MA26732A1 - Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation - Google Patents

Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation

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Publication number
MA26732A1
MA26732A1 MA25976A MA25976A MA26732A1 MA 26732 A1 MA26732 A1 MA 26732A1 MA 25976 A MA25976 A MA 25976A MA 25976 A MA25976 A MA 25976A MA 26732 A1 MA26732 A1 MA 26732A1
Authority
MA
Morocco
Prior art keywords
preparation
inhibitor
pharmaceutical composition
novel pharmaceutical
treatment
Prior art date
Application number
MA25976A
Other languages
English (en)
Inventor
David Saltarelli Mario
Adams Lowe John Iii
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA26732A1 publication Critical patent/MA26732A1/fr

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/13—Amines
    • A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

L'INVENTION CONCERNE DES COMPOSITIONS PHARMACEUTIQUES COMPRENANT UN COMPOSÉ INHIBITEUR DE NOS, SEUL OU EN ASSOCIATION AVEC UN ANTAGONISTE DES RÉCEPTEURS DE NK-1 OU UN SSRI. ELLE CONCERNE ÉGALEMENT UN PROCÉDÉ POUR LEUR PRÉPARATION. - APPLICATION : UTILISATION DE CES COMPOSITIONS POUR LE TRAITEMENT DE DIVERS TROUBLES DONT LE TRAITEMENT PEUT eTRE EFFECTUÉ OU FACILITÉ PAR LA MODOFICATION DES RYTHMES CIRCADIENS.
MA25976A 1999-05-21 2000-05-17 Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation MA26732A1 (fr)

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JP (1) JP2003523941A (fr)
KR (1) KR20020010916A (fr)
CN (1) CN1617743A (fr)
AP (1) AP2001002326A0 (fr)
AR (1) AR022640A1 (fr)
AU (1) AU2935300A (fr)
BG (1) BG106208A (fr)
BR (1) BR0010820A (fr)
CA (1) CA2374668A1 (fr)
CO (1) CO5160295A1 (fr)
DZ (1) DZ3041A1 (fr)
EA (1) EA200101110A1 (fr)
EE (1) EE200100611A (fr)
GT (1) GT200000071A (fr)
HN (1) HN2000000045A (fr)
HR (1) HRP20010862A2 (fr)
HU (1) HUP0301287A3 (fr)
IL (1) IL145955A0 (fr)
IS (1) IS6126A (fr)
MA (1) MA26732A1 (fr)
MX (1) MXPA01011978A (fr)
NO (1) NO20015651L (fr)
OA (1) OA11943A (fr)
PA (1) PA8494601A1 (fr)
PE (1) PE20010157A1 (fr)
PL (1) PL358538A1 (fr)
SK (1) SK16602001A3 (fr)
TN (1) TNSN00106A1 (fr)
TR (1) TR200103351T2 (fr)
UY (1) UY26148A1 (fr)
WO (1) WO2000071107A2 (fr)
ZA (1) ZA200109555B (fr)

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Publication number Priority date Publication date Assignee Title
DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
AU2004249441B2 (en) * 2003-06-24 2009-11-12 Neurosearch A/S Novel 8-aza-bicyclo(3.2.1)octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
EP2152271B1 (fr) 2007-06-08 2015-10-21 Janssen Pharmaceutica, N.V. Dérivés de piperidine/piperazine
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
CA2687918C (fr) 2007-06-08 2016-11-08 Janssen Pharmaceutica N.V. Derives de piperidine/piperazine
AU2008258487B2 (en) 2007-06-08 2012-11-15 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
JP5579170B2 (ja) 2008-06-05 2014-08-27 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｄｇａｔ阻害剤とｐｐａｒ作動薬を含有する薬剤組み合わせ物
US8889674B2 (en) 2009-03-05 2014-11-18 Shionogi & Co., Ltd. Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism
JP6440625B2 (ja) 2012-11-14 2018-12-19 ザ・ジョンズ・ホプキンス・ユニバーシティー 精神分裂病を処置するための方法および組成物
US20220267269A1 (en) * 2019-06-14 2022-08-25 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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HN2000000045A (es) 2001-03-02
EP1178784A1 (fr) 2002-02-13
EA200101110A1 (ru) 2002-08-29
PL358538A1 (en) 2004-08-09
CN1617743A (zh) 2005-05-18
IS6126A (is) 2001-10-26
AP2001002326A0 (en) 2001-12-31
KR20020010916A (ko) 2002-02-06
NO20015651L (no) 2002-01-18
EE200100611A (et) 2003-02-17
HRP20010862A2 (en) 2003-06-30
BR0010820A (pt) 2002-03-05
NO20015651D0 (no) 2001-11-20
JP2003523941A (ja) 2003-08-12
CA2374668A1 (fr) 2000-11-30
DZ3041A1 (fr) 2004-03-27
HUP0301287A3 (en) 2005-03-29
GT200000071A (es) 2001-11-08
IL145955A0 (en) 2002-07-25
TR200103351T2 (tr) 2002-06-21
OA11943A (en) 2006-04-12
SK16602001A3 (sk) 2003-03-04
TNSN00106A1 (fr) 2005-11-10
WO2000071107A2 (fr) 2000-11-30
BG106208A (en) 2002-09-30
CO5160295A1 (es) 2002-05-30
UY26148A1 (es) 2000-12-29
HUP0301287A2 (hu) 2003-08-28
AR022640A1 (es) 2002-09-04
PA8494601A1 (es) 2002-08-29
AU2935300A (en) 2000-12-12
MXPA01011978A (es) 2002-05-06
PE20010157A1 (es) 2001-02-16
ZA200109555B (en) 2004-04-07
WO2000071107A8 (fr) 2002-01-24

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