ES8506317A1 - Un procedimiento para la preparacion de derivados de 1,1-dioxido del acido 6 alfa-(aminometil)-penicilanico. - Google Patents

Un procedimiento para la preparacion de derivados de 1,1-dioxido del acido 6 alfa-(aminometil)-penicilanico.

Info

Publication number
ES8506317A1
ES8506317A1 ES533148A ES533148A ES8506317A1 ES 8506317 A1 ES8506317 A1 ES 8506317A1 ES 533148 A ES533148 A ES 533148A ES 533148 A ES533148 A ES 533148A ES 8506317 A1 ES8506317 A1 ES 8506317A1
Authority
ES
Spain
Prior art keywords
dioxide
derivatives
aminomethyl
penicillanic acid
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES533148A
Other languages
English (en)
Spanish (es)
Other versions
ES533148A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES533148A0 publication Critical patent/ES533148A0/es
Publication of ES8506317A1 publication Critical patent/ES8506317A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ES533148A 1983-06-06 1984-06-05 Un procedimiento para la preparacion de derivados de 1,1-dioxido del acido 6 alfa-(aminometil)-penicilanico. Expired ES8506317A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/501,476 US4502990A (en) 1983-06-06 1983-06-06 Process for 6-(aminomethyl)penicillanic acid 1,1-dioxide and derivatives thereof

Publications (2)

Publication Number Publication Date
ES533148A0 ES533148A0 (es) 1985-07-01
ES8506317A1 true ES8506317A1 (es) 1985-07-01

Family

ID=23993716

Family Applications (1)

Application Number Title Priority Date Filing Date
ES533148A Expired ES8506317A1 (es) 1983-06-06 1984-06-05 Un procedimiento para la preparacion de derivados de 1,1-dioxido del acido 6 alfa-(aminometil)-penicilanico.

Country Status (21)

Country Link
US (1) US4502990A (2)
EP (1) EP0128718B1 (2)
JP (1) JPS606692A (2)
KR (1) KR870000313B1 (2)
AT (1) ATE24513T1 (2)
AU (1) AU545506B2 (2)
CA (1) CA1209983A (2)
DE (1) DE3461801D1 (2)
DK (1) DK275984A (2)
ES (1) ES8506317A1 (2)
FI (1) FI842252L (2)
GR (1) GR81626B (2)
HU (1) HU191667B (2)
IL (1) IL72002A (2)
NO (1) NO842247L (2)
NZ (1) NZ208380A (2)
PH (1) PH19283A (2)
PL (1) PL144041B1 (2)
PT (1) PT78690A (2)
YU (1) YU97184A (2)
ZA (1) ZA844183B (2)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990006928A1 (en) * 1985-10-29 1990-06-28 Barth Wayne E 6-(1-carbamoyl-1-hydroxymethyl)penicillanic acid derivatives
US4868296A (en) * 1985-10-29 1989-09-19 Pfizer Inc. 6-(1-carbamoyl-1-hydroxymethyl) penicillanic acid derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4207323A (en) * 1975-11-21 1980-06-10 Merck & Co., Inc. 6-Substituted methyl penicillins, derivatives and analogues thereof
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4237051A (en) * 1979-04-19 1980-12-02 Schering Corporation Stereospecific production of 6- or 7-carbon-substituted-β-lactams
US4309347A (en) * 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
RO84910B (ro) * 1982-01-11 1984-09-30 Pfizer Inc. Procedeu pentru prepararea unor derivati 1, 1-dioxizi ai acidului 6-aminoalchilpenicilanic

Also Published As

Publication number Publication date
ZA844183B (en) 1986-01-29
KR870000313B1 (ko) 1987-02-26
PL248045A1 (en) 1985-07-30
PL144041B1 (en) 1988-04-30
AU545506B2 (en) 1985-07-18
GR81626B (2) 1984-12-11
JPS606692A (ja) 1985-01-14
FI842252A0 (fi) 1984-06-05
HUT34203A (en) 1985-02-28
ES533148A0 (es) 1985-07-01
PT78690A (en) 1984-07-01
ATE24513T1 (de) 1987-01-15
CA1209983A (en) 1986-08-19
AU2907784A (en) 1984-12-13
EP0128718B1 (en) 1986-12-30
YU97184A (en) 1986-06-30
EP0128718A1 (en) 1984-12-19
US4502990A (en) 1985-03-05
HU191667B (en) 1987-03-30
IL72002A (en) 1988-03-31
NZ208380A (en) 1987-05-29
FI842252A7 (fi) 1984-12-07
DK275984D0 (da) 1984-06-04
DE3461801D1 (en) 1987-02-05
DK275984A (da) 1984-12-07
KR850000447A (ko) 1985-02-27
NO842247L (no) 1984-12-07
PH19283A (en) 1986-03-04
FI842252L (fi) 1984-12-07
IL72002A0 (en) 1984-10-31

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