ES528003A0 - Un procedimiento para preparar derivados de cefem - Google Patents

Un procedimiento para preparar derivados de cefem

Info

Publication number
ES528003A0
ES528003A0 ES528003A ES528003A ES528003A0 ES 528003 A0 ES528003 A0 ES 528003A0 ES 528003 A ES528003 A ES 528003A ES 528003 A ES528003 A ES 528003A ES 528003 A0 ES528003 A0 ES 528003A0
Authority
ES
Spain
Prior art keywords
procedure
cefem derivatives
preparing
preparing cefem
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES528003A
Other languages
English (en)
Other versions
ES8506025A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai Co Ltd
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP21772682A external-priority patent/JPS59108791A/ja
Priority claimed from JP3601783A external-priority patent/JPS59161389A/ja
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of ES528003A0 publication Critical patent/ES528003A0/es
Publication of ES8506025A1 publication Critical patent/ES8506025A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
ES528003A 1982-12-14 1983-12-13 Un procedimiento para preparar derivados de cefem Expired ES8506025A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP21772682A JPS59108791A (ja) 1982-12-14 1982-12-14 ７−カルボキシメトキシフエニルアセトアミド−３−セフエム誘導体、その製造方法およびそれからなる抗菌剤
JP3601783A JPS59161389A (ja) 1983-03-07 1983-03-07 ７−カルボキシメトキシフエニルアセトアミドセフエム誘導体，その製造法およびそれからなる抗菌剤

Publications (2)

Publication Number Publication Date
ES528003A0 true ES528003A0 (es) 1985-06-16
ES8506025A1 ES8506025A1 (es) 1985-06-16

Family

ID=26375029

Family Applications (2)

Application Number Title Priority Date Filing Date
ES528003A Expired ES8506025A1 (es) 1982-12-14 1983-12-13 Un procedimiento para preparar derivados de cefem
ES534297A Granted ES534297A0 (es) 1982-12-14 1984-07-13 Un procedimiento para preparar derivados de cefem

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES534297A Granted ES534297A0 (es) 1982-12-14 1984-07-13 Un procedimiento para preparar derivados de cefem

Country Status (16)

Country Link
US (1) US4546176A (es)
KR (1) KR840007012A (es)
AT (1) ATA435283A (es)
AU (1) AU2082783A (es)
BE (1) BE898442A (es)
CH (1) CH656131A5 (es)
DE (1) DE3345093A1 (es)
DK (1) DK572183A (es)
ES (2) ES8506025A1 (es)
FR (1) FR2569195B1 (es)
GB (1) GB2132613B (es)
IT (1) IT1169969B (es)
NL (1) NL8304272A (es)
PH (1) PH20168A (es)
SE (1) SE8306882L (es)
YU (1) YU237283A (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5232918A (en) * 1987-07-23 1993-08-03 Imperial Chemical Industries Plc Cephalosporin derivatives
CA2001203C (en) * 1988-10-24 2001-02-13 Thomas P. Demuth, Jr. Novel antimicrobial dithiocarbamoyl quinolones
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
US5491139A (en) * 1988-10-24 1996-02-13 The Procter & Gamble Company Antimicrobial quinolonyl lactams
US5180719A (en) * 1988-10-24 1993-01-19 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactam esters
US5273973A (en) * 1988-10-24 1993-12-28 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl esters
EP0366189A3 (en) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Novel antimicrobial lactam-quinolones
WO1991016327A1 (en) * 1990-04-18 1991-10-31 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactams
US5244892A (en) * 1990-10-16 1993-09-14 Kyorin Pharmaceutical Co., Ltd. Cephem compounds, and antibacterial agents
BR9508513A (pt) * 1994-08-02 1998-06-02 Procter & Gamble Processo para a produção de antimicrobianos de quinolonil lactama e novos compostos intermediários
MX9700871A (es) * 1994-08-02 1997-05-31 Procter & Gamble Procedimiento para hacer compuestos antimicrobianos.
US7091196B2 (en) * 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
AU2004217919A1 (en) * 2003-03-05 2004-09-16 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using the same
WO2005042554A1 (en) * 2003-10-30 2005-05-12 Rib-X Pharmaceuticals, Inc. Bifunctional macrolide heterocyclic compounds and methods of making and using the same
JP2007512256A (ja) * 2003-11-18 2007-05-17 リブ−エックス ファーマシューティカルズ，インコーポレイテッド 二官能性マクロライド複素環化合物ならびにこれらを製造する方法およびこれらを使用する方法
EP2716647A3 (en) * 2004-02-27 2014-08-20 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR208171A1 (es) * 1972-09-29 1976-12-09 Ciba Geigy Ag Procedimiento para la obtencion de nuevos derivados del acido cef-3-em-4-carboxilico
US4338439A (en) * 1976-08-26 1982-07-06 Eli Lilly And Company 7-[2-[(Substituted benzoyl]amino]acetamido]cephalosporins
SE8009049L (sv) * 1980-03-04 1981-09-05 Eisai Co Ltd 7alfa-metoxicefalosporinderivat, sett for framstellning derav och antibakteriella lekemedel innehallande dessa foreningar
US4468394A (en) * 1981-04-02 1984-08-28 Eisai Co., Ltd. Cephalosporin compounds

Also Published As

Publication number Publication date
IT1169969B (it) 1987-06-03
SE8306882L (sv) 1984-06-15
FR2569195B1 (fr) 1987-01-09
GB2132613B (en) 1986-05-08
US4546176A (en) 1985-10-08
DK572183A (da) 1984-06-27
AU2082783A (en) 1984-06-21
ES8505691A1 (es) 1985-06-01
GB2132613A (en) 1984-07-11
DK572183D0 (da) 1983-12-13
YU237283A (en) 1986-04-30
FR2569195A1 (fr) 1986-02-21
NL8304272A (nl) 1984-07-02
SE8306882D0 (sv) 1983-12-13
GB8329554D0 (en) 1983-12-07
CH656131A5 (de) 1986-06-13
ES534297A0 (es) 1985-06-01
BE898442A (fr) 1984-06-13
PH20168A (en) 1986-10-09
KR840007012A (ko) 1984-12-04
ES8506025A1 (es) 1985-06-16
DE3345093A1 (de) 1984-06-14
IT8324122A0 (it) 1983-12-12
ATA435283A (de) 1986-12-15

Similar Documents

Publication Publication Date Title
ES546916A0 (es) Un procedimiento para preparar derivados de guanina
ES538190A0 (es) Un procedimiento para preparar derivados de pirimidina
ES532538A0 (es) Un procedimiento para preparar un derivado de carbostirilo
ES530024A0 (es) Un procedimiento para preparar derivados de pirazinona
ES537104A0 (es) Un procedimiento para preparar derivados de tiazina
ES557808A0 (es) Un procedimiento para preparar derivados de octahidro(f) quinoleina
ES523195A0 (es) Un procedimiento para preparar alquil-glicosidos
ES537668A0 (es) Un procedimiento para preparar n-formil-3-fenoxi-1-azetidincarboxamidas
ES528304A0 (es) Un procedimiento para preparar derivados de pirimidona
ES534297A0 (es) Un procedimiento para preparar derivados de cefem
ES525941A0 (es) Un procedimiento para preparar nuevos derivados de eteno
ES523419A0 (es) Un metodo para preparar derivados de 4-hidroxi-2-quinolona
ES535568A0 (es) Un procedimiento para preparar derivados de piridazinona
ES533059A0 (es) Un procedimiento para preparar derivados de aminoglicosido
ES523193A0 (es) Un procedimiento para preparar 3-fenoxi-1-azetidincarbo-xznmidas
ES530019A0 (es) Un metodo para preparar derivados de 3-metilflavona
ES526088A0 (es) Un procedimiento para preparar derivados de ciclobutano
ES525007A0 (es) Un procedimiento para producir derivados de tiazol
ES519936A0 (es) Un procedimiento para preparar derivados de pirimidona.
ES534356A0 (es) Un metodo para preparar derivados de fenotiazina
ES526177A0 (es) Un procedimiento para preparar derivados de pirimidona
ES530855A0 (es) Un procedimiento para preparar derivados de benzotiazina
ES529478A0 (es) Un procedimiento para preparar derivados de mitomicina
ES506302A0 (es) Un procedimiento para preparar derivados de tetrahidroiso- quinoleinas
ES527738A0 (es) Un procedimiento para preparar derivados de piridona