EE200300033A - Tsüklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon - Google Patents

Tsüklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Info

Publication number
EE200300033A
EE200300033A EEP200300033A EEP200300033A EE200300033A EE 200300033 A EE200300033 A EE 200300033A EE P200300033 A EEP200300033 A EE P200300033A EE P200300033 A EEP200300033 A EE P200300033A EE 200300033 A EE200300033 A EE 200300033A
Authority
EE
Estonia
Prior art keywords
cyclopentanoindoles
medicament
preparation
pharmaceutical composition
composition containing
Prior art date
Application number
EEP200300033A
Other languages
English (en)
Inventor
Labelle Marc
Sturino Claudio
Roy Bruno
Berthelette Carl
Boyd Michael
Lachance Nicolas
Scheigetz John
Original Assignee
Merck Frosst Canada & Co.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Frosst Canada & Co. filed Critical Merck Frosst Canada & Co.
Publication of EE200300033A publication Critical patent/EE200300033A/et
Publication of EE05287B1 publication Critical patent/EE05287B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/38TPC being performed in particular situations
    • H04W52/46TPC being performed in particular situations in multi-hop networks, e.g. wireless relay networks
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/94[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/02Access restriction performed under specific conditions
    • H04W48/04Access restriction performed under specific conditions based on user or terminal location or mobility data, e.g. moving direction, speed
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/06TPC algorithms
    • H04W52/14Separate analysis of uplink or downlink
    • H04W52/146Uplink power control
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/28TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission
    • H04W52/288TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non-transmission taking into account the usage mode, e.g. hands-free, data transmission or telephone
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W48/00Access restriction; Network selection; Access point selection
    • H04W48/20Selecting an access point
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/245TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters taking into account received signal strength
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04WWIRELESS COMMUNICATION NETWORKS
    • H04W52/00Power management, e.g. Transmission Power Control [TPC] or power classes
    • H04W52/04Transmission power control [TPC]
    • H04W52/18TPC being performed according to specific parameters
    • H04W52/24TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
    • H04W52/247TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters where the output power of a terminal is based on a path parameter sent by another terminal

Landscapes

  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Signal Processing (AREA)
  • Computer Networks & Wireless Communication (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Computer Security & Cryptography (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Steroid Compounds (AREA)
  • Materials For Photolithography (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
EEP200300033A 2000-07-25 2001-07-23 Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon EE05287B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22068300P 2000-07-25 2000-07-25
PCT/CA2001/001069 WO2002008186A2 (en) 2000-07-25 2001-07-23 Cyclopentanoindoles, compositions containing such compounds and methods of treatment

Publications (2)

Publication Number Publication Date
EE200300033A true EE200300033A (et) 2004-10-15
EE05287B1 EE05287B1 (et) 2010-04-15

Family

ID=22824535

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300033A EE05287B1 (et) 2000-07-25 2001-07-23 Tsklopentanoindoolid, nende kasutamine ravimi valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Country Status (33)

Country Link
US (1) US6410583B1 (et)
EP (1) EP1305286B1 (et)
JP (1) JP4119745B2 (et)
KR (1) KR100746814B1 (et)
CN (1) CN1214007C (et)
AT (1) ATE284388T1 (et)
AU (2) AU2001277430B2 (et)
BG (1) BG66084B1 (et)
BR (1) BR0112756A (et)
CA (1) CA2416867C (et)
CZ (1) CZ2003236A3 (et)
DE (1) DE60107687T2 (et)
DK (1) DK1305286T3 (et)
DZ (1) DZ3402A1 (et)
EA (1) EA006765B1 (et)
EC (1) ECSP034428A (et)
EE (1) EE05287B1 (et)
ES (1) ES2231526T3 (et)
GE (1) GEP20053595B (et)
HR (1) HRP20021039B1 (et)
HU (1) HUP0301745A3 (et)
IL (2) IL153406A0 (et)
IS (1) IS2170B (et)
MX (1) MXPA03000710A (et)
NO (1) NO325011B1 (et)
NZ (1) NZ523106A (et)
PL (1) PL207342B1 (et)
PT (1) PT1305286E (et)
RS (1) RS50491B (et)
SK (1) SK287507B6 (et)
UA (1) UA73787C2 (et)
WO (1) WO2002008186A2 (et)
ZA (1) ZA200300554B (et)

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US6784172B2 (en) 2000-11-03 2004-08-31 Wyeth Processes for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
AR031199A1 (es) 2000-11-03 2003-09-10 Wyeth Corp Ciclohepta/b//1,4/diacepino/6,7,1-hi/indoles y derivados
US6759405B2 (en) 2000-11-03 2004-07-06 Wyeth Cycloocta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
US6777407B2 (en) 2000-11-03 2004-08-17 Wyeth Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
AR038136A1 (es) * 2002-01-24 2004-12-29 Merck Frosst Canada Inc Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento
TW200307540A (en) 2002-04-25 2003-12-16 Wyeth Corp [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents
TW200307682A (en) 2002-04-25 2003-12-16 Wyeth Corp 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
TWI312781B (en) 2002-04-25 2009-08-01 [1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
TW200400963A (en) 2002-05-21 2004-01-16 Wyeth Corp R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease
TW200400818A (en) 2002-05-21 2004-01-16 Wyeth Corp Method for the use of pyranoindole derivatives to treat infection with hepatitis C virus
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AU2004240705A1 (en) * 2003-05-20 2004-12-02 Merck Frosst Canada & Co. Fluoro-methanesulfonyl-substituted cycloalkanoindoles and their use as prostaglandin D2 antagonists
CA2527773A1 (en) * 2003-06-12 2004-12-23 Merck Frosst Canada Ltd. Cycloalkanepyrrolopyridines as dp receptor antagonists
US20080153817A1 (en) * 2003-08-07 2008-06-26 Dirk Beher Treatment for Alzheimer's Disease and Related Conditions
US20050107350A1 (en) * 2003-08-22 2005-05-19 Pharmacia Corporation Method for the treatment or prevention of bone disorders with a cyclooxygenase-2 inhibitor alone and in combination with a bone disorder treatment agent and compositions therewith
PE20050483A1 (es) 2003-10-31 2005-08-25 Arena Pharm Inc Derivados de tetrazol de formula (i), sus composiciones farmaceuticas y procesos para producir composiciones farmaceuticas
US7019022B2 (en) * 2003-12-15 2006-03-28 Merck Frosst Canada & Co. Substituted tetrahydrocarbazole and cyclopentanoindole derivatives
WO2006008119A1 (en) 2004-07-16 2006-01-26 Proteosys Ag Muscarinic antagonists with parp and sir modulatng activity as agents for inflammatory diseases
HN2005000795A (es) * 2004-10-15 2010-08-19 Aventis Pharma Inc Pirimidinas como antagonistas del receptor de prostaglandina d2
GT200500317A (es) 2004-11-05 2006-10-27 Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos
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US20100260841A1 (en) * 2007-02-08 2010-10-14 Paolini John F Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions
EA019252B1 (ru) 2008-07-23 2014-02-28 Арена Фармасьютикалз, Инк. ЗАМЕЩЕННЫЕ ПРОИЗВОДНЫЕ (1,2,3,4-ТЕТРАГИДРОЦИКЛОПЕНТА[b]ИНДОЛ-3-ИЛ)УКСУСНОЙ КИСЛОТЫ, ПРИМЕНИМЫЕ В ЛЕЧЕНИИ АУТОИММУННЫХ И ВОСПАЛИТЕЛЬНЫХ РАССТРОЙСТВ
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Also Published As

Publication number Publication date
JP4119745B2 (ja) 2008-07-16
BR0112756A (pt) 2003-06-24
UA73787C2 (en) 2005-09-15
PL207342B1 (pl) 2010-12-31
SK932003A3 (en) 2003-06-03
HUP0301745A3 (en) 2010-03-29
NO20030374L (no) 2003-01-24
EA200300171A1 (ru) 2003-06-26
HRP20021039B1 (hr) 2011-03-31
ES2231526T3 (es) 2005-05-16
CN1443165A (zh) 2003-09-17
CA2416867A1 (en) 2002-01-31
CN1214007C (zh) 2005-08-10
AU2001277430B2 (en) 2006-05-25
WO2002008186A3 (en) 2002-03-21
KR20030024810A (ko) 2003-03-26
HUP0301745A2 (hu) 2003-09-29
PL363168A1 (pl) 2004-11-15
PT1305286E (pt) 2005-04-29
CZ2003236A3 (cs) 2003-05-14
IL153406A (en) 2008-03-20
EP1305286B1 (en) 2004-12-08
AU7743001A (en) 2002-02-05
EA006765B1 (ru) 2006-04-28
HK1058934A1 (en) 2004-06-11
IL153406A0 (en) 2003-07-06
BG107438A (bg) 2003-09-30
ATE284388T1 (de) 2004-12-15
ECSP034428A (es) 2003-03-10
GEP20053595B (en) 2005-08-10
DE60107687D1 (de) 2005-01-13
KR100746814B1 (ko) 2007-08-06
RS50491B (sr) 2010-03-02
ZA200300554B (en) 2004-04-23
IS2170B (is) 2006-11-15
WO2002008186A2 (en) 2002-01-31
NZ523106A (en) 2005-01-28
DE60107687T2 (de) 2005-12-01
SK287507B6 (sk) 2010-12-07
CA2416867C (en) 2008-03-25
BG66084B1 (bg) 2011-03-31
US6410583B1 (en) 2002-06-25
HRP20021039A2 (en) 2004-10-31
YU97902A (sh) 2006-05-25
IS6655A (is) 2002-12-12
DK1305286T3 (da) 2005-03-14
DZ3402A1 (fr) 2002-01-31
EP1305286A2 (en) 2003-05-02
NO325011B1 (no) 2008-01-14
EE05287B1 (et) 2010-04-15
NO20030374D0 (no) 2003-01-24
MXPA03000710A (es) 2003-06-04
JP2004504380A (ja) 2004-02-12

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