ES2001923A6 - Procedimiento para preparar 3-amino-dihidro-(1)-benzo(tio)piranos. - Google Patents
Procedimiento para preparar 3-amino-dihidro-(1)-benzo(tio)piranos.Info
- Publication number
- ES2001923A6 ES2001923A6 ES8601568A ES8601568A ES2001923A6 ES 2001923 A6 ES2001923 A6 ES 2001923A6 ES 8601568 A ES8601568 A ES 8601568A ES 8601568 A ES8601568 A ES 8601568A ES 2001923 A6 ES2001923 A6 ES 2001923A6
- Authority
- ES
- Spain
- Prior art keywords
- amino
- formula
- benzothiopyrane
- benzopyrane
- dihydro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- ONJRTQUWKRDCTA-UHFFFAOYSA-N 2h-thiochromene Chemical compound C1=CC=C2C=CCSC2=C1 ONJRTQUWKRDCTA-UHFFFAOYSA-N 0.000 title 1
- SVWDNDQOXZHBRM-UHFFFAOYSA-N 3,4-dihydro-2h-chromen-3-amine Chemical compound C1=CC=C2CC(N)COC2=C1 SVWDNDQOXZHBRM-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 230000005494 condensation Effects 0.000 abstract 1
- 238000009833 condensation Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 150000004880 oxines Chemical class 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/74—Benzo[b]pyrans, hydrogenated in the carbocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
- C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D335/06—Benzothiopyrans; Hydrogenated benzothiopyrans
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrane Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Dental Preparations (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR 3-AMINO-DIHIDRO1-BENZO(TIO)PIRANOS DE FORMULA GENERAL EN LA QUE R1 A R5 Y Z TIENEN EL SIGNIFICADO DADO EN LA DESCRIPCION POR CONDENSACION DE UN COMPUESTO DE FORMULA II CON UN COMPUESTO DE FORMULA III DONDE R1 A R5 Y Z TIENEN EL SIGNIFICADO ANTERIORMENTE INDICADO Y X TIENE EL SIGNIFICADO DADO EN LA DESCRIPCION. ESTOS COMPUESTOS DE FORMULA I TIENEN UTILIDAD COMO MODULADORES DE RECEPTORES DEL SISTEMA NERVIOSO CENTRAL.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77206885A | 1985-09-03 | 1985-09-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2001923A6 true ES2001923A6 (es) | 1988-07-01 |
Family
ID=25093804
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES8601568A Expired ES2001923A6 (es) | 1985-09-03 | 1986-09-02 | Procedimiento para preparar 3-amino-dihidro-(1)-benzo(tio)piranos. |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP0222996B1 (es) |
| JP (1) | JPS6259273A (es) |
| KR (1) | KR900003883B1 (es) |
| AT (1) | ATE63744T1 (es) |
| AU (1) | AU596113B2 (es) |
| DD (1) | DD249480A5 (es) |
| DE (1) | DE3679378D1 (es) |
| DK (1) | DK418486A (es) |
| ES (1) | ES2001923A6 (es) |
| FI (1) | FI86720C (es) |
| GR (1) | GR862239B (es) |
| HU (1) | HU202853B (es) |
| IL (1) | IL79920A (es) |
| NO (1) | NO863507L (es) |
| NZ (1) | NZ217432A (es) |
| PH (1) | PH22522A (es) |
| PT (1) | PT83300B (es) |
| ZA (1) | ZA866685B (es) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4957928A (en) * | 1986-06-26 | 1990-09-18 | Ciba-Geigy Corporation | Hydrogenated 1-benzooxacycloalkylpyridinecarboxylic acid compounds |
| US4801605A (en) * | 1986-08-29 | 1989-01-31 | Ciba-Geigy Corporation | 3-amino-dihydro-[1]-benzopyrans and benzothiopyrans |
| SE8605504D0 (sv) * | 1986-12-19 | 1986-12-19 | Astra Laekemedel Ab | Novel chroman derivatives |
| EP0322361A3 (de) * | 1987-12-23 | 1990-01-24 | Ciba-Geigy Ag | Weitere hydrierte 1-Benzooxacycloalkylpyridincarbonsäureverbindungen |
| AU631588B2 (en) * | 1988-12-23 | 1992-12-03 | Beecham Group Plc | Benzopyran derivatives and related compounds |
| WO1990012795A1 (en) * | 1989-04-27 | 1990-11-01 | The Upjohn Company | Substituted 3-amino chromans |
| SE8904127D0 (sv) * | 1989-12-07 | 1989-12-07 | Astra Ab | New biocyclic amino-substituted compounds |
| SE8904361D0 (sv) * | 1989-12-22 | 1989-12-22 | Astra Ab | New chroman and thiochroman derivatives |
| US5616610A (en) * | 1989-12-22 | 1997-04-01 | Astra Aktiebolag | (R)-5-carbamoyl-8-fluoro-3-N,N-disubstituted-amino-3,4-dihydro-2H-1-benzopyrans |
| US5420151A (en) * | 1989-12-22 | 1995-05-30 | Aktiebolaget Astra | Chroman derivatives |
| FR2660657B1 (fr) * | 1990-04-09 | 1993-05-07 | Adir | Nouveaux derives du 3-aminochromane, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US5273994A (en) * | 1990-04-09 | 1993-12-28 | Adir Et Compagnie | 3-aminochroman compounds |
| FR2678617B1 (fr) * | 1991-07-01 | 1995-01-20 | Adir | Nouveau procede de synthese d'enantiomeres de derives du 3-amino chromane. |
| FR2681325B1 (fr) * | 1991-09-16 | 1993-12-17 | Fabre Medicament Pierre | Derives de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique. |
| HRP920935A2 (en) * | 1991-10-08 | 1995-08-31 | Astra Ab | New therapeutically active compound |
| FR2689509B1 (fr) * | 1992-04-01 | 1994-06-03 | Adir | Nouveaux derives spiraniques du 3-amino chromane, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent. |
| CZ282172B6 (cs) * | 1992-11-30 | 1997-05-14 | Smithkline Beecham Plc | Benzpyranové analogy pro léčení úzkosti, mánie, deprese nebo symptomů po přerušení podávání drog nebo léčiv, způsob přípravy těchto sloučenin, jejich použití a farmaceutický prostředek obsahující tyto sloučeniny |
| US7125904B2 (en) | 2002-10-11 | 2006-10-24 | Portela & C.A., S.A. | Peripherally-selective inhibitors of dopamine-β-hydroxylase and method of their preparation |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3607886A (en) * | 1969-04-24 | 1971-09-21 | Parke Davis & Co | Chromanamines |
| US3629289A (en) * | 1969-04-24 | 1971-12-21 | Parke Davis & Co | Chromanamines |
| US4203895A (en) * | 1978-04-14 | 1980-05-20 | Warner-Lambert Company | Process for the preparation of cis-(±)-3,4-dihydro-N,N,2-trimethyl-2H-1-benzopyran-3-amine and intermediates produced thereby |
-
1986
- 1986-09-01 GR GR862239A patent/GR862239B/el unknown
- 1986-09-01 DE DE8686112104T patent/DE3679378D1/de not_active Expired - Lifetime
- 1986-09-01 PH PH34204A patent/PH22522A/en unknown
- 1986-09-01 AT AT86112104T patent/ATE63744T1/de not_active IP Right Cessation
- 1986-09-01 EP EP86112104A patent/EP0222996B1/de not_active Expired - Lifetime
- 1986-09-02 HU HU863786A patent/HU202853B/hu not_active IP Right Cessation
- 1986-09-02 ZA ZA866685A patent/ZA866685B/xx unknown
- 1986-09-02 IL IL79920A patent/IL79920A/xx unknown
- 1986-09-02 DK DK418486A patent/DK418486A/da unknown
- 1986-09-02 NZ NZ217432A patent/NZ217432A/xx unknown
- 1986-09-02 DD DD86294093A patent/DD249480A5/de not_active IP Right Cessation
- 1986-09-02 ES ES8601568A patent/ES2001923A6/es not_active Expired
- 1986-09-02 NO NO863507A patent/NO863507L/no unknown
- 1986-09-03 PT PT83300A patent/PT83300B/pt not_active IP Right Cessation
- 1986-09-03 KR KR1019860007357A patent/KR900003883B1/ko not_active Expired
- 1986-09-03 AU AU62317/86A patent/AU596113B2/en not_active Ceased
- 1986-09-03 FI FI863558A patent/FI86720C/fi not_active IP Right Cessation
- 1986-09-03 JP JP61206047A patent/JPS6259273A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FI863558A0 (fi) | 1986-09-03 |
| EP0222996A3 (en) | 1987-12-02 |
| EP0222996A2 (de) | 1987-05-27 |
| DE3679378D1 (de) | 1991-06-27 |
| PT83300B (pt) | 1989-05-12 |
| PT83300A (en) | 1986-10-01 |
| NO863507D0 (no) | 1986-09-02 |
| KR900003883B1 (ko) | 1990-06-04 |
| DK418486A (da) | 1987-03-04 |
| ATE63744T1 (de) | 1991-06-15 |
| PH22522A (en) | 1988-10-17 |
| FI86720C (fi) | 1992-10-12 |
| AU596113B2 (en) | 1990-04-26 |
| NO863507L (no) | 1987-03-04 |
| ZA866685B (en) | 1987-04-29 |
| FI863558A7 (fi) | 1987-03-04 |
| HU202853B (en) | 1991-04-29 |
| GR862239B (en) | 1986-12-31 |
| EP0222996B1 (de) | 1991-05-22 |
| HUT44771A (en) | 1988-04-28 |
| FI86720B (fi) | 1992-06-30 |
| IL79920A (en) | 1991-07-18 |
| KR870003088A (ko) | 1987-04-15 |
| JPS6259273A (ja) | 1987-03-14 |
| AU6231786A (en) | 1987-03-05 |
| NZ217432A (en) | 1990-03-27 |
| DK418486D0 (da) | 1986-09-02 |
| DD249480A5 (de) | 1987-09-09 |
| IL79920A0 (en) | 1986-12-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| SA6 | Expiration date (snapshot 920101) |
Free format text: 2006-09-02 |
|
| FD1A | Patent lapsed |
Effective date: 20001102 |