ES8605817A1 - Procedimiento para preparar un compuesto seleccionado del grupo constituido de 7-halo-7-desoxilincomicina y analogos de la misma - Google Patents

Procedimiento para preparar un compuesto seleccionado del grupo constituido de 7-halo-7-desoxilincomicina y analogos de la misma

Info

Publication number: ES8605817A1
Authority: ES; Spain
Prior art keywords: halo; lincomycin; deoxylincomycin; analogs; free bases
Prior art date: 1984-11-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES548152A

Other languages

English (en)

Spanish (es)

Other versions

ES548152A0 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pharmacia and Upjohn Co

Original Assignee

Upjohn Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-11-29

Filing date

1985-10-23

Publication date

1986-04-01

1985-10-23 Application filed by Upjohn Co filed Critical Upjohn Co

1986-04-01 Publication of ES548152A0 publication Critical patent/ES548152A0/es

1986-04-01 Publication of ES8605817A1 publication Critical patent/ES8605817A1/es

Status Expired legal-status Critical Current

Links

229960005287 lincomycin Drugs 0.000 abstract 4
ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 abstract 3
OJMMVQQUTAEWLP-UHFFFAOYSA-N Lincomycin Natural products CN1CC(CCC)CC1C(=O)NC(C(C)O)C1C(O)C(O)C(O)C(SC)O1 OJMMVQQUTAEWLP-UHFFFAOYSA-N 0.000 abstract 2
-1 THIONYL HALIDE Chemical class 0.000 abstract 2
OJMMVQQUTAEWLP-KIDUDLJLSA-N lincomycin Chemical compound CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@@H](C)O)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 OJMMVQQUTAEWLP-KIDUDLJLSA-N 0.000 abstract 2
FYSNRJHAOHDILO-UHFFFAOYSA-N thionyl chloride Chemical group ClS(Cl)=O FYSNRJHAOHDILO-UHFFFAOYSA-N 0.000 abstract 2
AEEIMWYSDWZKAT-HJTGYUAHSA-N (2r,3r,4s,5r,6r)-2-[(1r,2r)-1-amino-2-hydroxypropyl]-6-methylsulfanyloxane-3,4,5-triol Chemical compound CS[C@H]1O[C@H]([C@H](N)[C@@H](C)O)[C@H](O)[C@H](O)[C@H]1O AEEIMWYSDWZKAT-HJTGYUAHSA-N 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
229940088710 antibiotic agent Drugs 0.000 abstract 1
229960002227 clindamycin Drugs 0.000 abstract 1
KDLRVYVGXIQJDK-AWPVFWJPSA-N clindamycin Chemical compound CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@H](C)Cl)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 KDLRVYVGXIQJDK-AWPVFWJPSA-N 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Genetics & Genomics (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Crystallography & Structural Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Cephalosporin Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Indole Compounds (AREA)

ES548152A 1984-11-29 1985-10-23 Procedimiento para preparar un compuesto seleccionado del grupo constituido de 7-halo-7-desoxilincomicina y analogos de la misma Expired ES8605817A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US67615784A	1984-11-29	1984-11-29

Publications (2)

Publication Number	Publication Date
ES548152A0 ES548152A0 (es)	1986-04-01
ES8605817A1 true ES8605817A1 (es)	1986-04-01

Family

ID=24713464

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ES548152A Expired ES8605817A1 (es)	1984-11-29	1985-10-23	Procedimiento para preparar un compuesto seleccionado del grupo constituido de 7-halo-7-desoxilincomicina y analogos de la misma

Country Status (19)

Country	Link
US (1)	US4710565A (2)
EP (1)	EP0183505B1 (2)
JP (1)	JPH0649714B2 (2)
KR (1)	KR930003492B1 (2)
CN (2)	CN1004002B (2)
AT (1)	ATE50265T1 (2)
AU (1)	AU574232B2 (2)
CA (1)	CA1238319A (2)
DE (1)	DE3575930D1 (2)
DK (1)	DK165010C (2)
ES (1)	ES8605817A1 (2)
FI (1)	FI78708C (2)
GR (1)	GR852861B (2)
HU (1)	HU199497B (2)
IL (1)	IL76778A (2)
MX (1)	MX162251A (2)
PT (1)	PT81496B (2)
SU (1)	SU1405705A3 (2)
ZA (1)	ZA858117B (2)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4568741A (en) *	1984-05-15	1986-02-04	The Upjohn Company	Synthesis of 7-halo-7-deoxylincomycins
JP2531877Y2 (ja) *	1988-12-15	1997-04-09	日東工器株式会社	電磁式ダイアフラムポンプ
JP2531876Y2 (ja) *	1988-12-15	1997-04-09	日東工器株式会社	電磁式ダイアフラムポンプ用マグネットホルダ
JP2544782Y2 (ja) *	1988-12-27	1997-08-20	日東工器株式会社	電磁式ダイアフラムポンプ用マグネットホルダ
US6565882B2 (en)	2000-02-24	2003-05-20	Advancis Pharmaceutical Corp	Antibiotic composition with inhibitor
US6544555B2 (en)	2000-02-24	2003-04-08	Advancis Pharmaceutical Corp.	Antibiotic product, use and formulation thereof
US20020068078A1 (en)	2000-10-13	2002-06-06	Rudnic Edward M.	Antifungal product, use and formulation thereof
US6541014B2 (en)	2000-10-13	2003-04-01	Advancis Pharmaceutical Corp.	Antiviral product, use and formulation thereof
DE60204897T2 (de) *	2001-08-28	2006-05-11	Pharmacia Corp.	Kristalline freie base von clindamycin
KR20050056195A (ko) *	2002-08-15	2005-06-14	비큐론 파마슈티컬스 인코포레이티드	항박테리아 작용을 갖는 링코마이신 유도체
US7199105B2 (en) *	2002-08-15	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
EA014372B1 (ru)	2003-01-24	2010-10-29	Стифел Рисерч Оустрэйлиа Пти Лтд.	Пена на основе фосфата клиндамицина
US7199106B2 (en)	2003-06-17	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antimicrobial activity
US7256177B2 (en)	2003-06-17	2007-08-14	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
AU2004258953B2 (en)	2003-07-21	2011-02-10	Shionogi, Inc.	Antibiotic product, use and formulation thereof
WO2005009365A2 (en)	2003-07-21	2005-02-03	Advancis Pharmaceutical Corporation	Antibiotic product, use and formulation thereof
CA2533358C (en)	2003-07-21	2014-03-11	Advancis Pharmaceutical Corporation	Antibiotic product, use and formulation thereof
US8758820B2 (en)	2003-08-11	2014-06-24	Shionogi Inc.	Robust pellet
JP2007502294A (ja)	2003-08-12	2007-02-08	アドバンシスファーマスーティカルコーポレイション	抗生物質製剤、その使用法及び作成方法
US8246996B2 (en)	2003-08-29	2012-08-21	Shionogi Inc.	Antibiotic product, use and formulation thereof
JP2007513869A (ja)	2003-09-15	2007-05-31	アドバンシスファーマスーティカルコーポレイション	抗生物質製剤、その使用法及び作成方法
US7361743B2 (en) *	2004-02-11	2008-04-22	Pfizer Inc	Lincomycin derivatives possessing antibacterial activity
US8715727B2 (en)	2004-07-02	2014-05-06	Shionogi Inc.	Tablet for pulsed delivery
US8357394B2 (en)	2005-12-08	2013-01-22	Shionogi Inc.	Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en)	2006-12-04	2014-07-15	Shionogi Inc.	Modified release amoxicillin products
AU2007220123A1 (en) *	2006-02-28	2007-09-07	V.B. Medicare Pvt. Ltd.	Process for the production of a chlorinating reagent and its use in the preparation of chlorinated sugars
ES2560540T3 (es)	2006-03-31	2016-02-19	Stiefel Research Australia Pty Ltd	Gel en suspensión espumable
US8299052B2 (en)	2006-05-05	2012-10-30	Shionogi Inc.	Pharmaceutical compositions and methods for improved bacterial eradication
CN101205245B (zh) *	2007-12-06	2011-04-06	河南天方药业股份有限公司	盐酸克林霉素的制备方法
CN102675146A (zh) *	2012-05-22	2012-09-19	山东凯盛新材料股份有限公司	新型固体氯化剂（氯亚甲基）二甲基氯化铵的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3496163A (en) *	1965-02-08	1970-02-17	Upjohn Co	7-halo-7-deoxylincomycins and process for preparing the same
US3435025A (en) *	1966-03-18	1969-03-25	Upjohn Co	7-deoxylincomycin and analogs and isomers thereof and process for making the same
US3580904A (en) *	1969-04-03	1971-05-25	Upjohn Co	7-halo-7-deoxy-lincomycin derivatives
US3574186A (en) *	1969-10-08	1971-04-06	Upjohn Co	Process for making 7-chloro-7-deoxylincomycin and related compounds and novel intermediates produced therein
US4568741A (en) *	1984-05-15	1986-02-04	The Upjohn Company	Synthesis of 7-halo-7-deoxylincomycins

1985
- 1985-04-01 CN CN85101921.8A patent/CN1004002B/zh not_active Expired
- 1985-10-11 CA CA000492862A patent/CA1238319A/en not_active Expired
- 1985-10-18 AU AU48837/85A patent/AU574232B2/en not_active Expired
- 1985-10-22 ZA ZA858117A patent/ZA858117B/xx unknown
- 1985-10-22 IL IL76778A patent/IL76778A/xx not_active IP Right Cessation
- 1985-10-23 ES ES548152A patent/ES8605817A1/es not_active Expired
- 1985-11-14 CN CN85108244A patent/CN1016694B/zh not_active Expired
- 1985-11-14 PT PT81496A patent/PT81496B/pt unknown
- 1985-11-19 MX MX661A patent/MX162251A/es unknown
- 1985-11-22 DK DK542785A patent/DK165010C/da not_active IP Right Cessation
- 1985-11-25 AT AT85308539T patent/ATE50265T1/de not_active IP Right Cessation
- 1985-11-25 DE DE8585308539T patent/DE3575930D1/de not_active Expired - Lifetime
- 1985-11-25 EP EP85308539A patent/EP0183505B1/en not_active Expired - Lifetime
- 1985-11-27 GR GR852861A patent/GR852861B/el unknown
- 1985-11-28 SU SU853984283A patent/SU1405705A3/ru active
- 1985-11-28 JP JP60269229A patent/JPH0649714B2/ja not_active Expired - Lifetime
- 1985-11-28 FI FI854711A patent/FI78708C/fi not_active IP Right Cessation
- 1985-11-28 KR KR1019850008893A patent/KR930003492B1/ko not_active Expired - Lifetime
- 1985-11-29 HU HU854580A patent/HU199497B/hu unknown
1986
- 1986-01-24 US US06/822,044 patent/US4710565A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CA1238319A (en)	1988-06-21
EP0183505A3 (en)	1987-06-24
IL76778A0 (en)	1986-02-28
EP0183505B1 (en)	1990-02-07
DK542785A (da)	1986-05-30
CN85101921A (zh)	1987-01-10
ATE50265T1 (de)	1990-02-15
SU1405705A3 (ru)	1988-06-23
EP0183505A2 (en)	1986-06-04
DK165010C (da)	1993-02-22
JPH0649714B2 (ja)	1994-06-29
HUT40806A (en)	1987-02-27
DK165010B (da)	1992-09-28
CN1016694B (zh)	1992-05-20
FI854711A0 (fi)	1985-11-28
KR860004077A (ko)	1986-06-16
ES548152A0 (es)	1986-04-01
JPS61137892A (ja)	1986-06-25
MX162251A (es)	1991-04-17
GR852861B (2)	1986-03-28
DK542785D0 (da)	1985-11-22
CN1004002B (zh)	1989-04-26
HU199497B (en)	1990-02-28
FI854711L (fi)	1986-05-30
FI78708B (fi)	1989-05-31
DE3575930D1 (de)	1990-03-15
IL76778A (en)	1991-09-16
ZA858117B (en)	1986-06-25
KR930003492B1 (ko)	1993-05-01
PT81496A (en)	1985-12-01
CN85108244A (zh)	1986-08-20
FI78708C (fi)	1989-09-11
AU4883785A (en)	1986-06-05
US4710565A (en)	1987-12-01
PT81496B (pt)	1987-11-11
AU574232B2 (en)	1988-06-30

Legal Events

Date	Code	Title	Description
1998-04-16	PC1A	Transfer granted
2008-03-16	FD1A	Patent lapsed	Effective date: 20051219

Publication	Publication Date	Title
ES8605817A1 (es)	1986-04-01	Procedimiento para preparar un compuesto seleccionado del grupo constituido de 7-halo-7-desoxilincomicina y analogos de la misma
ES2110003T3 (es)	1998-02-01	Nuevas composiciones a base de derivados de la clase de los taxanos.
ES8802017A1 (es)	1988-03-16	Un procedimiento para preparar derivados de diamidas sustituidas con 7-oxabicicloheptano y sus analogos de prostaglandina
ES2061660T3 (es)	1994-12-16	Eteres azabiciclicos.
AR223143A1 (es)	1981-07-31	Un procedimiento para preparar el isomero sin de los compuestos del acido 3-cefem-4-carboxilico sustituido en las posiciones 3 y 7
ES8800132A1 (es)	1987-10-16	Un procedimiento para la produccion de compuestos de fenetanolamina
ES8801284A1 (es)	1987-12-16	Procedimiento para preparar nuevos compuestos de benzotiofeno y benzofurano
IT1036091B (it)	1979-10-30	Apparecchiatura per la fornitura di filo a telai rettilineei per maglieria
ES8705408A1 (es)	1987-05-01	Un procedimiento para preparar un derivado de 1,5-benzotiazepina.
AR241017A2 (es)	1991-04-30	"procedimiento para la preparacion de fenil-silfonil-oxi-bencimidazol-carbamatos sustituidos."
AR240924A2 (es)	1991-03-27	"procedimiento para preparar derivados de 1,3-oxazolidin-2-ona y sus sales".
ES2038974T3 (es)	1993-08-16	Metodo para incrementar selectivamente la proporcion de componentes principales individuales del complejo antibiotico a/16686.
ES8505179A1 (es)	1985-05-16	Un procedimiento para la preparacion de imidazobenzodiacepinas
ES8607299A1 (es)	1986-06-01	Procedimiento para preparar (2-oxo-1,2,3,5-tetrahidroimida- zo(2,1-b)quinazolinil)-oxialquilamidas
IT1042479B (it)	1980-01-30	Procedimento per risolvere otticamente la dl 2 4 idrossifeil glicina
ES8506270A1 (es)	1985-07-01	Un procedimiento para preparar compuestos analogos de la 7-oxabicicloheptano-prostaglandina
IT1054584B (it)	1981-11-30	Modificazione cristallina del cloruro di magnesio anidro
IT1037434B (it)	1979-11-10	Procedimento di preparazione di espansi di poliuretano ad elasticita migltorata
IT1078054B (it)	1985-05-08	Apparecchiature per rivelare la trama in macchine per tessitura senza navetta
AR241015A2 (es)	1991-04-30	"procedimiento para preparar acidos 16-fenoxiprostatrienoicos"
IT1089104B (it)	1985-06-18	Disposizione per la inserzione di fili di trama
ES8505962A1 (es)	1985-06-16	Un procedimiento para preparar nuevos derivados amidinicos de 4-fenilimidazol sustituido en la posicion 2
ES478328A1 (es)	1979-11-01	Un procedimiento para la preparacion de nuevos derivados de pirido 2,1-b quinazolina.
ES8401485A1 (es)	1983-12-01	Un procedimiento de preparacion de nuevas 8-(3-(1,2-bencisoxazol-3-il)propil)-1-fenil-1,3,8-triazaspiro(4,5)decan-4-onas.
ES2135384T3 (es)	1999-11-01	Derivados de 1,4-dihidropiridina opticamente activos y procedimientos para producirlos.