ES265263A1 - Method for the production of indol derivatives (Machine-translation by Google Translate, not legally binding) - Google Patents
Method for the production of indol derivatives (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES265263A1 ES265263A1 ES0265263A ES265263A ES265263A1 ES 265263 A1 ES265263 A1 ES 265263A1 ES 0265263 A ES0265263 A ES 0265263A ES 265263 A ES265263 A ES 265263A ES 265263 A1 ES265263 A1 ES 265263A1
- Authority
- ES
- Spain
- Prior art keywords
- groups
- alkyl
- formula
- nucleus
- lower alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- SIKJAQJRHWYJAI-UHFFFAOYSA-N Indole Chemical class C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- RWRDLPDLKQPQOW-UHFFFAOYSA-N Pyrrolidine Chemical compound C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 150000002367 halogens Chemical group 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 150000002475 indoles Chemical class 0.000 abstract 3
- YNAVUWVOSKDBBP-UHFFFAOYSA-N Morpholine Chemical compound C1COCCN1 YNAVUWVOSKDBBP-UHFFFAOYSA-N 0.000 abstract 2
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 abstract 2
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical group [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000004103 aminoalkyl group Chemical class 0.000 abstract 1
- 229940054051 antipsychotic indole derivative Drugs 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 239000002184 metal Chemical group 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
Method for the production of indole derivatives, of the formula: ** (See formula) ** and salts thereof, in which formula R1 represents hydrogen, halogen, an alkyl or lower alkoxy group, or a nitro group, R2 and R3, which may be the same or different, represent hydrogen, halogen, alkyl groups, or lower alkoxy, acyl groups, benzyl groups, phenyl groups or substituted phenyl groups, the possible halogen substituent being alkyl or lower alkoxy groups, hydroxy groups or nitro groups and X is an N-substituted aminoalkyl group, in which the alkyl groups are linear or branched with 1-5 carbon atoms, and in which 1 or both substituents are alkyl or cycloalkyl groups, or, together with the nitrogen atom, form a saturated heterocyclic nucleus, such as pyrrolidine, piperidine, morpholine, piperazine or a nucleus of N-alkyl or N-cycloalkylpiperazine, or, X, by itself, constitutes said saturated heterocyclic nucleus, which is attached by one of the carbon atoms to the nitrogen atom of the indole nucleus, ca characterized by a compound of the formula ** (See formula) ** wherein R1, R2 and R3 have the above meaning and Z represents hydrogen or a metal atom, is reacted with a reactive ester of an alcohol, of the formula XOH, wherein X has the above meaning, after which , the resulting indole derivative is isolated, if desired, in salt form. (Machine-translation by Google Translate, not legally binding)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES0265263A ES265263A1 (en) | 1961-02-28 | 1961-02-28 | Method for the production of indol derivatives (Machine-translation by Google Translate, not legally binding) |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES0265263A ES265263A1 (en) | 1961-02-28 | 1961-02-28 | Method for the production of indol derivatives (Machine-translation by Google Translate, not legally binding) |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES265263A1 true ES265263A1 (en) | 1961-05-16 |
Family
ID=34493535
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES0265263A Expired ES265263A1 (en) | 1961-02-28 | 1961-02-28 | Method for the production of indol derivatives (Machine-translation by Google Translate, not legally binding) |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES265263A1 (en) |
-
1961
- 1961-02-28 ES ES0265263A patent/ES265263A1/en not_active Expired
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