ES2170101T3 - Compuesto ciclodepsipeptido. - Google Patents

Compuesto ciclodepsipeptido.

Info

Publication number
ES2170101T3
ES2170101T3 ES94925614T ES94925614T ES2170101T3 ES 2170101 T3 ES2170101 T3 ES 2170101T3 ES 94925614 T ES94925614 T ES 94925614T ES 94925614 T ES94925614 T ES 94925614T ES 2170101 T3 ES2170101 T3 ES 2170101T3
Authority
ES
Spain
Prior art keywords
compound
salt
cyclodepsipeptide
cyclodepsipeptide compound
low rent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94925614T
Other languages
English (en)
Inventor
Hitoshi Nishiyama
Masaru Ohgaki
Ryo Yamanishi
Toshihiko Hara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astellas Pharma Inc
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Application granted granted Critical
Publication of ES2170101T3 publication Critical patent/ES2170101T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Dental Preparations (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Manufacture Of Tobacco Products (AREA)

Abstract

UN COMPUESTO DE LA FORMULA: EN DONDE A ES UN GRUPO DE BENCILO QUE TIENE UN SUSTITUYENTE(S) ADECUADO (S), A{SUP,A}, B Y D SON CADA UNO ALQUILO BAJO, C ES HIDROGENO O ALQUILO BAJO, O UNA SAL DE LOS MISMOS. EL COMPUESTO O SU SAL DE LA PRESENTE INVENCION TIENE EXCELENTES ACTIVIDADES PARASITICIDAS COMO PARASITICIDAS (ANTIHELMINTICAS) PARA ANIMALES Y CUERPOS HUMANOS.
ES94925614T 1993-09-06 1994-08-31 Compuesto ciclodepsipeptido. Expired - Lifetime ES2170101T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP24632393 1993-09-06

Publications (1)

Publication Number Publication Date
ES2170101T3 true ES2170101T3 (es) 2002-08-01

Family

ID=17146855

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94925614T Expired - Lifetime ES2170101T3 (es) 1993-09-06 1994-08-31 Compuesto ciclodepsipeptido.

Country Status (16)

Country Link
US (1) US5646244A (es)
EP (1) EP0718293B1 (es)
JP (1) JP3263947B2 (es)
KR (1) KR100392172B1 (es)
CN (1) CN1061039C (es)
AT (1) ATE214379T1 (es)
AU (1) AU686222B2 (es)
BR (1) BR9407711A (es)
CA (1) CA2171088A1 (es)
DE (1) DE69430128T2 (es)
DK (1) DK0718293T3 (es)
ES (1) ES2170101T3 (es)
NZ (1) NZ271739A (es)
PT (1) PT718293E (es)
TW (1) TW318844B (es)
WO (1) WO1995007272A1 (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0872481B1 (en) * 1995-06-30 2009-03-18 Astellas Pharma Inc. Depsipeptide derivative, process for production thereof, and novel intermediate therefor
KR19990044489A (ko) * 1995-09-07 1999-06-25 로렌스 티. 마이젠헬더 환식 구충제
DE69721055T2 (de) 1996-10-07 2004-02-19 Fujisawa Pharmaceutical Co., Ltd. Verfahren zur herstellung von depsipeptiden und zwischenprodukten davon
DE19713626A1 (de) 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
US6355615B1 (en) * 1997-06-04 2002-03-12 Bayer Aktiengesellschaft Desoxycyclodepsipeptides and their use for combatting endoparasites
KR100551651B1 (ko) 1997-11-10 2006-02-13 아스텔라스세이야쿠 가부시키가이샤 뎁시펩티드 유도체의 신규 결정 및 그의 제조 방법
DE19921887A1 (de) * 1999-05-12 2000-11-16 Bayer Ag Endoparasitizide Mittel
DE19962145A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel/Depsipeptide
DE19962147A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel / PF 1022-221
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102008022520A1 (de) * 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) * 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031283A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
DE102008031284A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
CN102224151A (zh) 2008-11-20 2011-10-19 万能药生物有限公司 新的抗微生物剂
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
RU2012102094A (ru) 2009-06-26 2013-08-10 Панацеа Биотек Лтд. Новые азабициклогексаны
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
RS62130B1 (sr) 2015-05-20 2021-08-31 Boehringer Ingelheim Animal Health Usa Inc Antihelmintička depsipeptidna jedinjenja
EP3397638B1 (en) 2015-12-28 2023-08-23 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
BR112019009977A2 (pt) 2016-11-16 2019-08-27 Boehringer Ingelheim Animal Health Usa Inc compostos depsipeptídicos anti-helmínticos
RU2747149C9 (ru) 2017-11-29 2021-06-29 ЗОЕТИС СЕРВИСИЗ ЭлЭлСи Анти-эндопаразитарные депсипептиды
ES3030701T3 (en) 2018-05-10 2025-07-01 Zoetis Services Llc Endoparasitic depsipeptides
US20220071183A1 (en) 2019-01-10 2022-03-10 Zoetis Services Llc Anthelmintic laboratory animal model for heartworm
EP4262789A1 (en) 2020-12-21 2023-10-25 Boehringer Ingelheim Vetmedica GmbH Parasiticidal collar comprising isoxazoline compounds
WO2025233804A1 (en) * 2024-05-07 2025-11-13 Animol Discovery, Inc. Method of treating heartworm with emodepside

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
JP3207870B2 (ja) * 1991-04-15 2001-09-10 明治製菓株式会社 環状デプシペプチドおよびその製造法
DK0634408T3 (da) * 1992-03-17 2002-04-22 Fujisawa Pharmaceutical Co Depsipeptidderivater, fremstilling og anvendelse deraf
CN1073560C (zh) * 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung

Also Published As

Publication number Publication date
AU686222B2 (en) 1998-02-05
DK0718293T3 (da) 2002-04-22
CN1061039C (zh) 2001-01-24
KR100392172B1 (ko) 2004-04-03
KR960704868A (ko) 1996-10-09
NZ271739A (en) 1996-09-25
BR9407711A (pt) 1997-02-12
CN1133592A (zh) 1996-10-16
DE69430128T2 (de) 2002-09-05
WO1995007272A1 (fr) 1995-03-16
EP0718293B1 (en) 2002-03-13
JP3263947B2 (ja) 2002-03-11
PT718293E (pt) 2002-08-30
AU7546394A (en) 1995-03-27
EP0718293A4 (en) 1997-04-16
ATE214379T1 (de) 2002-03-15
TW318844B (es) 1997-11-01
DE69430128D1 (en) 2002-04-18
CA2171088A1 (en) 1995-03-16
US5646244A (en) 1997-07-08
EP0718293A1 (en) 1996-06-26

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