HRP20120681T1 - Stabilni kristal 4-oksokinolinskog spoja - Google Patents

Stabilni kristal 4-oksokinolinskog spoja Download PDF

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Publication number
HRP20120681T1
HRP20120681T1 HRP20120681TT HRP20120681T HRP20120681T1 HR P20120681 T1 HRP20120681 T1 HR P20120681T1 HR P20120681T T HRP20120681T T HR P20120681TT HR P20120681 T HRP20120681 T HR P20120681T HR P20120681 T1 HRP20120681 T1 HR P20120681T1
Authority
HR
Croatia
Prior art keywords
crystal
crystal according
ray powder
mixed
dihydroquinoline
Prior art date
Application number
HRP20120681TT
Other languages
English (en)
Croatian (hr)
Inventor
Satoh Motohide
Motomura Takahisa
Matsuda Takashi
Kondo Kentaro
Ando Koji
Matsuda Koji
Miyake Shuji
Uehara Hideto
Original Assignee
Japan Tobacco
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079161&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20120681(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco filed Critical Japan Tobacco
Publication of HRP20120681T1 publication Critical patent/HRP20120681T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
HRP20120681TT 2004-05-20 2005-05-19 Stabilni kristal 4-oksokinolinskog spoja HRP20120681T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2004150979 2004-05-20
PCT/JP2005/009604 WO2005113508A1 (en) 2004-05-20 2005-05-19 Stable crystal of 4-oxoquinoline compound

Publications (1)

Publication Number Publication Date
HRP20120681T1 true HRP20120681T1 (hr) 2012-09-30

Family

ID=35079161

Family Applications (2)

Application Number Title Priority Date Filing Date
HRP20231588TT HRP20231588T3 (hr) 2004-05-20 2005-05-19 Kombinacija koja sadrži stabilni kristal 4-oksokinolinskog spoja
HRP20120681TT HRP20120681T1 (hr) 2004-05-20 2005-05-19 Stabilni kristal 4-oksokinolinskog spoja

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HRP20231588TT HRP20231588T3 (hr) 2004-05-20 2005-05-19 Kombinacija koja sadrži stabilni kristal 4-oksokinolinskog spoja

Country Status (33)

Country Link
US (7) US7635704B2 (lt)
EP (4) EP2514746A1 (lt)
JP (1) JP3754064B2 (lt)
KR (1) KR20080064909A (lt)
CN (1) CN1956961B (lt)
AR (2) AR049280A1 (lt)
AU (1) AU2005245296B2 (lt)
BE (1) BE2024C511I2 (lt)
BR (1) BRPI0510114B8 (lt)
CA (1) CA2566922C (lt)
CY (4) CY1113010T1 (lt)
DK (2) DK3281939T3 (lt)
ES (2) ES2960824T3 (lt)
FI (2) FI3281939T3 (lt)
FR (1) FR23C1040I1 (lt)
HR (2) HRP20231588T3 (lt)
HU (2) HUE064615T2 (lt)
IL (1) IL179250A0 (lt)
LT (2) LT3281939T (lt)
LU (1) LUC00334I2 (lt)
MX (1) MXPA06013405A (lt)
MY (1) MY134672A (lt)
NO (8) NO339223B1 (lt)
NZ (1) NZ551839A (lt)
PE (2) PE20120361A1 (lt)
PL (2) PL1636190T3 (lt)
PT (2) PT1636190E (lt)
RS (2) RS52375B (lt)
RU (1) RU2330845C1 (lt)
SI (2) SI3281939T1 (lt)
TW (1) TWI329015B (lt)
WO (1) WO2005113508A1 (lt)
ZA (1) ZA200610647B (lt)

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AR068403A1 (es) 2007-09-11 2009-11-18 Gilead Sciences Inc Proceso e intermediarios para la preparacion de inhibidores de integrasa
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WO2010137032A2 (en) * 2009-05-14 2010-12-02 Matrix Laboratories Ltd. Novel polymorphic forms of elvitegravir and its pharmaceutically acceptable salts
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KR101663436B1 (ko) 2012-07-06 2016-10-06 제넨테크, 인크. N-치환된 벤즈아미드 및 이의 사용 방법
CA2878699C (en) 2012-08-03 2018-09-11 Gilead Sciences, Inc. Process and intermediates for preparing integrase inhibitors
CN103819402B (zh) * 2012-11-17 2016-03-30 上海迪赛诺化学制药有限公司 埃替拉韦中间体及其制备方法和应用
CN103864682B (zh) * 2012-12-18 2016-12-28 上海迪赛诺化学制药有限公司 一种制备iii型埃替拉韦晶体的方法
EA030003B1 (ru) 2012-12-21 2018-06-29 Джилид Сайэнс, Инк. Полициклическое карбамоилпиридоновое соединение и его фармацевтическое применение для лечения вич-инфекции
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TWI677489B (zh) 2014-06-20 2019-11-21 美商基利科學股份有限公司 多環型胺甲醯基吡啶酮化合物之合成
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Also Published As

Publication number Publication date
US20180029989A1 (en) 2018-02-01
LTPA2024001I1 (lt) 2024-04-10
AR096100A2 (es) 2015-12-09
RS52375B (sr) 2012-12-31
EP1636190B1 (en) 2012-06-27
BRPI0510114B8 (pt) 2021-05-25
NO20220690A1 (no) 2007-02-07
CY2024008I2 (el) 2024-09-20
LT3281939T (lt) 2023-11-27
PL3281939T3 (pl) 2024-03-18
CY2015009I1 (el) 2024-09-20
CY1113010T1 (el) 2016-04-13
US7635704B2 (en) 2009-12-22
EP4299563A3 (en) 2024-02-28
CY2015009I2 (el) 2024-09-20
NO339223B1 (no) 2016-11-21
PT3281939T (pt) 2023-11-22
SI1636190T1 (sl) 2012-09-28
NO20190051A1 (no) 2007-02-07
ES2388441T3 (es) 2012-10-15
US20190185433A1 (en) 2019-06-20
NO20230913A1 (no) 2007-02-07
PL1636190T3 (pl) 2012-10-31
EP4299563A2 (en) 2024-01-03
RS64845B1 (sr) 2023-12-29
CA2566922A1 (en) 2005-12-01
HRP20231588T3 (hr) 2024-03-15
EP3281939A1 (en) 2018-02-14
JP2006001927A (ja) 2006-01-05
NO20065790L (no) 2007-02-07
ES2960824T3 (es) 2024-03-06
CN1956961A (zh) 2007-05-02
JP3754064B2 (ja) 2006-03-08
IL179250A0 (en) 2007-03-08
WO2005113508A1 (en) 2005-12-01
EP3281939B1 (en) 2023-10-18
AR049280A1 (es) 2006-07-12
HUS2400006I1 (hu) 2024-04-28
CY2024008I1 (el) 2024-09-20
MY134672A (en) 2007-12-31
NZ551839A (en) 2009-11-27
KR20080064909A (ko) 2008-07-09
RU2330845C1 (ru) 2008-08-10
CA2566922C (en) 2011-01-11
US20060030710A1 (en) 2006-02-09
BRPI0510114A (pt) 2007-09-25
HK1083341A1 (en) 2006-06-30
NO20200873A1 (no) 2007-02-07
LUC00334I2 (lt) 2024-07-01
NO2024034I1 (no) 2024-07-15
HUE064615T2 (hu) 2024-04-28
US20100204271A1 (en) 2010-08-12
EP1636190A1 (en) 2006-03-22
MXPA06013405A (es) 2007-03-01
TWI329015B (en) 2010-08-21
FR23C1040I1 (fr) 2023-12-29
PE20120361A1 (es) 2012-05-03
DK1636190T3 (da) 2012-09-24
ZA200610647B (en) 2008-06-25
DK3281939T3 (da) 2024-01-22
US8981103B2 (en) 2015-03-17
AU2005245296A1 (en) 2005-12-01
LTC3281939I2 (lt) 2025-04-25
US20150361044A1 (en) 2015-12-17
BE2024C511I2 (lt) 2024-10-08
FIC20240008I1 (fi) 2024-03-20
NO20240384A1 (no) 2007-02-07
AU2005245296B2 (en) 2010-08-12
US20250091995A1 (en) 2025-03-20
PT1636190E (pt) 2012-08-20
EP2514746A1 (en) 2012-10-24
TW200600097A (en) 2006-01-01
CN1956961B (zh) 2010-05-26
NO20161297A1 (no) 2007-02-07
PE20060358A1 (es) 2006-05-12
NO347902B1 (no) 2024-05-06
SI3281939T1 (sl) 2024-02-29
FI3281939T3 (fi) 2023-10-23
US20220235009A1 (en) 2022-07-28
BRPI0510114B1 (pt) 2020-09-15
CY1126560T1 (el) 2024-09-20

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