ES2044910T3 - Procedimiento de preparacion de derivados de n-(metilsulfonilfenil-etil)-2-propenamidas. - Google Patents

Procedimiento de preparacion de derivados de n-(metilsulfonilfenil-etil)-2-propenamidas.

Info

Publication number
ES2044910T3
ES2044910T3 ES87119048T ES87119048T ES2044910T3 ES 2044910 T3 ES2044910 T3 ES 2044910T3 ES 87119048 T ES87119048 T ES 87119048T ES 87119048 T ES87119048 T ES 87119048T ES 2044910 T3 ES2044910 T3 ES 2044910T3
Authority
ES
Spain
Prior art keywords
etil
derivatives
metilsulfonilpenil
propenamides
preparation procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87119048T
Other languages
English (en)
Inventor
Bella Davide Della
Giancarlo Jommi
Mario Fantucci
Dario Chiarino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Zambon SpA
Original Assignee
Zambon SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon SpA filed Critical Zambon SpA
Application granted granted Critical
Publication of ES2044910T3 publication Critical patent/ES2044910T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

SE DESCRIBE EL COMPUESTO N-[(1S, 2R)-1-FLUOROMETIL-2-HIDROXI2-(4-METILSULFONIL)-FENIL)-ETIL]-2-PROPENAMIDA Y LOS DERIVADOS DE LA MISMA, EN DONDE EL HIDROXI EN LA POSICION 2 ESTA ESTERIFICADO POR UN ACIDO MONO O DICARBOXILICO O POR UN AMINOACIDO. TALES COMPUESTOS TIENEN ACTIVIDAD ANTIBIOTICA, Y SON UTILES EN TERAPIA HUMANA Y VETERINARIA.
ES87119048T 1986-12-23 1987-12-22 Procedimiento de preparacion de derivados de n-(metilsulfonilfenil-etil)-2-propenamidas. Expired - Lifetime ES2044910T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT22826/86A IT1198238B (it) 1986-12-23 1986-12-23 Composti ad attivita' antibiotica

Publications (1)

Publication Number Publication Date
ES2044910T3 true ES2044910T3 (es) 1994-01-16

Family

ID=11200890

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87119048T Expired - Lifetime ES2044910T3 (es) 1986-12-23 1987-12-22 Procedimiento de preparacion de derivados de n-(metilsulfonilfenil-etil)-2-propenamidas.

Country Status (8)

Country Link
US (1) US4918095A (es)
EP (1) EP0272684B1 (es)
JP (1) JPS63190870A (es)
AT (1) ATE64379T1 (es)
DE (1) DE3770788D1 (es)
ES (1) ES2044910T3 (es)
GR (1) GR3002135T3 (es)
IT (1) IT1198238B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5243056A (en) * 1983-06-02 1993-09-07 Zambon S.P.A. Intermediates for the preparation of 1-(phenyl)-1-hydroxy-2-amino-3-fluoro propane derivatives
US5332835A (en) * 1984-02-03 1994-07-26 Zambon S.P.A. Process for fluorinating 1-phenyl-2-amino-1,3-propanediol compounds and new oxazoline compounds useful in this process
US5153328A (en) * 1984-02-03 1992-10-06 Zambon S.P.A. 2 Hydrocarbyl-4 substituted methyl 5 (4 substituted phenyl)-oxazolines
CN1649829A (zh) * 2002-03-08 2005-08-03 先灵-普劳有限公司 新型氟苯尼考类抗生素
DE102004037173B3 (de) * 2004-07-30 2005-12-15 Bruker Biospin Ag Vorrichtung zur kryogenverlustfreien Kühlung einer Kryostatanordnung
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
WO2008076259A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
IL187245A0 (en) * 2007-11-08 2008-12-29 Hadasit Med Res Service Synthetic sphingolipid analogs

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2727070A (en) * 1950-02-25 1955-12-13 Parke Davis & Co Substituted propanols and processes for their manufacture
US2727071A (en) * 1950-06-16 1955-12-13 Parke Davis & Co Process for obtaining substituted chloropropanols from oxazolines
US2759972A (en) * 1951-10-01 1956-08-21 Sterling Drug Inc 2-amino and acylamino-1-(hydrocarbylsulphonylphenyl)-1, 3-propanediols
US2759971A (en) * 1951-10-01 1956-08-21 Sterling Drug Inc 2-amino and acylamino-1-(hydrocarbylmercaptophenyl)-1, 3-propanediols and preparation thereof
US2717268A (en) * 1952-12-16 1955-09-06 Parke Davis & Co Process for preparing phenyldichloro-acetamidopropanediols
US2876261A (en) * 1955-09-15 1959-03-03 Parke Davis & Co Alpha-di-chloroacetamido-beta-chloro-p-nitropropiophenone and method of production
US2759927A (en) * 1955-12-27 1956-08-21 Sterling Drug Inc Hexamethylenetetramine adducts of haloaceto-mercaptophenones
US2776992A (en) * 1956-03-14 1957-01-08 Du Pont Trifluoromethylsulfonylphenyldichloracetamidopropandiol
US2759970A (en) * 1956-05-09 1956-08-21 Sterling Drug Inc Acylamidoaceto-mercaptophenones
US3012073A (en) * 1960-04-11 1961-12-05 Du Pont Trifluoro methylthiophenyl-dichloro-acet-amides-1, 3-propanediol
US4235892A (en) * 1979-02-05 1980-11-25 Schering Corporation, Patent Dept. 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor

Also Published As

Publication number Publication date
IT8622826A0 (it) 1986-12-23
EP0272684B1 (en) 1991-06-12
JPS63190870A (ja) 1988-08-08
US4918095A (en) 1990-04-17
DE3770788D1 (de) 1991-07-18
EP0272684A2 (en) 1988-06-29
EP0272684A3 (en) 1988-12-28
ATE64379T1 (de) 1991-06-15
IT1198238B (it) 1988-12-21
GR3002135T3 (en) 1992-12-30

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