ES2102871T3 - Agentes antiparasitarios. - Google Patents

Agentes antiparasitarios.

Info

Publication number
ES2102871T3
ES2102871T3 ES94924798T ES94924798T ES2102871T3 ES 2102871 T3 ES2102871 T3 ES 2102871T3 ES 94924798 T ES94924798 T ES 94924798T ES 94924798 T ES94924798 T ES 94924798T ES 2102871 T3 ES2102871 T3 ES 2102871T3
Authority
ES
Spain
Prior art keywords
sub
oleandrosil
alpha
halo
independently
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94924798T
Other languages
English (en)
Inventor
Christopher James Dutton
Stephen Paul Gibson
Michael John Witty
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER
Pfizer Inc
Original Assignee
PFIZER
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER, Pfizer Inc filed Critical PFIZER
Application granted granted Critical
Publication of ES2102871T3 publication Critical patent/ES2102871T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

SE PRESENTAN DERIVADOS ANTIPARASITARIOS DE LA AVERMECTINA DE LA FORMULA (I), EN DONDE LA LINEA ROTA REPRESENTA UN ENLACE OPCIONAL, R1 Y R4 ESTAN AUSENTES CUANDO ESTE ENLACE ESTA PRESENTE, R1 Y R4 SON INDEPENDIENTEMENTE H, OH, HALO, OXIMINO, O UN RADICAL ORGANICO, R2, R6 Y R7 SON RADICALES ORGANICOS Y R3 ES ALFA-OLEANDROSIL O 4''-(ALFA-OLEANDROSIL)-ALFA-OLEANDROSIL OPCIONALMENTE SUSTITUIDO EN LA POSICION 4'' O 4", Y R12 Y R13 SON INDEPENDIENTEMENTE H, CN, CONH{SUB,2}, ALQUILO C{SUB,1-8} O ARILO OPCIONALMENTE SUSTITUIDO CON AL MENOS UN HALO, OH, ALCOXIDO C{SUB,1-8} O UN GRUPO DE ALQUILTIO C{SUB,1-6}.
ES94924798T 1993-08-04 1994-07-22 Agentes antiparasitarios. Expired - Lifetime ES2102871T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939316129A GB9316129D0 (en) 1993-08-04 1993-08-04 Antiprasatic agents

Publications (1)

Publication Number Publication Date
ES2102871T3 true ES2102871T3 (es) 1997-08-01

Family

ID=10739933

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94924798T Expired - Lifetime ES2102871T3 (es) 1993-08-04 1994-07-22 Agentes antiparasitarios.

Country Status (14)

Country Link
US (1) US5883080A (es)
EP (1) EP0712411B1 (es)
JP (1) JP2837958B2 (es)
AT (1) ATE154358T1 (es)
AU (1) AU679555B2 (es)
CA (1) CA2168731C (es)
DE (1) DE69403804T2 (es)
DK (1) DK0712411T3 (es)
ES (1) ES2102871T3 (es)
FI (1) FI960486A7 (es)
GB (1) GB9316129D0 (es)
GR (1) GR3024209T3 (es)
NZ (1) NZ271349A (es)
WO (1) WO1995004746A1 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2753377B1 (fr) * 1996-09-19 1999-09-24 Rhone Merieux Nouvelle association parasiticide a base de 1-n-phenylpyra- zoles et de lactones macrocycliques endectocides
US6426333B1 (en) 1996-09-19 2002-07-30 Merial Spot-on formulations for combating parasites
US6998131B2 (en) * 1996-09-19 2006-02-14 Merial Limited Spot-on formulations for combating parasites
AU2001277712A1 (en) * 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
US20040087519A1 (en) * 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
US7831519B2 (en) * 2003-12-17 2010-11-09 First Data Corporation Methods and systems for electromagnetic initiation of secure transactions
WO2010106325A2 (en) 2009-03-18 2010-09-23 Omnipharm Limited Parasiticidal formulation
CN103360444B (zh) * 2012-04-03 2016-05-11 浙江海正药业股份有限公司 抗寄生虫药赛拉菌素的合成新工艺
WO2024135828A1 (ja) 2022-12-23 2024-06-27 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 エバーメクチン誘導体

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS62252788A (ja) * 1986-04-25 1987-11-04 Sankyo Co Ltd １３−ヒドロキシミルベマイシン誘導体およびその製造法
JP2666936B2 (ja) * 1987-11-13 1997-10-22 株式会社シグマ スロットマシンのリール駆動装置
GB8726730D0 (en) * 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
GB8815967D0 (en) * 1988-07-05 1988-08-10 Pfizer Ltd Antiparasitic agents
US5411946A (en) * 1993-02-24 1995-05-02 Merck & Co., Inc. Avermectin derivatives
PL174488B1 (pl) * 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt

Also Published As

Publication number Publication date
WO1995004746A1 (en) 1995-02-16
DE69403804D1 (de) 1997-07-17
US5883080A (en) 1999-03-16
CA2168731C (en) 1999-03-30
JP2837958B2 (ja) 1998-12-16
FI960486A0 (fi) 1996-02-02
EP0712411B1 (en) 1997-06-11
EP0712411A1 (en) 1996-05-22
FI960486L (fi) 1996-02-02
DK0712411T3 (da) 1997-07-14
AU7495394A (en) 1995-02-28
GR3024209T3 (en) 1997-10-31
ATE154358T1 (de) 1997-06-15
AU679555B2 (en) 1997-07-03
GB9316129D0 (en) 1993-09-22
DE69403804T2 (de) 1997-09-18
NZ271349A (en) 1997-11-24
JPH08508043A (ja) 1996-08-27
CA2168731A1 (en) 1995-02-16
FI960486A7 (fi) 1996-02-02

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