ES553609A0 - Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides - Google Patents

Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides

Info

Publication number
ES553609A0
ES553609A0 ES553609A ES553609A ES553609A0 ES 553609 A0 ES553609 A0 ES 553609A0 ES 553609 A ES553609 A ES 553609A ES 553609 A ES553609 A ES 553609A ES 553609 A0 ES553609 A0 ES 553609A0
Authority
ES
Spain
Prior art keywords
isocian
steroids
preparation procedure
sulfonyl methylene
sulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES553609A
Other languages
English (en)
Other versions
ES8800263A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gist Brocades NV
Original Assignee
Gist Brocades NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades NV filed Critical Gist Brocades NV
Publication of ES8800263A1 publication Critical patent/ES8800263A1/es
Publication of ES553609A0 publication Critical patent/ES553609A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/005—3 membered carbocyclic rings in position 12
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES553609A 1983-04-29 1986-04-01 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides Expired ES8800263A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP83200616A EP0123734A1 (en) 1983-04-29 1983-04-29 17-(Isocyano-sulfonylmethylene)-steroids, 17-(formamido-sulfonylmethylene)-steroids and their preparation

Publications (2)

Publication Number Publication Date
ES8800263A1 ES8800263A1 (es) 1987-11-01
ES553609A0 true ES553609A0 (es) 1987-11-01

Family

ID=8190949

Family Applications (2)

Application Number Title Priority Date Filing Date
ES532029A Expired ES8608537A1 (es) 1983-04-29 1984-04-28 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides
ES553609A Expired ES8800263A1 (es) 1983-04-29 1986-04-01 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES532029A Expired ES8608537A1 (es) 1983-04-29 1984-04-28 Procedimiento de preparacion de 17-(isociano-sulfonilmetileno)-esteroides, 17-(formamido-sulfonilmetileno)-esteroides

Country Status (17)

Country Link
US (1) US4647410A (es)
EP (2) EP0123734A1 (es)
JP (2) JPS59206399A (es)
KR (1) KR860001469B1 (es)
AU (1) AU568643B2 (es)
CA (1) CA1257249A (es)
DE (1) DE3461381D1 (es)
DK (2) DK166545B1 (es)
ES (2) ES8608537A1 (es)
FI (1) FI82061C (es)
GR (1) GR81997B (es)
HU (2) HU194277B (es)
IE (1) IE57328B1 (es)
IL (1) IL71658A (es)
NO (1) NO167093C (es)
NZ (1) NZ207985A (es)
PT (1) PT78503B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0123735A1 (en) * 1983-04-29 1984-11-07 Gist-Brocades N.V. New process for the preparation of 20-keto-delta-16-steroids and new intermediate compounds formed in this process
US5194602A (en) * 1988-04-08 1993-03-16 Gist-Brocades N.V. 9α-hydroxy-17-methylene steroids, process for their preparation and their use in the preparation of corticosteroids
HU226413B1 (en) * 1991-06-25 2008-11-28 Aventis Pharma Sa Novel 16-(nitro-substituted methyl)pregna-1,4-dien-3,20-dion derivatives and process for producing them
FR2681069B1 (fr) * 1991-09-06 1995-04-28 Roussel Uclaf Nouveau procede de preparation de l'hydrocortisone et nouveaux intermediaires.
FR2683530B1 (fr) * 1991-11-08 1994-01-21 Roussel Uclaf Nouveau procede de preparation de derives 20-oxo 17 alpha, 21-dihydroxyles du pregnane et nouveaux intermediaires.
EA009176B1 (ru) 1995-12-11 2007-12-28 Дж.Д.Серл Энд Ко. Способ получения 7-альфа-карбоксил-9,11-эпоксистероидов и промежуточных продуктов, используемых для их получения, и общий способ эпоксидирования по олефиновым двойным связям
WO1998025948A2 (en) 1996-12-11 1998-06-18 G.D. Searle & Co. Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
US6887991B1 (en) 1996-12-11 2005-05-03 G. D. Searle & Company Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
ES2347027T3 (es) 1998-05-22 2010-10-22 The Board Of Trustees Of The Leland Stanford Junior University Moleculas bifuncionales y terapias basadas en las mismas.
EP2341423A1 (en) 1999-11-02 2011-07-06 Canon Kabushiki Kaisha Print control method and apparatus
US7235655B2 (en) 2002-03-22 2007-06-26 Pharmacia & Upjohn Company Processes to prepare eplerenone
EP2671507A3 (en) 2005-04-28 2014-02-19 Proteus Digital Health, Inc. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
CA2752373C (en) 2009-02-20 2017-10-10 To-Bbb Holding B.V. Glutathione-based drug delivery system
IL255113B (en) 2009-05-06 2022-09-01 Laboratory Skin Care Inc Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
CN105481924B (zh) * 2015-11-24 2017-08-15 浙江省诸暨合力化学对外贸易有限公司 一种黄体酮的制备方法
EP4392036A4 (en) * 2021-08-26 2026-03-11 Univ Brandeis SELECTIVE CYTOCHROME P450 SUBTYPE INHIBITORS BASED ON ISONITRILE

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7807631A (nl) * 1978-07-17 1980-01-21 Gist Brocades Nv Isocyanoderivaten en hun bereiding.
FR2462445A1 (fr) * 1979-07-31 1981-02-13 Roussel Uclaf Nouveaux derives 17-/(hydroxymethyl) (formamido) methylene/steroides, leur procede de preparation et leur application a l'introduction de la chaine laterale hydroxyacetyle
FR2486947A1 (fr) * 1980-07-15 1982-01-22 Roussel Uclaf Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto

Also Published As

Publication number Publication date
DK22192D0 (da) 1992-02-21
FI82061C (fi) 1991-01-10
ES8800263A1 (es) 1987-11-01
FI841679A0 (fi) 1984-04-27
KR840008461A (ko) 1984-12-15
KR860001469B1 (ko) 1986-09-26
PT78503B (en) 1986-05-20
IE841038L (en) 1984-10-29
ES532029A0 (es) 1986-07-16
DE3461381D1 (en) 1987-01-08
US4647410A (en) 1987-03-03
NO167093B (no) 1991-06-24
NO167093C (no) 1991-10-02
AU568643B2 (en) 1988-01-07
PT78503A (en) 1984-05-01
HU193207B (en) 1987-08-28
EP0124934A1 (en) 1984-11-14
CA1257249A (en) 1989-07-11
DK166545B1 (da) 1993-06-07
JPH0559097A (ja) 1993-03-09
EP0124934B1 (en) 1986-11-20
HUT34220A (en) 1985-02-28
FI82061B (fi) 1990-09-28
FI841679A7 (fi) 1984-10-30
IL71658A0 (en) 1984-07-31
NO841700L (no) 1984-10-30
HU194277B (en) 1988-01-28
JPH053478B2 (es) 1993-01-14
DK212184D0 (da) 1984-04-27
IL71658A (en) 1988-03-31
NZ207985A (en) 1986-11-12
JPS59206399A (ja) 1984-11-22
JPH0717673B2 (ja) 1995-03-01
DK166831B1 (da) 1993-07-19
ES8608537A1 (es) 1986-07-16
GR81997B (es) 1984-12-12
IE57328B1 (en) 1992-07-29
EP0123734A1 (en) 1984-11-07
DK22192A (da) 1992-02-21
DK212184A (da) 1984-10-30
AU2713384A (en) 1984-11-01

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