ES276648A1 - Procedimiento para la fabricación de derivados de benzodiazepina - Google Patents

Procedimiento para la fabricación de derivados de benzodiazepina

Info

Publication number
ES276648A1
ES276648A1 ES276648A ES276648A ES276648A1 ES 276648 A1 ES276648 A1 ES 276648A1 ES 276648 A ES276648 A ES 276648A ES 276648 A ES276648 A ES 276648A ES 276648 A1 ES276648 A1 ES 276648A1
Authority
ES
Spain
Prior art keywords
manufacture
hydrogen
nitro
benzodiazepine derivatives
acid addition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES276648A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of ES276648A1 publication Critical patent/ES276648A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • C07D243/28—Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES276648A 1961-04-20 1962-04-19 Procedimiento para la fabricación de derivados de benzodiazepina Expired ES276648A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10422761A 1961-04-20 1961-04-20

Publications (1)

Publication Number Publication Date
ES276648A1 true ES276648A1 (es) 1962-10-16

Family

ID=22299329

Family Applications (1)

Application Number Title Priority Date Filing Date
ES276648A Expired ES276648A1 (es) 1961-04-20 1962-04-19 Procedimiento para la fabricación de derivados de benzodiazepina

Country Status (5)

Country Link
BE (1) BE616024A (es)
CH (1) CH411912A (es)
ES (1) ES276648A1 (es)
GB (1) GB986903A (es)
SE (1) SE301976B (es)

Also Published As

Publication number Publication date
SE301976B (es) 1968-07-01
BE616024A (fr) 1962-10-05
CH411912A (de) 1966-04-30
GB986903A (en) 1965-03-24

Similar Documents

Publication Publication Date Title
ES267248A1 (es) Procedimiento para la obtenciën de la l-isopropilo-4-hidroxi-6-bencilo-pirazolo (3,4-d) piramidina y de sus sales
ES303009A1 (es) Procedimiento para la preparacion de compuestos de imidazolidina.
ES319653A1 (es) Un procedimiento para la preparacion de derivados de imidazol.
ES394761A1 (es) Un metodo de preparar un derivado de 2-amino-1,5-benzodia- zocina.
GB972962A (en) A process for the manufacture of benzodiazepine derivatives
ES465346A1 (es) Procedimiento para preparar imidazoles 4,5-disustituidos.
ES286241A1 (es) Un procedimiento para la fabricación de derivados benzodiazepínicos
ES324458A1 (es) Un procedimiento para la preparacion de derivados de benzodiazepina.
ES298897A1 (es) Un procedimiento para la preparación de derivados de benzodiazepina
ES302128A1 (es) Procedimiento para la preparacion de nuevas n-arilsulfonilureas n'-sustituidas.
ES283029A1 (es) Procedimiento para la fabricación de derivados benzodiazepínicos
ES285855A1 (es) Un procedimiento para la fabricación de derivados benzodiazepínicos
ES283604A1 (es) Procedimiento de obtención de derivados de naftaleno
GB977228A (en) Silver propiolic acid esters and process for their manufacture
ES266946A1 (es) Procedimiento de obtenciën de nuevos derivados de acido 2,6-dialkilbenzoico
ES305413A1 (es) Un procedimiento para la preparacion de derivados de benzodiazepina.
ES264004A1 (es) Procedimiento para la fabricaciën de compuestos benzodiazepinicos que contienen fluor
ES310920A1 (es) Procedimiento para la obtencion de compuestos heterociclicospiperidinicos.
ES317893A1 (es) Un procedimiento para la preparacion de derivados de benzodiazepina.
ES327403A1 (es) Procedimiento para la preparacion de nuevos derivados de guanidina.
ES312701A1 (es) Procedimiento de produccion de 2-benzoxazolinonas.
ES248822A1 (es) Un método para preparar nuevos compuestos de tetraciclina
ES382147A1 (es) Un procedimiento para preparar compuestos de morfolina n- sustituidos.
ES292054A1 (es) Procedimiento de preparación de un derivado de la benzotiadiacina, de acción hipotensiva
ES287549A1 (es) Procedimiento para la producción del ácido n-(2,3-dimetilfenil)-antranílico y sus sales