HRP20110048T1 - Spojevi piperidina i njihova upotreba - Google Patents

Spojevi piperidina i njihova upotreba Download PDF

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Publication number
HRP20110048T1
HRP20110048T1 HR20110048T HRP20110048T HRP20110048T1 HR P20110048 T1 HRP20110048 T1 HR P20110048T1 HR 20110048 T HR20110048 T HR 20110048T HR P20110048 T HRP20110048 T HR P20110048T HR P20110048 T1 HRP20110048 T1 HR P20110048T1
Authority
HR
Croatia
Prior art keywords
methyl
thiazole
amino
dichloro
carbonyl
Prior art date
Application number
HR20110048T
Other languages
English (en)
Croatian (hr)
Inventor
Basarab Gregory
Hill Pamela
Zhou Fei
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HRP20110048T1 publication Critical patent/HRP20110048T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HR20110048T 2007-06-12 2008-06-11 Spojevi piperidina i njihova upotreba HRP20110048T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94344007P 2007-06-12 2007-06-12
PCT/GB2008/050431 WO2008152418A1 (en) 2007-06-12 2008-06-11 Piperidine compounds and uses thereof

Publications (1)

Publication Number Publication Date
HRP20110048T1 true HRP20110048T1 (hr) 2011-03-31

Family

ID=39673349

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110048T HRP20110048T1 (hr) 2007-06-12 2008-06-11 Spojevi piperidina i njihova upotreba

Country Status (29)

Country Link
US (1) US20080312255A1 (de)
EP (1) EP2158199B1 (de)
JP (1) JP2010529184A (de)
KR (1) KR20100038095A (de)
CN (1) CN102648199A (de)
AR (1) AR066977A1 (de)
AT (1) ATE488514T1 (de)
AU (1) AU2008263580A1 (de)
BR (1) BRPI0812473A2 (de)
CA (1) CA2689076A1 (de)
CL (1) CL2008001740A1 (de)
CO (1) CO6311102A2 (de)
CY (1) CY1111442T1 (de)
DE (1) DE602008003575D1 (de)
DK (1) DK2158199T3 (de)
ES (1) ES2354647T3 (de)
HR (1) HRP20110048T1 (de)
IL (1) IL202367A0 (de)
MX (1) MX2009013501A (de)
NZ (1) NZ582516A (de)
PE (1) PE20090555A1 (de)
PL (1) PL2158199T3 (de)
PT (1) PT2158199E (de)
RU (1) RU2010100352A (de)
SA (1) SA08290357B1 (de)
SI (1) SI2158199T1 (de)
TW (1) TW200906412A (de)
UY (1) UY31141A1 (de)
WO (1) WO2008152418A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ561613A (en) 2005-02-18 2010-12-24 Astrazeneca Ab Antibacterial piperidine derivatives
TW201026695A (en) * 2008-12-12 2010-07-16 Astrazeneca Ab Piperidine compounds and uses thereof-596
TW201026694A (en) * 2008-12-12 2010-07-16 Astrazeneca Ab Compound 468
WO2011024004A1 (en) 2009-08-26 2011-03-03 Astrazeneca Ab Heterocyclic urea derivatives useful for treatment of bacterial infection
US9364405B2 (en) 2013-03-13 2016-06-14 Avon Products, Inc. Tyrosinase inhibitors
US20150174034A1 (en) 2013-03-13 2015-06-25 Avon Products, Inc. Tyrosinase inhibitors
KR20180054650A (ko) 2015-09-30 2018-05-24 다이이찌 산쿄 가부시키가이샤 히드록시알킬 티아디아졸 유도체
EP3596071A1 (de) 2017-03-14 2020-01-22 Daiichi Sankyo Company, Limited N-phosphonoxymethyl-prodrugs von hydroxyalkylthiadiazolderivaten
CA3057431A1 (en) 2017-03-24 2018-09-27 Taisho Pharmaceutical Co., Ltd. 2(1h)-quinolinone derivative
WO2020048949A1 (en) 2018-09-03 2020-03-12 Univerza V Ljubljani New class of dna gyrase and/or topoisomerase iv inhibitors with activity against gram-positive and gram-negative bacteria
CN110172435B (zh) * 2019-06-06 2020-12-29 江南大学 一种催化合成2,5-二甲基吡嗪的重组菌
EP4263503A1 (de) 2020-12-17 2023-10-25 Univerza V Ljubljani Neue n-phenylpyrrolamid-inhibitoren der dna-gyrase und topoisomerase iv mit antibakterieller wirkung
CN115466246B (zh) * 2021-06-11 2024-02-06 中国医学科学院药物研究所 吡咯酰哌啶胺类化合物及其用途

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3963480A (en) * 1973-04-11 1976-06-15 Sterling Drug Inc. Herbicidal pyrrole-2-carboxamides
US4046775A (en) * 1973-04-11 1977-09-06 Sterling Drug Inc. 4,5-Dihalopyrrole-2-carboxamides
US4791112A (en) * 1987-02-02 1988-12-13 The Boc Group, Inc. N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds
US4912109A (en) * 1987-02-02 1990-03-27 Boc, Inc. N-heterocyclic-N-(4-piperidinyl) amides and pharmaceutical compositions and methods employing such compounds
US5739135A (en) * 1993-09-03 1998-04-14 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
EA005680B1 (ru) * 2000-01-18 2005-04-28 Вертекс Фармасьютикалз Инкорпорейтед Ингибиторы гиразы и их применение для лечения бактериальной инфекции
DE60309701T2 (de) * 2002-06-13 2007-09-06 Vertex Pharmaceuticals Inc., Cambridge 2-ureido-6-heteroaryl-3h-benzoimidazol-4-carbonsäurederivate und verwandte verbindungen als gyrase und/oder topoisomerase iv inhibitoren zur behandlung von bakteriellen infektionen
TW200526626A (en) * 2003-09-13 2005-08-16 Astrazeneca Ab Chemical compounds
GB0321509D0 (en) * 2003-09-13 2003-10-15 Astrazeneca Ab Chemical compounds
US20050197336A1 (en) * 2004-03-08 2005-09-08 Miikana Therapeutics Corporation Inhibitors of histone deacetylase
US7345043B2 (en) * 2004-04-01 2008-03-18 Miikana Therapeutics Inhibitors of histone deacetylase
NZ561613A (en) * 2005-02-18 2010-12-24 Astrazeneca Ab Antibacterial piperidine derivatives
TW200819437A (en) * 2006-08-17 2008-05-01 Astrazeneca Ab Chemical compounds

Also Published As

Publication number Publication date
DE602008003575D1 (de) 2010-12-30
NZ582516A (en) 2012-03-30
CL2008001740A1 (es) 2009-07-17
WO2008152418A1 (en) 2008-12-18
CY1111442T1 (el) 2015-08-05
PL2158199T3 (pl) 2011-04-29
ES2354647T3 (es) 2011-03-16
MX2009013501A (es) 2010-01-18
DK2158199T3 (da) 2011-02-07
CA2689076A1 (en) 2008-12-18
BRPI0812473A2 (pt) 2014-12-02
HK1140198A1 (en) 2010-10-08
US20080312255A1 (en) 2008-12-18
TW200906412A (en) 2009-02-16
ATE488514T1 (de) 2010-12-15
EP2158199B1 (de) 2010-11-17
CN102648199A (zh) 2012-08-22
AU2008263580A1 (en) 2008-12-18
PT2158199E (pt) 2011-01-19
JP2010529184A (ja) 2010-08-26
AR066977A1 (es) 2009-09-23
CO6311102A2 (es) 2011-08-22
PE20090555A1 (es) 2009-06-04
UY31141A1 (es) 2009-01-30
KR20100038095A (ko) 2010-04-12
RU2010100352A (ru) 2011-07-20
SI2158199T1 (sl) 2011-02-28
IL202367A0 (en) 2010-06-30
SA08290357B1 (ar) 2011-06-22
EP2158199A1 (de) 2010-03-03

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