HU202222B - Process for producing thiophene derivatives and pharmaceutical compositions comprising same as active ingredient - Google Patents

Process for producing thiophene derivatives and pharmaceutical compositions comprising same as active ingredient Download PDF

Info

Publication number
HU202222B
HU202222B HU883616A HU361688A HU202222B HU 202222 B HU202222 B HU 202222B HU 883616 A HU883616 A HU 883616A HU 361688 A HU361688 A HU 361688A HU 202222 B HU202222 B HU 202222B
Authority
HU
Hungary
Prior art keywords
formula
thienyl
phenyl
ethyl
preparation
Prior art date
Application number
HU883616A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT50466A (en
Inventor
Kimiaki Hayashi
Yasuhiko Ozaki
Kenji Yamada
Hideyuki Takenaga
Ichizo Inoue
Original Assignee
Tanabe Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co filed Critical Tanabe Seiyaku Co
Publication of HUT50466A publication Critical patent/HUT50466A/hu
Publication of HU202222B publication Critical patent/HU202222B/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Dowels (AREA)
  • Joining Of Building Structures In Genera (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
HU883616A 1987-07-09 1988-07-08 Process for producing thiophene derivatives and pharmaceutical compositions comprising same as active ingredient HU202222B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP62171669A JPS6416778A (en) 1987-07-09 1987-07-09 Thiophene derivative

Publications (2)

Publication Number Publication Date
HUT50466A HUT50466A (en) 1990-02-28
HU202222B true HU202222B (en) 1991-02-28

Family

ID=15927497

Family Applications (1)

Application Number Title Priority Date Filing Date
HU883616A HU202222B (en) 1987-07-09 1988-07-08 Process for producing thiophene derivatives and pharmaceutical compositions comprising same as active ingredient

Country Status (15)

Country Link
US (1) US4946862A (de)
EP (1) EP0298703B1 (de)
JP (1) JPS6416778A (de)
KR (1) KR890002088A (de)
CN (1) CN1039245A (de)
AT (1) ATE61362T1 (de)
AU (1) AU600149B2 (de)
DE (1) DE3861928D1 (de)
DK (1) DK382288A (de)
ES (1) ES2036682T3 (de)
FI (1) FI882874L (de)
FR (1) FR2617842B1 (de)
GR (1) GR3001622T3 (de)
HU (1) HU202222B (de)
IL (1) IL86741A0 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5017723A (en) * 1990-02-26 1991-05-21 Jouveinal S.A. Substituted ethylamines, their preparation process, their use as medicine and their synthesising agents
FR2658822A1 (fr) * 1990-02-28 1991-08-30 Jouveinal Sa N-cycloalkylalkylamines, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese.
CA2037123A1 (en) * 1990-02-26 1991-08-27 Jouveinal S.A. Substituted ethylamines, their process of preparation, their use as medication and their synthetic intermediates
EP0445013B1 (de) * 1990-02-26 1994-06-08 Jouveinal S.A. N-cycloalkyl-Alkylamine, Verfahren zu ihrer Herstellung, ihre Verwendung als Arzneimittel und Zwischenprodukte zu ihrer Synthese
FR2658817B1 (fr) * 1990-02-28 1993-02-05 Jouveinal Sa Ethylamines substituees, leur procede de preparation, leur utilisation comme medicament et leurs intermediaires de synthese.
IE913279A1 (en) * 1990-09-26 1992-04-08 Astra Ab (2-Thienyl)alkylamine Derivatives Having Neuroprotective¹Properties
US5362886A (en) * 1993-10-12 1994-11-08 Eli Lilly And Company Asymmetric synthesis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3109845A (en) * 1960-02-04 1963-11-05 Thomae Gmbh Dr K 1-cyclohexyl, 1-cyclohexenyl, 1-furyl, and 1-thienyl, tertiary amino substituted methanes
FR1344455A (fr) * 1962-10-17 1963-11-29 Jouveinal Lab Amino-alcools, leurs esters et leur procédé de préparation
US4128561A (en) * 1975-12-12 1978-12-05 Parcor Process for the preparation of 2-(2-thienyl)-ethylamine and derivatives thereof
JPS5516416A (en) * 1978-07-21 1980-02-05 Hitachi Ltd Board drowing-out bar
JPS58105946A (ja) * 1981-12-18 1983-06-24 Tanabe Seiyaku Co Ltd アミノブタノ−ルエステル誘導体の製法

Also Published As

Publication number Publication date
EP0298703B1 (de) 1991-03-06
IL86741A0 (en) 1988-11-30
DK382288A (da) 1989-01-10
GR3001622T3 (en) 1992-11-23
HUT50466A (en) 1990-02-28
DK382288D0 (da) 1988-07-08
ATE61362T1 (de) 1991-03-15
US4946862A (en) 1990-08-07
AU600149B2 (en) 1990-08-02
JPS6416778A (en) 1989-01-20
FI882874A7 (fi) 1989-01-10
ES2036682T3 (es) 1993-06-01
KR890002088A (ko) 1989-04-08
FR2617842B1 (fr) 1991-05-31
AU1880788A (en) 1989-01-12
FI882874A0 (fi) 1988-06-16
EP0298703A1 (de) 1989-01-11
FI882874L (fi) 1989-01-10
FR2617842A1 (fr) 1989-01-13
DE3861928D1 (de) 1991-04-11
CN1039245A (zh) 1990-01-31

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