HRP20010862A2 - New pharmaceutical combinations for nos inhibitors - Google Patents

New pharmaceutical combinations for nos inhibitors Download PDF

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Publication number
HRP20010862A2
HRP20010862A2 HR20010862A HRP20010862A HRP20010862A2 HR P20010862 A2 HRP20010862 A2 HR P20010862A2 HR 20010862 A HR20010862 A HR 20010862A HR P20010862 A HRP20010862 A HR P20010862A HR P20010862 A2 HRP20010862 A2 HR P20010862A2
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HR
Croatia
Prior art keywords
pyridin
phenyl
ylamine
amino
ethoxy
Prior art date
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HR20010862A
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English (en)
Croatian (hr)
Inventor
Mario David Saltarelli
John Adams Lowe Iii
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Pfizer Prod Inc
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Publication date
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Publication of HRP20010862A2 publication Critical patent/HRP20010862A2/hr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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HR20010862A 1999-05-21 2000-03-16 New pharmaceutical combinations for nos inhibitors HRP20010862A2 (en)

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DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
UA82517C2 (uk) 2003-06-24 2008-04-25 Ньюросерч А/С Нові похідні 8-аза-біцикло[3.2.1]октану та їх застосування як інгібіторів ресорбції моноамінових медіаторів
EP1634598A1 (en) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Use of piperazine derivatives and analogues for the manufacture of a medicament for the prophylaxis and/or treatment of disorders of food ingestion
WO2008148840A1 (en) 2007-06-08 2008-12-11 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
PE20090362A1 (es) 2007-06-08 2009-04-04 Janssen Pharmaceutica Nv Derivados de piperidina/piperazina como moduladores de dgat
AU2008258560C1 (en) 2007-06-08 2014-04-10 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
PE20140572A1 (es) 2008-06-05 2014-05-16 Janssen Pharmaceutica Nv Combinaciones de drogas que comprenden un inhibidor de dgat y un agonista de ppar
EP2404902A1 (en) * 2009-03-05 2012-01-11 Shionogi&Co., Ltd. Piperidine and pyrrolidine derivatives having npy y5 receptor antagonism
WO2014078568A1 (en) 2012-11-14 2014-05-22 The Johns Hopkins University Methods and compositions for treating schizophrenia
WO2020252383A2 (en) * 2019-06-14 2020-12-17 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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DZ3041A1 (fr) 2004-03-27
EA200101110A1 (ru) 2002-08-29
NO20015651D0 (no) 2001-11-20
GT200000071A (es) 2001-11-08
TR200103351T2 (tr) 2002-06-21
PL358538A1 (pl) 2004-08-09
MXPA01011978A (es) 2002-05-06
OA11943A (en) 2006-04-12
IL145955A0 (en) 2002-07-25
CN1617743A (zh) 2005-05-18
AU2935300A (en) 2000-12-12
CA2374668A1 (en) 2000-11-30
IS6126A (is) 2001-10-26
KR20020010916A (ko) 2002-02-06
SK16602001A3 (sk) 2003-03-04
EE200100611A (et) 2003-02-17
WO2000071107A2 (en) 2000-11-30
HN2000000045A (es) 2001-03-02
AR022640A1 (es) 2002-09-04
EP1178784A1 (en) 2002-02-13
NO20015651L (no) 2002-01-18
AP2001002326A0 (en) 2001-12-31
PA8494601A1 (es) 2002-08-29
UY26148A1 (es) 2000-12-29
PE20010157A1 (es) 2001-02-16
BR0010820A (pt) 2002-03-05
HUP0301287A2 (hu) 2003-08-28
CO5160295A1 (es) 2002-05-30
ZA200109555B (en) 2004-04-07
MA26732A1 (fr) 2004-12-20
TNSN00106A1 (fr) 2005-11-10
HUP0301287A3 (en) 2005-03-29
JP2003523941A (ja) 2003-08-12
BG106208A (en) 2002-09-30
WO2000071107A8 (en) 2002-01-24

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