ECSP21093576A - Agonistas del receptor del péptido-1 similar al glucagón - Google Patents

Agonistas del receptor del péptido-1 similar al glucagón

Info

Publication number
ECSP21093576A
ECSP21093576A ECSENADI202193576A ECDI202193576A ECSP21093576A EC SP21093576 A ECSP21093576 A EC SP21093576A EC SENADI202193576 A ECSENADI202193576 A EC SENADI202193576A EC DI202193576 A ECDI202193576 A EC DI202193576A EC SP21093576 A ECSP21093576 A EC SP21093576A
Authority
EC
Ecuador
Prior art keywords
glucagon
peptide
receptor agonists
agonists
receptor
Prior art date
Application number
ECSENADI202193576A
Other languages
English (en)
Inventor
Todd Fields
Fucheng Qu
David Andrew Coates
Joseph Daniel Ho
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of ECSP21093576A publication Critical patent/ECSP21093576A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se adjunta resumen de la invención
ECSENADI202193576A 2019-06-28 2021-12-28 Agonistas del receptor del péptido-1 similar al glucagón ECSP21093576A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962868117P 2019-06-28 2019-06-28
US201962904906P 2019-09-24 2019-09-24

Publications (1)

Publication Number Publication Date
ECSP21093576A true ECSP21093576A (es) 2022-01-31

Family

ID=71575804

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI202193576A ECSP21093576A (es) 2019-06-28 2021-12-28 Agonistas del receptor del péptido-1 similar al glucagón

Country Status (34)

Country Link
US (3) US11655242B2 (es)
EP (2) EP3989972B1 (es)
JP (1) JP7256300B2 (es)
KR (1) KR102738278B1 (es)
CN (1) CN114008033B (es)
AU (1) AU2020309064B2 (es)
CA (1) CA3144055C (es)
CL (1) CL2021003419A1 (es)
CO (1) CO2021017433A2 (es)
CR (1) CR20210599A (es)
DK (1) DK3989972T3 (es)
DO (1) DOP2021000273A (es)
EC (1) ECSP21093576A (es)
ES (1) ES2970173T3 (es)
FI (1) FI3989972T3 (es)
HR (1) HRP20231586T1 (es)
HU (1) HUE065080T2 (es)
IL (2) IL322973A (es)
JO (1) JOP20210337B1 (es)
LT (1) LT3989972T (es)
MD (1) MD3989972T2 (es)
MX (1) MX2021015328A (es)
MY (1) MY198745A (es)
PE (1) PE20220590A1 (es)
PH (1) PH12021553251A1 (es)
PL (1) PL3989972T3 (es)
PT (1) PT3989972T (es)
RS (1) RS64940B1 (es)
SA (1) SA521431209B1 (es)
SI (1) SI3989972T1 (es)
TW (1) TWI751585B (es)
UA (1) UA130869C2 (es)
WO (1) WO2020263695A1 (es)
ZA (1) ZA202109587B (es)

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KR102563111B1 (ko) * 2020-03-18 2023-08-04 주식회사 엘지화학 Glp-1 수용체 효능제, 이를 포함하는 약학적 조성물 및 이의 제조방법
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KR20240053617A (ko) 2021-08-30 2024-04-24 민드랭크 에이아이 리미티드 Glp1r 작용제로서의 신규 아릴 에테르 치환 헤테로시클릭 화합물
KR20240056719A (ko) 2021-09-08 2024-04-30 시오노기 앤드 컴파니, 리미티드 항비만 작용이 관여하는 질환의 예방 및 치료용 의약
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Also Published As

Publication number Publication date
CR20210599A (es) 2021-12-22
IL288479A (en) 2022-01-01
CA3144055C (en) 2024-01-02
KR102738278B1 (ko) 2024-12-06
NZ783212A (en) 2025-03-28
EP3989972A1 (en) 2022-05-04
SI3989972T1 (sl) 2024-01-31
US20200407347A1 (en) 2020-12-31
CL2021003419A1 (es) 2022-09-23
HUE065080T2 (hu) 2024-04-28
UA130869C2 (uk) 2026-06-03
WO2020263695A1 (en) 2020-12-30
EP4302826A3 (en) 2024-04-17
IL288479B2 (en) 2026-08-01
IL322973A (en) 2025-10-01
BR112021023923A2 (pt) 2022-01-25
JOP20210337A1 (ar) 2023-01-30
EP3989972B1 (en) 2023-11-08
PH12021553251A1 (en) 2022-09-05
MD3989972T2 (ro) 2024-05-31
US20230250092A1 (en) 2023-08-10
ZA202109587B (en) 2024-07-31
US20250002482A1 (en) 2025-01-02
SA521431209B1 (ar) 2024-08-05
US11655242B2 (en) 2023-05-23
IL288479B1 (en) 2026-04-01
CN114008033B (zh) 2025-01-10
JOP20210337B1 (ar) 2024-04-18
ES2970173T3 (es) 2024-05-27
KR20220012924A (ko) 2022-02-04
TWI751585B (zh) 2022-01-01
CO2021017433A2 (es) 2022-04-19
MY198745A (en) 2023-09-21
PT3989972T (pt) 2023-12-04
PE20220590A1 (es) 2022-04-22
LT3989972T (lt) 2023-12-27
HRP20231586T1 (hr) 2024-03-15
RS64940B1 (sr) 2024-01-31
PL3989972T3 (pl) 2024-03-25
EP4302826A2 (en) 2024-01-10
TW202115040A (zh) 2021-04-16
AU2020309064B2 (en) 2023-08-17
DOP2021000273A (es) 2022-03-15
JP7256300B2 (ja) 2023-04-11
MX2021015328A (es) 2022-01-18
AU2020309064A1 (en) 2022-01-27
CN114008033A (zh) 2022-02-01
CA3144055A1 (en) 2020-12-30
DK3989972T3 (da) 2023-12-04
FI3989972T3 (fi) 2024-01-24
JP2022540044A (ja) 2022-09-14

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