HRP20190919T1 - Derivati n1-acil- 5-fluoropirimidinona - Google Patents

Derivati n1-acil- 5-fluoropirimidinona Download PDF

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Publication number
HRP20190919T1
HRP20190919T1 HRP20190919TT HRP20190919T HRP20190919T1 HR P20190919 T1 HRP20190919 T1 HR P20190919T1 HR P20190919T T HRP20190919T T HR P20190919TT HR P20190919 T HRP20190919 T HR P20190919T HR P20190919 T1 HRP20190919 T1 HR P20190919T1
Authority
HR
Croatia
Prior art keywords
alkyl
benzyl
optionally substituted
phenyl
compound
Prior art date
Application number
HRP20190919TT
Other languages
English (en)
Croatian (hr)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W. Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20190919(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of HRP20190919T1 publication Critical patent/HRP20190919T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HRP20190919TT 2009-08-07 2010-08-05 Derivati n1-acil- 5-fluoropirimidinona HRP20190919T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
EP10807171.3A EP2519512B1 (en) 2009-08-07 2010-08-05 N1-acyl- 5-fluoropyrimidinone derivatives
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
HRP20190919T1 true HRP20190919T1 (hr) 2019-09-20

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20190919TT HRP20190919T1 (hr) 2009-08-07 2010-08-05 Derivati n1-acil- 5-fluoropirimidinona

Country Status (33)

Country Link
US (1) US8470839B2 (2)
EP (1) EP2519512B1 (2)
JP (1) JP5748754B2 (2)
KR (1) KR101792285B1 (2)
CN (1) CN102548981B (2)
AU (1) AU2010279402B2 (2)
BR (1) BR112012002810B1 (2)
CA (1) CA2768510C (2)
CL (1) CL2012000316A1 (2)
CO (1) CO6491117A2 (2)
CR (1) CR20120030A (2)
CY (1) CY1122115T1 (2)
DK (1) DK2519512T3 (2)
EA (1) EA023411B1 (2)
EC (1) ECSP12011653A (2)
ES (1) ES2728966T3 (2)
HN (1) HN2012000269A (2)
HR (1) HRP20190919T1 (2)
HU (1) HUE045290T2 (2)
IL (1) IL217952A (2)
IN (1) IN2012DN00539A (2)
LT (1) LT2519512T (2)
MX (1) MX2012001620A (2)
NI (1) NI201200022A (2)
NZ (1) NZ597570A (2)
PE (1) PE20120688A1 (2)
PL (1) PL2519512T3 (2)
PT (1) PT2519512T (2)
SI (1) SI2519512T1 (2)
TR (1) TR201908180T4 (2)
UA (1) UA106889C2 (2)
WO (1) WO2011017538A1 (2)
ZA (1) ZA201200819B (2)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-Substituted-5-fluoro-3,6-dihydro-6-imino-2 (1H) -pyrimidinone derivatives as fungicidal compositions for use in plant protection
HUE047711T2 (hu) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
UA117123C2 (uk) * 2012-12-28 2018-06-25 Адама Махтешім Лтд. Похідні 1-(заміщений бензоїл)-5-фтор-4-іміно-3-метил-3,4-дигідропіримідин-2(1h)-ону
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EP3097096A4 (en) 2013-12-31 2017-10-11 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法
MX2022011088A (es) 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (2) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
MX9800136A (es) 1995-07-05 1998-03-29 Du Pont Pirimidinonas fungicidas.
IL125589A0 (en) 1996-03-11 1999-03-12 Novartis Ag Pyrimidin-4-one derivatives as pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
US20080004253A1 (en) 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
AR070228A1 (es) 2008-01-22 2010-03-25 Dow Agrosciences Llc Derivados de 5-fluoro pirimidina
WO2010047866A2 (en) 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
ME02254B (me) 2009-01-23 2015-12-31 Euro Celtique Sa Derivati hidroksamske kiseline
AU2010279411B2 (en) 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
CY1122115T1 (el) 2020-11-25
CA2768510C (en) 2018-05-15
CO6491117A2 (es) 2012-07-31
LT2519512T (lt) 2019-07-25
CN102548981A (zh) 2012-07-04
CL2012000316A1 (es) 2014-06-27
UA106889C2 (uk) 2014-10-27
ZA201200819B (en) 2013-05-29
IL217952A (en) 2017-11-30
NI201200022A (es) 2012-05-22
CR20120030A (es) 2012-03-28
JP2013501723A (ja) 2013-01-17
AU2010279402B2 (en) 2015-04-16
TR201908180T4 (tr) 2019-06-21
EA023411B1 (ru) 2016-06-30
EP2519512A1 (en) 2012-11-07
AU2010279402A1 (en) 2012-02-02
BR112012002810A2 (pt) 2015-09-15
HN2012000269A (es) 2015-04-27
EA201270253A1 (ru) 2012-07-30
CN102548981B (zh) 2015-05-13
JP5748754B2 (ja) 2015-07-15
SI2519512T1 (sl) 2019-09-30
MX2012001620A (es) 2012-04-11
PL2519512T3 (pl) 2019-09-30
US20110034490A1 (en) 2011-02-10
WO2011017538A1 (en) 2011-02-10
DK2519512T3 (da) 2019-05-27
NZ597570A (en) 2014-04-30
KR20120041786A (ko) 2012-05-02
ES2728966T3 (es) 2019-10-29
IL217952A0 (en) 2012-03-29
HK1172894A1 (en) 2013-05-03
EP2519512A4 (en) 2013-01-16
IN2012DN00539A (2) 2015-06-12
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
US8470839B2 (en) 2013-06-25
EP2519512B1 (en) 2019-03-20
PE20120688A1 (es) 2012-06-06
BR112012002810B1 (pt) 2018-12-11
CA2768510A1 (en) 2011-02-10
KR101792285B1 (ko) 2017-10-31
PT2519512T (pt) 2019-06-04

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