ID21654A - Proses derivatisasi selektif taksana - Google Patents

Proses derivatisasi selektif taksana

Info

Publication number: ID21654A
Authority: ID; Indonesia
Prior art keywords: sup; prosecutive; hydroxytaxane; acyloxy; selective derivatization
Prior art date: 1997-08-18

Application number

IDW990217A

Other languages

English (en)

Inventor

Robert A Holton

Zhuming Zhang

Paul A Clark

Original Assignee

Univ Florida State

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-08-18

Filing date

1998-08-17

Publication date

1999-07-08

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27368950&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID21654(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1998-08-17 Application filed by Univ Florida State filed Critical Univ Florida State

1999-07-08 Publication of ID21654A publication Critical patent/ID21654A/id

Links

238000000034 method Methods 0.000 title abstract 3
238000001212 derivatisation Methods 0.000 title 1
229940123237 Taxane Drugs 0.000 abstract 2
125000001183 hydrocarbyl group Chemical group 0.000 abstract 2
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
DHKHKXVYLBGOIT-UHFFFAOYSA-N acetaldehyde Diethyl Acetal Natural products CCOC(C)OCC DHKHKXVYLBGOIT-UHFFFAOYSA-N 0.000 abstract 1
125000002777 acetyl group Chemical class [H]C([H])([H])C(*)=O 0.000 abstract 1
239000003377 acid catalyst Substances 0.000 abstract 1
239000003795 chemical substances by application Substances 0.000 abstract 1
125000001072 heteroaryl group Chemical group 0.000 abstract 1
DKPFODGZWDEEBT-QFIAKTPHSA-N taxane Chemical class C([C@]1(C)CCC[C@@H](C)[C@H]1C1)C[C@H]2[C@H](C)CC[C@@H]1C2(C)C DKPFODGZWDEEBT-QFIAKTPHSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C07F7/1872—Preparation; Treatments not provided for in C07F7/20
- C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Epoxy Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Fats And Perfumes (AREA)
Percussion Or Vibration Massage (AREA)
Soil Working Implements (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Saccharide Compounds (AREA)

IDW990217A 1997-08-18 1998-08-17 Proses derivatisasi selektif taksana ID21654A (id)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US5600097P	1997-08-18	1997-08-18
US8126598P	1998-04-09	1998-04-09
US09/063,477 US7288665B1 (en)	1997-08-18	1998-04-20	Process for selective derivatization of taxanes

Publications (1)

Publication Number	Publication Date
ID21654A true ID21654A (id)	1999-07-08

Family

ID=27368950

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IDW990217A ID21654A (id)	1997-08-18	1998-08-17	Proses derivatisasi selektif taksana

Country Status (25)

Country	Link
US (5)	US7288665B1 (id)
EP (6)	EP1170293B1 (id)
JP (1)	JP2001504864A (id)
KR (1)	KR100596989B1 (id)
CN (3)	CN100351246C (id)
AT (3)	ATE341540T1 (id)
AU (1)	AU744987B2 (id)
BR (1)	BR9806145A (id)
CA (2)	CA2597799A1 (id)
CY (1)	CY1105399T1 (id)
CZ (1)	CZ296580B6 (id)
DE (3)	DE69837684T2 (id)
DK (3)	DK1170292T3 (id)
ES (3)	ES2259646T3 (id)
HU (1)	HUP0300425A3 (id)
ID (1)	ID21654A (id)
IL (3)	IL129386A0 (id)
NO (4)	NO325139B1 (id)
NZ (1)	NZ335156A (id)
PL (3)	PL201641B1 (id)
PT (3)	PT956284E (id)
RU (1)	RU2225402C2 (id)
SG (1)	SG97986A1 (id)
WO (1)	WO1999009021A1 (id)
ZA (1)	ZA987394B (id)

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1998
- 1998-04-20 US US09/063,477 patent/US7288665B1/en not_active Expired - Fee Related
- 1998-08-17 NZ NZ335156A patent/NZ335156A/en not_active IP Right Cessation
- 1998-08-17 CA CA002597799A patent/CA2597799A1/en not_active Abandoned
- 1998-08-17 ES ES01203288T patent/ES2259646T3/es not_active Expired - Lifetime
- 1998-08-17 WO PCT/US1998/017016 patent/WO1999009021A1/en not_active Ceased
- 1998-08-17 JP JP51349899A patent/JP2001504864A/ja not_active Ceased
- 1998-08-17 RU RU99110384/04A patent/RU2225402C2/ru not_active IP Right Cessation
- 1998-08-17 PL PL377991A patent/PL201641B1/pl not_active IP Right Cessation
- 1998-08-17 PT PT98942080T patent/PT956284E/pt unknown
- 1998-08-17 EP EP01203288A patent/EP1170293B1/en not_active Expired - Lifetime
- 1998-08-17 EP EP01203287A patent/EP1170292B1/en not_active Expired - Lifetime
- 1998-08-17 DK DK01203287T patent/DK1170292T3/da active
- 1998-08-17 DE DE69837684T patent/DE69837684T2/de not_active Expired - Lifetime
- 1998-08-17 HU HU0300425A patent/HUP0300425A3/hu unknown
- 1998-08-17 DE DE69834584T patent/DE69834584T2/de not_active Expired - Fee Related
- 1998-08-17 PT PT01203287T patent/PT1170292E/pt unknown
- 1998-08-17 CN CNB2005100641228A patent/CN100351246C/zh not_active Expired - Fee Related
- 1998-08-17 ES ES98942080T patent/ES2274579T3/es not_active Expired - Lifetime
- 1998-08-17 PT PT01203288T patent/PT1170293E/pt unknown
- 1998-08-17 CN CNA2006101492418A patent/CN1974563A/zh active Pending
- 1998-08-17 IL IL12938698A patent/IL129386A0/xx not_active IP Right Cessation
- 1998-08-17 BR BR9806145-3A patent/BR9806145A/pt not_active Application Discontinuation
- 1998-08-17 ID IDW990217A patent/ID21654A/id unknown
- 1998-08-17 AT AT98942080T patent/ATE341540T1/de not_active IP Right Cessation
- 1998-08-17 AT AT01203287T patent/ATE360624T1/de not_active IP Right Cessation
- 1998-08-17 EP EP05108674A patent/EP1671960A2/en not_active Withdrawn
- 1998-08-17 DK DK01203288T patent/DK1170293T3/da active
- 1998-08-17 PL PL98377990A patent/PL193674B1/pl not_active IP Right Cessation
- 1998-08-17 PL PL98332723A patent/PL332723A1/xx not_active IP Right Cessation
- 1998-08-17 KR KR1019997003388A patent/KR100596989B1/ko not_active Expired - Fee Related
- 1998-08-17 CA CA002268662A patent/CA2268662A1/en not_active Abandoned
- 1998-08-17 CZ CZ0133299A patent/CZ296580B6/cs not_active IP Right Cessation
- 1998-08-17 ES ES01203287T patent/ES2286073T3/es not_active Expired - Lifetime
- 1998-08-17 AT AT01203288T patent/ATE326455T1/de not_active IP Right Cessation
- 1998-08-17 DE DE69836072T patent/DE69836072T2/de not_active Expired - Lifetime
- 1998-08-17 EP EP01203286A patent/EP1193262A1/en not_active Withdrawn
- 1998-08-17 ZA ZA987394A patent/ZA987394B/xx unknown
- 1998-08-17 EP EP07104179A patent/EP1795528A1/en not_active Withdrawn
- 1998-08-17 CN CNB98801341XA patent/CN1205196C/zh not_active Expired - Fee Related
- 1998-08-17 DK DK98942080T patent/DK0956284T3/da active
- 1998-08-17 EP EP98942080A patent/EP0956284B1/en not_active Expired - Lifetime
- 1998-08-17 AU AU90211/98A patent/AU744987B2/en not_active Ceased
- 1998-08-17 SG SG200006873A patent/SG97986A1/en unknown
1999
- 1999-04-16 NO NO19991838A patent/NO325139B1/no not_active IP Right Cessation
- 1999-06-17 US US09/335,408 patent/US6191287B1/en not_active Expired - Lifetime
2000
- 2000-06-07 US US09/588,933 patent/US6291691B1/en not_active Expired - Fee Related
- 2000-09-28 US US09/672,270 patent/US6706896B1/en not_active Expired - Fee Related
2005
- 2005-06-09 US US11/148,833 patent/US20050272944A1/en not_active Abandoned
- 2005-09-29 NO NO20054512A patent/NO20054512L/no unknown
- 2005-09-29 NO NO20054513A patent/NO20054513L/no unknown
- 2005-09-29 NO NO20054514A patent/NO20054514L/no unknown
2006
- 2006-06-26 CY CY20061100861T patent/CY1105399T1/el unknown
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Also Published As

Publication number	Publication date
EP1671960A2 (en)	2006-06-21
DE69836072T2 (de)	2007-01-11
CZ133299A3 (cs)	1999-11-17
EP1170293A2 (en)	2002-01-09
PT956284E (pt)	2006-12-29
CY1105399T1 (el)	2010-04-28
KR20000068782A (ko)	2000-11-25
KR100596989B1 (ko)	2006-07-07
CN1974563A (zh)	2007-06-06
US7288665B1 (en)	2007-10-30
PL201641B1 (pl)	2009-04-30
ES2286073T3 (es)	2007-12-01
RU2225402C2 (ru)	2004-03-10
NZ335156A (en)	2001-10-26
EP0956284A1 (en)	1999-11-17
EP1170292B1 (en)	2007-04-25
ES2274579T3 (es)	2007-05-16
US20050272944A1 (en)	2005-12-08
PT1170293E (pt)	2006-07-31
HUP0300425A2 (hu)	2003-09-29
CN1690053A (zh)	2005-11-02
DE69837684T2 (de)	2007-09-06
CZ296580B6 (cs)	2006-04-12
EP0956284B1 (en)	2006-10-04
EP1170292A2 (en)	2002-01-09
NO991838D0 (no)	1999-04-16
EP1170293B1 (en)	2006-05-17
EP1170292A3 (en)	2002-04-03
AU744987B2 (en)	2002-03-07
IL129386A0 (en)	2000-02-17
DE69837684D1 (de)	2007-06-06
US6291691B1 (en)	2001-09-18
HUP0300425A3 (en)	2005-12-28
DK1170292T3 (da)	2007-08-27
BR9806145A (pt)	2000-01-18
AU9021198A (en)	1999-03-08
ATE326455T1 (de)	2006-06-15
SG97986A1 (en)	2003-08-20
PL193674B1 (pl)	2007-03-30
NO20054512L (no)	1999-06-18
US6191287B1 (en)	2001-02-20
US6706896B1 (en)	2004-03-16
ZA987394B (en)	1999-05-14
CN100351246C (zh)	2007-11-28
DE69836072D1 (de)	2006-11-16
EP1193262A1 (en)	2002-04-03
ATE360624T1 (de)	2007-05-15
NO325139B1 (no)	2008-02-11
DE69834584T2 (de)	2006-11-23
CN1205196C (zh)	2005-06-08
ATE341540T1 (de)	2006-10-15
ES2259646T3 (es)	2006-10-16
IL184320A0 (en)	2007-10-31
WO1999009021A1 (en)	1999-02-25
EP0956284A4 (en)	2001-12-05
CA2597799A1 (en)	1999-02-25
NO991838L (no)	1999-06-18
EP1795528A1 (en)	2007-06-13
CA2268662A1 (en)	1999-02-25
JP2001504864A (ja)	2001-04-10
IL184321A0 (en)	2007-10-31
PL332723A1 (en)	1999-10-11
NO20054514L (no)	1999-06-18
NO20054513L (no)	1999-06-18
CN1239476A (zh)	1999-12-22
DK1170293T3 (da)	2006-09-11
PT1170292E (pt)	2007-05-31
DE69834584D1 (de)	2006-06-22
EP1170293A3 (en)	2002-04-03
DK0956284T3 (da)	2007-02-12

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