ES2094729T3 - Compuestos macrolidos. - Google Patents

Compuestos macrolidos.

Info

Publication number
ES2094729T3
ES2094729T3 ES89305579T ES89305579T ES2094729T3 ES 2094729 T3 ES2094729 T3 ES 2094729T3 ES 89305579 T ES89305579 T ES 89305579T ES 89305579 T ES89305579 T ES 89305579T ES 2094729 T3 ES2094729 T3 ES 2094729T3
Authority
ES
Spain
Prior art keywords
group
hydrogen atom
compounds
hydroxyl group
chem
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES89305579T
Other languages
English (en)
Inventor
Gordon C Lawrence
Michael J Dawson
David Noble
Richard A Fletton
Stephen Joseph Lane
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Application granted granted Critical
Publication of ES2094729T3 publication Critical patent/ES2094729T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Veterinary Medicine (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Molecular Biology (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyrane Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Furan Compounds (AREA)
  • Devices For Conveying Motion By Means Of Endless Flexible Members (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

LA INVENCION SE REFIERE A COMPUESTOS DE FORMULA(I) Y A SUS SALES, EN LA QUE R1 ES UN GRUPO METILO, ETILO O ISOPROPILO SUSTITUIDO CADA UNO POR UIN GRUPO HIDROXILO, O R1 ES UN GRUPO CH2NR7 O - CH(CH3)R7 (DONDE M ES CERO O 1 Y R7 ES CHO O CO2H); Y1 ES - CH2 -, Y2 ES - CH - Y X ES UN GRUPO (II) (EN DONDE R2 Y R3 PUEDEN SER DIFERENTES; R4 ES UN GRUPO OR8 (DONDE R8 ES OH O OH SUSTITUIDO QUE PUEDE TENER HASTA 25 C), O R4 Y R5 JUNTO CON EL C AL QUE ESTAN UNIDOS SON > C = O O > C = NOR9A (SIENDO R9A UN H O UN GRUPO ALQUILO O ALQUENILO DE HASTA 8 C); Y R6 ES H O OH. LOS COMPUESTOS PUEDEN EMPLEARSE PARA EL CONTROL DE NEMATODOS, ACAROS, INSECTOS U OTRAS PLAGAS.
ES89305579T 1988-06-03 1989-06-02 Compuestos macrolidos. Expired - Lifetime ES2094729T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888813150A GB8813150D0 (en) 1988-06-03 1988-06-03 Chemical compounds

Publications (1)

Publication Number Publication Date
ES2094729T3 true ES2094729T3 (es) 1997-02-01

Family

ID=10638007

Family Applications (1)

Application Number Title Priority Date Filing Date
ES89305579T Expired - Lifetime ES2094729T3 (es) 1988-06-03 1989-06-02 Compuestos macrolidos.

Country Status (19)

Country Link
US (1) US5108992A (es)
EP (1) EP0345078B1 (es)
JP (1) JP2540633B2 (es)
KR (1) KR900000368A (es)
AT (1) ATE144985T1 (es)
AU (1) AU628823B2 (es)
BR (1) BR8902534A (es)
CA (1) CA1318628C (es)
DD (1) DD284049A5 (es)
DE (1) DE68927420T2 (es)
DK (1) DK273189A (es)
ES (1) ES2094729T3 (es)
GB (1) GB8813150D0 (es)
GR (1) GR3022392T3 (es)
HU (1) HU205390B (es)
IE (1) IE81096B1 (es)
NZ (1) NZ229388A (es)
PT (1) PT90746B (es)
ZA (1) ZA894193B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8721647D0 (en) * 1987-09-15 1987-10-21 Pfizer Ltd Antiparasitic agents
US5015662A (en) * 1988-10-18 1991-05-14 Merck & Co., Inc. Anthelmintic bioconversion products
US4988824A (en) * 1989-09-11 1991-01-29 Maulding Donald R Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds
US5140042A (en) * 1990-09-12 1992-08-18 Merck & Co., Inc. 28-hydroxy ivermectin aglycone
GB9027721D0 (en) * 1990-12-20 1991-02-13 Beecham Group Plc Novel compounds
GB9205007D0 (en) * 1992-03-07 1992-04-22 Pfizer Ltd Antiparasitic agents
JP3703677B2 (ja) * 2000-03-01 2005-10-05 ヒゲタ醤油株式会社 新規マクロライド系化合物ｊｋ
EP1478625A1 (en) * 2002-02-27 2004-11-24 Pfizer Products Inc. Processes and intermediates useful in preparing beta-3-adrenergic receptor agonists
JP4857656B2 (ja) * 2005-08-23 2012-01-18 東レ株式会社 耐弾防御衣料
MX2012004133A (es) * 2009-10-07 2012-05-08 Wyeth Llc Composiciones que comprenden adyuvante, macrolido y antigeno proteico y procedimientos de uso de las mismas.

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
US4857509A (en) * 1985-01-22 1989-08-15 Ciba-Geigy Corporation 13β-alkylmilbemycin derivatives for controlling parasites of animals and plants
US4666937A (en) * 1985-03-04 1987-05-19 Merck & Co., Inc. Avermectin bioconversion products
IL78621A (en) * 1985-04-30 1991-06-30 American Cyanamid Co Mylbemycin analogs,their preparation and pesticidal compositions containing them
JPH085893B2 (ja) * 1985-09-13 1996-01-24 アメリカン・サイアナミツド・カンパニー マクロライド抗生物質およびその製法
JPH0678342B2 (ja) * 1986-01-07 1994-10-05 三共株式会社 新規マクロライド化合物
ES2051731T3 (es) * 1986-01-23 1994-07-01 American Cyanamid Co Un procedimiento para preparar antibioticos macrolidos y su uso.
GB8606108D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Chemical compounds
IE62126B1 (en) * 1986-03-12 1994-12-14 American Cyanamid Co Macrolide compounds
CA1296329C (en) * 1986-06-06 1992-02-25 Derek R. Sutherland Macrolide compounds
US4916154A (en) * 1986-09-12 1990-04-10 American Cyanamid Company 23-Imino derivatives of LL-F28249 compounds
US5015662A (en) * 1988-10-18 1991-05-14 Merck & Co., Inc. Anthelmintic bioconversion products

Also Published As

Publication number Publication date
ATE144985T1 (de) 1996-11-15
HU205390B (en) 1992-04-28
JPH0285289A (ja) 1990-03-26
GB8813150D0 (en) 1988-07-06
HUT57833A (en) 1991-12-30
EP0345078B1 (en) 1996-11-06
PT90746A (pt) 1989-12-29
PT90746B (pt) 1994-10-31
DE68927420T2 (de) 1997-06-12
AU3599789A (en) 1990-01-11
CA1318628C (en) 1993-06-01
AU628823B2 (en) 1992-09-24
DK273189D0 (da) 1989-06-02
JP2540633B2 (ja) 1996-10-09
ZA894193B (en) 1990-05-30
DK273189A (da) 1989-12-04
EP0345078A2 (en) 1989-12-06
DD284049A5 (de) 1990-10-31
EP0345078A3 (en) 1991-01-23
NZ229388A (en) 1991-06-25
IE81096B1 (en) 2000-03-08
KR900000368A (ko) 1990-01-30
IE891747L (en) 1989-12-03
BR8902534A (pt) 1990-01-23
US5108992A (en) 1992-04-28
GR3022392T3 (en) 1997-04-30
DE68927420D1 (de) 1996-12-12

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