ECSP22046595A - Procesos e intermediario para la preparaci?n de oxetan-2-ilmetanamina - Google Patents
Procesos e intermediario para la preparaci?n de oxetan-2-ilmetanaminaInfo
- Publication number
- ECSP22046595A ECSP22046595A ECSENADI202246595A ECDI202246595A ECSP22046595A EC SP22046595 A ECSP22046595 A EC SP22046595A EC SENADI202246595 A ECSENADI202246595 A EC SENADI202246595A EC DI202246595 A ECDI202246595 A EC DI202246595A EC SP22046595 A ECSP22046595 A EC SP22046595A
- Authority
- EC
- Ecuador
- Prior art keywords
- preparation
- ilmethanamine
- oxetan
- processes
- salt
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/02—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D305/04—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D305/06—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Un proceso e intermediario para la preparaci?n de un compuesto de f?rmula I: o una sal del mismo.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962946146P | 2019-12-10 | 2019-12-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP22046595A true ECSP22046595A (es) | 2022-07-29 |
Family
ID=74003942
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSENADI202246595A ECSP22046595A (es) | 2019-12-10 | 2022-06-10 | Procesos e intermediario para la preparaci?n de oxetan-2-ilmetanamina |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US12473267B2 (es) |
| EP (1) | EP4073051B1 (es) |
| JP (1) | JP7292517B2 (es) |
| KR (1) | KR102635237B1 (es) |
| CN (1) | CN114728923B (es) |
| AU (1) | AU2020401539B2 (es) |
| CL (1) | CL2022001511A1 (es) |
| CO (1) | CO2022008127A2 (es) |
| DK (1) | DK4073051T3 (es) |
| EC (1) | ECSP22046595A (es) |
| ES (1) | ES2975599T3 (es) |
| FI (1) | FI4073051T3 (es) |
| HR (1) | HRP20240343T1 (es) |
| HU (1) | HUE067201T2 (es) |
| IL (1) | IL292707B2 (es) |
| LT (1) | LT4073051T (es) |
| MA (1) | MA58104B1 (es) |
| MD (1) | MD4073051T2 (es) |
| MX (1) | MX2022006984A (es) |
| PE (1) | PE20230183A1 (es) |
| PH (1) | PH12022551403A1 (es) |
| PL (1) | PL4073051T3 (es) |
| PT (1) | PT4073051T (es) |
| RS (1) | RS65238B1 (es) |
| SI (1) | SI4073051T1 (es) |
| UA (1) | UA127884C2 (es) |
| WO (1) | WO2021118906A1 (es) |
| ZA (1) | ZA202205170B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI4073051T1 (sl) | 2019-12-10 | 2024-04-30 | Eli Lilly And Company | Postopek in intermediat za pripravo oksetan-2-ilmetanamina |
| CN116217522B (zh) * | 2023-02-22 | 2025-06-24 | 广东莱佛士制药技术有限公司 | Glp-1受体激动剂关键中间体的手性纯化方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7208140B2 (en) * | 2003-02-19 | 2007-04-24 | Schering Aktiengesellschaft | Trimeric macrocyclic substituted benzene derivatives |
| UA114601C2 (uk) * | 2011-05-06 | 2017-07-10 | Егіш Дьйодьсердьяр Нільваношан Мюкеде Ресвеньтаршашаг | Спосіб одержання ривароксабану та проміжних сполук, які одержано в даному способі |
| EP2847177B1 (en) * | 2012-05-09 | 2017-10-11 | Boehringer Ingelheim International GmbH | Methods for making oxetan-3-ylmethanamines |
| KR102314286B1 (ko) * | 2016-12-16 | 2021-10-21 | 화이자 인코포레이티드 | Glp-1 수용체 작용제 및 이의 용도 |
| TWI707683B (zh) | 2018-06-13 | 2020-10-21 | 美商輝瑞股份有限公司 | Glp-1受體促效劑及其用途 |
| RU2765721C1 (ru) | 2018-06-15 | 2022-02-02 | Пфайзер Инк. | Агонисты glp-1 рецептора и их применение |
| CN109265389B (zh) * | 2018-08-31 | 2020-08-18 | 南京富润凯德生物医药有限公司 | 2-(氨基甲基)-1-氧杂-7-氮杂螺[3.5]壬烷衍生物、中间体及其制备方法 |
| SI4073051T1 (sl) | 2019-12-10 | 2024-04-30 | Eli Lilly And Company | Postopek in intermediat za pripravo oksetan-2-ilmetanamina |
-
2020
- 2020-12-07 SI SI202030381T patent/SI4073051T1/sl unknown
- 2020-12-07 JP JP2022534655A patent/JP7292517B2/ja active Active
- 2020-12-07 HR HRP20240343TT patent/HRP20240343T1/hr unknown
- 2020-12-07 MX MX2022006984A patent/MX2022006984A/es unknown
- 2020-12-07 PH PH1/2022/551403A patent/PH12022551403A1/en unknown
- 2020-12-07 KR KR1020227018626A patent/KR102635237B1/ko active Active
- 2020-12-07 EP EP20829133.6A patent/EP4073051B1/en active Active
- 2020-12-07 PT PT208291336T patent/PT4073051T/pt unknown
- 2020-12-07 US US17/779,447 patent/US12473267B2/en active Active
- 2020-12-07 MA MA58104A patent/MA58104B1/fr unknown
- 2020-12-07 MD MDE20221148T patent/MD4073051T2/ro unknown
- 2020-12-07 HU HUE20829133A patent/HUE067201T2/hu unknown
- 2020-12-07 WO PCT/US2020/063546 patent/WO2021118906A1/en not_active Ceased
- 2020-12-07 UA UAA202201389A patent/UA127884C2/uk unknown
- 2020-12-07 DK DK20829133.6T patent/DK4073051T3/da active
- 2020-12-07 CN CN202080082957.9A patent/CN114728923B/zh active Active
- 2020-12-07 ES ES20829133T patent/ES2975599T3/es active Active
- 2020-12-07 FI FIEP20829133.6T patent/FI4073051T3/fi active
- 2020-12-07 PE PE2022001046A patent/PE20230183A1/es unknown
- 2020-12-07 IL IL292707A patent/IL292707B2/en unknown
- 2020-12-07 RS RS20240243A patent/RS65238B1/sr unknown
- 2020-12-07 PL PL20829133.6T patent/PL4073051T3/pl unknown
- 2020-12-07 AU AU2020401539A patent/AU2020401539B2/en active Active
- 2020-12-07 LT LTEPPCT/US2020/063546T patent/LT4073051T/lt unknown
-
2022
- 2022-05-10 ZA ZA2022/05170A patent/ZA202205170B/en unknown
- 2022-06-08 CL CL2022001511A patent/CL2022001511A1/es unknown
- 2022-06-08 CO CONC2022/0008127A patent/CO2022008127A2/es unknown
- 2022-06-10 EC ECSENADI202246595A patent/ECSP22046595A/es unknown
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