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1H)-ona y su uso como fungicidas. Los compuestos de la presente invención pueden ofrecer protección contra hongos y hongos de tipo organismos incluyendo ascomicetos, basidiomicetos, deuteromicetos, y oomicetos.
ECIEPI201532926A 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona ECSP15032926A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
ECSP15032926A true ECSP15032926A (es) 2015-11-30

Family

ID=51022027

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201532926A ECSP15032926A (es) 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Country Status (18)

Country Link
US (1) US9271497B2 (es)
EP (2) EP3689142A1 (es)
JP (1) JP6336480B2 (es)
KR (1) KR20150103095A (es)
CN (1) CN104994859B (es)
AU (1) AU2013370470B2 (es)
BR (1) BR102013033840B1 (es)
CA (1) CA2893776A1 (es)
CL (1) CL2015001861A1 (es)
EC (1) ECSP15032926A (es)
GT (1) GT201500196A (es)
HK (1) HK1214518A1 (es)
IL (1) IL239562B (es)
MX (1) MX2015008443A (es)
RU (2) RU2656101C2 (es)
UA (1) UA117123C2 (es)
WO (1) WO2014105821A1 (es)
ZA (1) ZA201504195B (es)

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LT2938191T (lt) 2012-12-28 2018-05-10 Dow Agrosciences Llc Sinergistiniai fungicidiniai mišiniai, skirti grybelių kontrolei javuose
MX2015008444A (es) 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
KR102309245B1 (ko) 2012-12-31 2021-10-06 아다마 마켓심 리미티드 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체
FI3096619T3 (fi) 2013-12-31 2025-09-03 Adama Makhteshim Ltd Synergistisiä sienituhoaineseoksia sienten torjuntaan viljakasveissa
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
NZ732812A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamides and other compounds as fungicides
US20170290333A1 (en) 2014-12-30 2017-10-12 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
EP3240412A4 (en) 2014-12-30 2018-04-25 Dow Agrosciences LLC Use of picolinamide compounds with fungicidal activity
AU2015374375B2 (en) 2014-12-30 2019-03-21 Dow Agrosciences Llc Picolinamides with fungicidal activity
CA2972408A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
US11639334B2 (en) 2018-10-15 2023-05-02 Corteva Agriscience Llc Methods for synthesis of oxypicolinamides
US12414559B2 (en) 2018-11-05 2025-09-16 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
WO2021059160A1 (en) 2019-09-23 2021-04-01 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

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Also Published As

Publication number Publication date
JP6336480B2 (ja) 2018-06-06
RU2656101C2 (ru) 2018-05-31
IL239562A0 (en) 2015-08-31
CN104994859B (zh) 2018-10-26
AU2013370470B2 (en) 2018-05-10
RU2018118951A (ru) 2018-11-02
CN104994859A (zh) 2015-10-21
US9271497B2 (en) 2016-03-01
GT201500196A (es) 2016-03-02
AU2013370470A1 (en) 2015-07-02
EP3689142A1 (en) 2020-08-05
WO2014105821A1 (en) 2014-07-03
JP2016509589A (ja) 2016-03-31
CL2015001861A1 (es) 2015-10-02
IL239562B (en) 2018-02-28
BR102013033840B1 (pt) 2019-09-10
ZA201504195B (en) 2017-08-30
BR102013033840A2 (pt) 2015-10-06
RU2018118951A3 (es) 2019-02-26
RU2015131110A (ru) 2017-02-03
MX2015008443A (es) 2015-09-23
EP2945635A4 (en) 2016-05-25
HK1216147A1 (zh) 2016-10-21
EP2945635A1 (en) 2015-11-25
CA2893776A1 (en) 2014-07-03
US20150342188A1 (en) 2015-12-03
UA117123C2 (uk) 2018-06-25
HK1214518A1 (zh) 2016-07-29
KR20150103095A (ko) 2015-09-09

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