HU221804B1 - Napi egyszeri adagolásra alkalmas, minociklin hatóanyagot tartalmazó gyógyszerkészítmény és eljárás előállítására - Google Patents

Napi egyszeri adagolásra alkalmas, minociklin hatóanyagot tartalmazó gyógyszerkészítmény és eljárás előállítására Download PDF

Info

Publication number: HU221804B1
Authority: HU; Hungary
Prior art keywords: minocycline; deoxy; dimethylamino; release; coating
Prior art date: 1989-09-21

Application number

HU9006006A

Other languages

English (en)

Hungarian (hu)

Other versions

HU906006D0 (en

HUT59314A (en

Inventor

Keith Anthony Ellway

Madurai Gurusamy Ganesann

Jerry Bain Johnson

Kieran George Mooney

Nitin Vadilal Sheth

Joseph James Valorose

Original Assignee

American Cyanamid Co.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-09-21

Filing date

1990-09-21

Publication date

2003-01-28

1990-09-21 Application filed by American Cyanamid Co. filed Critical American Cyanamid Co.

1991-03-28 Publication of HU906006D0 publication Critical patent/HU906006D0/hu

1992-05-28 Publication of HUT59314A publication Critical patent/HUT59314A/hu

2003-01-28 Publication of HU221804B1 publication Critical patent/HU221804B1/hu

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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
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- A61K9/5015—Organic compounds, e.g. fats, sugars
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/65—Tetracyclines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
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- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/5005—Wall or coating material
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
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- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

HU9006006A 1989-09-21 1990-09-21 Napi egyszeri adagolásra alkalmas, minociklin hatóanyagot tartalmazó gyógyszerkészítmény és eljárás előállítására HU221804B1 (hu)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US41070889A	1989-09-21	1989-09-21

Publications (3)

Publication Number	Publication Date
HU906006D0 HU906006D0 (en)	1991-03-28
HUT59314A HUT59314A (en)	1992-05-28
HU221804B1 true HU221804B1 (hu)	2003-01-28

Family

ID=23625892

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU9006006A HU221804B1 (hu)	1989-09-21	1990-09-21	Napi egyszeri adagolásra alkalmas, minociklin hatóanyagot tartalmazó gyógyszerkészítmény és eljárás előállítására

Country Status (25)

Country	Link
US (2)	US5300304A (da)
EP (1)	EP0418565B1 (da)
JP (1)	JP3140764B2 (da)
KR (1)	KR100187950B1 (da)
CN (1)	CN1035039C (da)
AR (1)	AR244547A1 (da)
AT (1)	ATE114472T1 (da)
AU (1)	AU624998B2 (da)
CA (1)	CA2025703C (da)
CZ (1)	CZ283048B6 (da)
DD (1)	DD297558A5 (da)
DE (1)	DE69014513T2 (da)
DK (1)	DK0418565T3 (da)
ES (1)	ES2064564T3 (da)
FI (1)	FI96170C (da)
HU (1)	HU221804B1 (da)
IE (1)	IE66389B1 (da)
IL (1)	IL95423A (da)
NO (1)	NO177038C (da)
NZ (1)	NZ235319A (da)
PH (1)	PH30777A (da)
PL (1)	PL164770B1 (da)
PT (1)	PT95353B (da)
SK (1)	SK455990A3 (da)
ZA (1)	ZA907546B (da)

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US4173626A (en) *	1978-12-11	1979-11-06	Merck & Co., Inc.	Sustained release indomethacin
FR2447192A1 (fr) *	1979-01-25	1980-08-22	Adria Lab Inc	Forme galenique a liberation prolongee d'indoprofene
US4353887A (en) *	1979-08-16	1982-10-12	Ciba-Geigy Corporation	Divisible tablet having controlled and delayed release of the active substance
DK150008C (da) *	1981-11-20	1987-05-25	Benzon As Alfred	Fremgangsmaade til fremstilling af et farmaceutisk oralt polydepotpraeparat
JPS61210025A (ja) *	1985-03-14	1986-09-18	Teisan Seiyaku Kk	安定化された抗生物質複合顆粒製剤
GB8521494D0 (en) *	1985-08-29	1985-10-02	Zyma Sa	Controlled release tablet
US4837030A (en) *	1987-10-06	1989-06-06	American Cyanamid Company	Novel controlled release formulations of tetracycline compounds
EP0327295A3 (en) *	1988-02-01	1989-09-06	F.H. FAULDING & CO. LTD.	Tetracycline dosage form
US5133974A (en) *	1989-05-05	1992-07-28	Kv Pharmaceutical Company	Extended release pharmaceutical formulations
ATE114472T1 (de) *	1989-09-21	1994-12-15	American Cyanamid Co	System des typs ''einmal täglich'' zur gepulsten minocyclinabgabe.

1990
- 1990-08-20 AT AT90115881T patent/ATE114472T1/de not_active IP Right Cessation
- 1990-08-20 ES ES90115881T patent/ES2064564T3/es not_active Expired - Lifetime
- 1990-08-20 EP EP90115881A patent/EP0418565B1/en not_active Expired - Lifetime
- 1990-08-20 DE DE69014513T patent/DE69014513T2/de not_active Expired - Lifetime
- 1990-08-20 IL IL9542390A patent/IL95423A/en unknown
- 1990-08-20 DK DK90115881.6T patent/DK0418565T3/da active
- 1990-09-14 NZ NZ235319A patent/NZ235319A/xx unknown
- 1990-09-15 CN CN90107817A patent/CN1035039C/zh not_active Expired - Lifetime
- 1990-09-18 JP JP02246377A patent/JP3140764B2/ja not_active Expired - Lifetime
- 1990-09-19 SK SK4559-90A patent/SK455990A3/sk not_active IP Right Cessation
- 1990-09-19 PT PT95353A patent/PT95353B/pt not_active IP Right Cessation
- 1990-09-19 CA CA002025703A patent/CA2025703C/en not_active Expired - Lifetime
- 1990-09-19 PH PH41222A patent/PH30777A/en unknown
- 1990-09-19 CZ CS904559A patent/CZ283048B6/cs not_active IP Right Cessation
- 1990-09-20 AR AR90317918A patent/AR244547A1/es active
- 1990-09-20 FI FI904634A patent/FI96170C/fi active IP Right Grant
- 1990-09-20 AU AU63031/90A patent/AU624998B2/en not_active Expired
- 1990-09-20 NO NO904099A patent/NO177038C/no not_active IP Right Cessation
- 1990-09-20 PL PL90286971A patent/PL164770B1/pl unknown
- 1990-09-20 IE IE339890A patent/IE66389B1/en not_active IP Right Cessation
- 1990-09-20 ZA ZA907546A patent/ZA907546B/xx unknown
- 1990-09-20 KR KR1019900014932A patent/KR100187950B1/ko not_active Expired - Lifetime
- 1990-09-21 HU HU9006006A patent/HU221804B1/hu not_active IP Right Cessation
- 1990-09-21 DD DD90344125A patent/DD297558A5/de unknown
1992
- 1992-05-27 US US07/892,383 patent/US5300304A/en not_active Expired - Lifetime
1993
- 1993-07-14 US US08/091,322 patent/US5413777A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
KR910005875A (ko)	1991-04-27
IL95423A (en)	1994-11-11
ATE114472T1 (de)	1994-12-15
ES2064564T3 (es)	1995-02-01
KR100187950B1 (ko)	1999-06-01
US5413777A (en)	1995-05-09
CA2025703A1 (en)	1991-03-22
HK1000315A1 (en)	1998-02-27
FI96170B (fi)	1996-02-15
JPH03112930A (ja)	1991-05-14
NO177038C (no)	1995-07-12
AR244547A1 (es)	1993-11-30
AU624998B2 (en)	1992-06-25
CN1035039C (zh)	1997-06-04
NO904099L (no)	1991-03-22
NO177038B (no)	1995-04-03
EP0418565A2 (en)	1991-03-27
PT95353A (pt)	1991-08-14
NZ235319A (en)	1993-03-26
FI96170C (fi)	1996-05-27
HU906006D0 (en)	1991-03-28
CZ455990A3 (en)	1997-08-13
IE66389B1 (en)	1995-12-27
FI904634A0 (fi)	1990-09-20
DE69014513T2 (de)	1995-05-24
PT95353B (pt)	1998-05-29
DD297558A5 (de)	1992-01-16
PL286971A1 (en)	1992-01-27
EP0418565A3 (en)	1991-09-25
NO904099D0 (no)	1990-09-20
DE69014513D1 (de)	1995-01-12
PL164770B1 (pl)	1994-10-31
CA2025703C (en)	2002-08-27
CZ283048B6 (cs)	1997-12-17
IE903398A1 (en)	1991-04-10
AU6303190A (en)	1991-03-28
SK279358B6 (sk)	1998-10-07
DK0418565T3 (da)	1995-01-23
SK455990A3 (en)	1998-10-07
ZA907546B (en)	1991-07-31
CN1050320A (zh)	1991-04-03
US5300304A (en)	1994-04-05
JP3140764B2 (ja)	2001-03-05
IL95423A0 (en)	1991-06-30
HUT59314A (en)	1992-05-28
PH30777A (en)	1997-10-17
EP0418565B1 (en)	1994-11-30

Legal Events

Date	Code	Title	Description
2003-01-28	HFG4	Patent granted, date of granting	Effective date: 20021107
2010-06-28	MM4A	Lapse of definitive patent protection due to non-payment of fees

Publication	Publication Date	Title
HU221804B1 (hu)	2003-01-28	Napi egyszeri adagolásra alkalmas, minociklin hatóanyagot tartalmazó gyógyszerkészítmény és eljárás előállítására
US5262173A (en)	1993-11-16	Pulsatile once-a-day delivery systems for minocycline
HU202110B (en)	1991-02-28	Process for producing pharmaceutical compositions of controlled releasing, containing tetracyclin compounds
HU196037B (en)	1988-09-28	Process for producing pharmaceutics releasing active ingredient in three separate phases
KR20080059409A (ko)	2008-06-27	즉시방출형 및/또는 조절방출형 특성을 가진 약제학적 제형
ES2860694T3 (es)	2021-10-05	Composición farmacéutica de liberación sostenida que contiene rivastigmina
FI96481C (fi)	1996-07-10	Menetelmä pulssittaisten kerran päivässä annettavien minosykliinin vapautussysteemien valmistamiseksi
NO177553B (no)	1995-07-03	Fremgangsmåte for fremstilling av et farmasöytisk doseringssystem
NO177554B (no)	1995-07-03	Fremgangsmåte for fremstilling av en multiovertrukket sammensetning som utgjör et farmasöytisk doseringssystem
HK1009930B (en)	2000-04-20	Improved pulsatile once-a-day delivery systems for minocycline