FR2436145A1 - Derive de 3,4-dihydroxy-cinnamaldehyde, procede pour sa preparation et medicament le contenant - Google Patents

Derive de 3,4-dihydroxy-cinnamaldehyde, procede pour sa preparation et medicament le contenant

Info

Publication number
FR2436145A1
FR2436145A1 FR7923013A FR7923013A FR2436145A1 FR 2436145 A1 FR2436145 A1 FR 2436145A1 FR 7923013 A FR7923013 A FR 7923013A FR 7923013 A FR7923013 A FR 7923013A FR 2436145 A1 FR2436145 A1 FR 2436145A1
Authority
FR
France
Prior art keywords
dihydroxy
cinnamaldehyde
preparation
product
medicinal container
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
FR7923013A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Madaus Holding GmbH
Original Assignee
Dr Madaus GmbH and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Madaus GmbH and Co filed Critical Dr Madaus GmbH and Co
Publication of FR2436145A1 publication Critical patent/FR2436145A1/fr
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Steroid Compounds (AREA)

Abstract

L'invention concerne la préparation d'un dérivé de 3,4-dihydroxy-cinnamaldéhyde. On peut obtenir le composé désigné sous le nom de Americanine soit par diverses étapes d'extraction des fruits broyés et séchés de Phytolacca americana, soit par voie synthétique par dimérisation de 3,4-dihydroxy-cinnamaldéhyde et d'alcool 3,4-dihydroxycinnamique par addition oxydante ou par réaction de 3,4-dihydrozy-cinnamaldéhyde et d'allylpyrocatéchine en présence d'un oxydant; à acétyler le produit résultant, à oxyder les radicaux méthyle en fonction alcool et à saponifier le produit obtenu avec un alcali faible. Le produit est approprié à titre de médicament pour le traitement de certaines hépatopathies.
FR7923013A 1978-09-16 1979-09-14 Derive de 3,4-dihydroxy-cinnamaldehyde, procede pour sa preparation et medicament le contenant Pending FR2436145A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19782840467 DE2840467A1 (de) 1978-09-16 1978-09-16 3,4-dihydroxizimtaldehydderivat, dessen herstellung und arzneimittel

Publications (1)

Publication Number Publication Date
FR2436145A1 true FR2436145A1 (fr) 1980-04-11

Family

ID=6049691

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7923013A Pending FR2436145A1 (fr) 1978-09-16 1979-09-14 Derive de 3,4-dihydroxy-cinnamaldehyde, procede pour sa preparation et medicament le contenant

Country Status (18)

Country Link
JP (1) JPS5559182A (fr)
AR (3) AR221900A1 (fr)
AT (1) AT367417B (fr)
BE (1) BE878824A (fr)
CA (1) CA1128532A (fr)
CS (3) CS221521B2 (fr)
DE (1) DE2840467A1 (fr)
ES (3) ES8101578A1 (fr)
FR (1) FR2436145A1 (fr)
GB (1) GB2035300B (fr)
IT (1) IT7925651A0 (fr)
LU (1) LU81679A1 (fr)
NL (1) NL7906881A (fr)
PL (1) PL120977B1 (fr)
PT (1) PT70177A (fr)
SE (1) SE7907656L (fr)
SU (1) SU925246A3 (fr)
ZA (1) ZA794815B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2851919A1 (fr) * 2003-03-03 2004-09-10 Lmd Lignanes utilisables comme inhibiteurs de cathepsines et leurs applications

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2428680A1 (de) * 1974-06-14 1976-01-02 Madaus & Co Dr Neue substituierte 1-(2',4',6'/rihydroxyphenyl)-propandion-(1,2)- verbindungen und arzneimittel

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2428680A1 (de) * 1974-06-14 1976-01-02 Madaus & Co Dr Neue substituierte 1-(2',4',6'/rihydroxyphenyl)-propandion-(1,2)- verbindungen und arzneimittel

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
EXBK/78 *

Also Published As

Publication number Publication date
PL218339A1 (fr) 1980-12-01
GB2035300B (en) 1983-03-23
ATA607979A (de) 1981-11-15
IT7925651A0 (it) 1979-09-12
GB2035300A (en) 1980-06-18
ZA794815B (en) 1980-10-29
AR226094A1 (es) 1982-05-31
SU925246A3 (ru) 1982-04-30
SE7907656L (sv) 1980-03-17
ES484202A0 (es) 1980-12-16
LU81679A1 (de) 1980-01-24
AR225070A1 (es) 1982-02-15
ES8101580A1 (es) 1980-12-16
CA1128532A (fr) 1982-07-27
PT70177A (de) 1979-10-01
AT367417B (de) 1982-07-12
JPS5559182A (en) 1980-05-02
NL7906881A (nl) 1980-03-18
ES8101579A1 (es) 1980-12-16
CS221523B2 (en) 1983-04-29
ES8101578A1 (es) 1980-12-16
AR221900A1 (es) 1981-03-31
CS221521B2 (en) 1983-04-29
DE2840467A1 (de) 1980-03-20
ES488141A0 (es) 1980-12-16
BE878824A (fr) 1980-03-17
ES488140A0 (es) 1980-12-16
PL120977B1 (en) 1982-04-30
CS221522B2 (en) 1983-04-29

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