IL118768A - Diphenylmethane piperidine derivatives pharmaceutical compositions containing them and a method for their preparation - Google Patents

Diphenylmethane piperidine derivatives pharmaceutical compositions containing them and a method for their preparation

Info

Publication number: IL118768A
Authority: IL; Israel
Prior art keywords: diphenylmethane; preparation; pharmaceutical compositions; compositions containing; piperidine derivatives
Prior art date: 1995-07-12

Application number

IL11876896A

Other languages

English (en)

Other versions

IL118768A0 (en

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-07-12

Filing date

1996-07-01

Publication date

2000-10-31

1996-07-01 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

1996-10-31 Publication of IL118768A0 publication Critical patent/IL118768A0/xx

2000-10-31 Publication of IL118768A publication Critical patent/IL118768A/xx

Links

DMJREIQATMESOR-UHFFFAOYSA-N N1CCCCC1.C1(=CC=CC=C1)CC1=CC=CC=C1 Chemical class N1CCCCC1.C1(=CC=CC=C1)CC1=CC=CC=C1 DMJREIQATMESOR-UHFFFAOYSA-N 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Psychiatry (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)

IL11876896A 1995-07-12 1996-07-01 Diphenylmethane piperidine derivatives pharmaceutical compositions containing them and a method for their preparation IL118768A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP95201910		1995-07-12

Publications (2)

Publication Number	Publication Date
IL118768A0 IL118768A0 (en)	1996-10-31
IL118768A true IL118768A (en)	2000-10-31

Family

ID=8220478

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL11876896A IL118768A (en)	1995-07-12	1996-07-01	Diphenylmethane piperidine derivatives pharmaceutical compositions containing them and a method for their preparation

Country Status (26)

Country	Link
US (1)	US5935974A (cs)
EP (1)	EP0842170B1 (cs)
JP (1)	JPH11508907A (cs)
KR (1)	KR19990028807A (cs)
CN (1)	CN1091108C (cs)
AR (1)	AR003966A1 (cs)
AT (1)	ATE199150T1 (cs)
AU (1)	AU699370B2 (cs)
BR (1)	BR9609330A (cs)
CA (1)	CA2226851A1 (cs)
CZ (1)	CZ288909B6 (cs)
DE (1)	DE69611788T2 (cs)
DK (1)	DK0842170T3 (cs)
ES (1)	ES2156287T3 (cs)
GR (1)	GR3035849T3 (cs)
HU (1)	HUP9802762A3 (cs)
IL (1)	IL118768A (cs)
NO (1)	NO309765B1 (cs)
NZ (1)	NZ315318A (cs)
PL (1)	PL183837B1 (cs)
PT (1)	PT842170E (cs)
RU (1)	RU2162846C2 (cs)
TR (1)	TR199800027T1 (cs)
TW (1)	TW419477B (cs)
WO (1)	WO1997003065A1 (cs)
ZA (1)	ZA965691B (cs)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1999019324A2 (en) *	1997-10-07	1999-04-22	Akzo Nobel N.V.	Antipsychotic substituted piperidine derivatives
AU2279099A (en) *	1998-01-09	1999-07-26	Akzo Nobel N.V.	Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of depression
AU2517499A (en) *	1998-01-09	1999-07-26	Akzo Nobel N.V.	Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of movement disorders
AU5600100A (en)	1999-06-11	2001-01-02	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
WO2000076513A1 (en)	1999-06-11	2000-12-21	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
WO2000076511A1 (en)	1999-06-11	2000-12-21	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
US6358979B1 (en)	1999-06-11	2002-03-19	Merck & Co., Inc.	N-cyclopentyl modulators of chemokine receptor activity
US6500844B1 (en)	1999-06-11	2002-12-31	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
US6472410B1 (en)	1999-06-11	2002-10-29	Merck & Co., Inc.	N-cyclopentyl modulators of chemokine receptor activity
KR20010113007A (ko) *	2000-06-15	2001-12-24	주정호	항암제로서 유용한 ｎ-치환된 피페리디닐우레아 유도체 및그의 제조방법
TW200303304A (en) *	2002-02-18	2003-09-01	Astrazeneca Ab	Chemical compounds
US6770659B2 (en) *	2002-08-26	2004-08-03	Sk Corporation	Benzoyl piperidine compounds
KR20050085673A (ko) *	2002-12-18	2005-08-29	에프엠씨 코포레이션	Ｎ-(치환된 아릴메틸)-4-(이치환된 메틸)피페리딘 및피페라진
SE0400208D0 (sv) *	2004-02-02	2004-02-02	Astrazeneca Ab	Chemical compounds
TW200812582A (en) *	2006-04-06	2008-03-16	Astrazeneca Ab	Medicaments
MX381417B (es)	2014-08-28	2025-03-12	Asceneuron Sa	Inhibidores de glucosidasa.
WO2017106254A1 (en) *	2015-12-18	2017-06-22	Merck Sharp & Dohme Corp.	Glycosidase inhibitors and uses thereof
JP2019506430A (ja)	2016-02-25	2019-03-07	エースニューロン・ソシエテ・アノニム	グリコシダーゼ阻害剤
CN108884077A (zh)	2016-02-25	2018-11-23	阿森纽荣股份公司	糖苷酶抑制剂
US11261183B2 (en)	2016-02-25	2022-03-01	Asceneuron Sa	Sulfoximine glycosidase inhibitors
JP6971999B2 (ja)	2016-02-25	2021-11-24	エースニューロン・ソシエテ・アノニム	ピペラジン誘導体の酸付加塩
US11213525B2 (en)	2017-08-24	2022-01-04	Asceneuron Sa	Linear glycosidase inhibitors
WO2020039029A1 (en)	2018-08-22	2020-02-27	Asceneuron S. A.	Spiro compounds as glycosidase inhibitors
US12016852B2 (en)	2018-08-22	2024-06-25	Asceneuron Sa	Pyrrolidine glycosidase inhibitors
CA3110032A1 (en)	2018-08-22	2020-02-27	Asceneuron S.A.	Succinate and fumarate acid addition salts of piperazine derivatives
US11795165B2 (en)	2018-08-22	2023-10-24	Asceneuron Sa	Tetrahydro-benzoazepine glycosidase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US450780A (en) *		1891-04-21		Steam-engine
US4180583A (en) *	1972-01-28	1979-12-25	Richardson-Merrell Inc.	Olefinic 4-substituted piperidino derivatives as therapeutics
US3922276A (en) *	1974-12-11	1975-11-25	Robins Co Inc A H	1-Substituted-4-benzylidenepiperidines
US4666905A (en) *	1983-06-02	1987-05-19	Warner-Lambert Company	Diphenylmethylene piperidines compositions and methods for their use
US4540780A (en) *	1983-06-02	1985-09-10	Warner-Lambert Company	Diphenylmethylene piperidines
MX173362B (es) *	1987-03-02	1994-02-23	Pfizer	Compuestos de piperazinil heterociclicos y procedimiento para su preparacion

1996
- 1996-07-01 IL IL11876896A patent/IL118768A/xx not_active IP Right Cessation
- 1996-07-04 ZA ZA965691A patent/ZA965691B/xx unknown
- 1996-07-09 KR KR1019980700107A patent/KR19990028807A/ko not_active Ceased
- 1996-07-09 HU HU9802762A patent/HUP9802762A3/hu unknown
- 1996-07-09 AT AT96927006T patent/ATE199150T1/de not_active IP Right Cessation
- 1996-07-09 PT PT96927006T patent/PT842170E/pt unknown
- 1996-07-09 NZ NZ315318A patent/NZ315318A/en unknown
- 1996-07-09 DE DE69611788T patent/DE69611788T2/de not_active Expired - Fee Related
- 1996-07-09 ES ES96927006T patent/ES2156287T3/es not_active Expired - Lifetime
- 1996-07-09 US US08/983,059 patent/US5935974A/en not_active Expired - Fee Related
- 1996-07-09 PL PL96324451A patent/PL183837B1/pl unknown
- 1996-07-09 WO PCT/EP1996/003099 patent/WO1997003065A1/en not_active Ceased
- 1996-07-09 AU AU66993/96A patent/AU699370B2/en not_active Ceased
- 1996-07-09 RU RU98102392/04A patent/RU2162846C2/ru not_active IP Right Cessation
- 1996-07-09 CZ CZ199883A patent/CZ288909B6/cs not_active IP Right Cessation
- 1996-07-09 BR BR9609330A patent/BR9609330A/pt active Search and Examination
- 1996-07-09 CA CA002226851A patent/CA2226851A1/en not_active Abandoned
- 1996-07-09 EP EP96927006A patent/EP0842170B1/en not_active Expired - Lifetime
- 1996-07-09 TR TR1998/00027T patent/TR199800027T1/xx unknown
- 1996-07-09 DK DK96927006T patent/DK0842170T3/da active
- 1996-07-09 CN CN96195461A patent/CN1091108C/zh not_active Expired - Fee Related
- 1996-07-09 JP JP9505516A patent/JPH11508907A/ja active Pending
- 1996-07-12 AR ARP960103567A patent/AR003966A1/es active IP Right Grant
- 1996-07-29 TW TW085109218A patent/TW419477B/zh not_active IP Right Cessation
1998
- 1998-01-09 NO NO980109A patent/NO309765B1/no unknown
2001
- 2001-05-11 GR GR20010400699T patent/GR3035849T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
CN1190965A (zh)	1998-08-19
HK1010818A1 (en)	1999-07-02
ES2156287T3 (es)	2001-06-16
IL118768A0 (en)	1996-10-31
MX9800368A (es)	1998-03-31
EP0842170A1 (en)	1998-05-20
NO980109L (no)	1998-01-09
CN1091108C (zh)	2002-09-18
US5935974A (en)	1999-08-10
ATE199150T1 (de)	2001-02-15
DE69611788D1 (de)	2001-03-22
WO1997003065A1 (en)	1997-01-30
PL183837B1 (pl)	2002-07-31
CA2226851A1 (en)	1997-01-30
AU699370B2 (en)	1998-12-03
NO309765B1 (no)	2001-03-26
KR19990028807A (ko)	1999-04-15
DE69611788T2 (de)	2001-08-02
NZ315318A (en)	1999-10-28
EP0842170B1 (en)	2001-02-14
PL324451A1 (en)	1998-05-25
AU6699396A (en)	1997-02-10
HUP9802762A2 (hu)	1999-10-28
HUP9802762A3 (en)	2002-10-28
CZ8398A3 (cs)	1998-06-17
ZA965691B (en)	1997-01-24
RU2162846C2 (ru)	2001-02-10
PT842170E (pt)	2001-06-29
BR9609330A (pt)	1999-05-25
GR3035849T3 (en)	2001-08-31
CZ288909B6 (cs)	2001-09-12
DK0842170T3 (da)	2001-06-18
TR199800027T1 (xx)	1998-05-21
TW419477B (en)	2001-01-21
JPH11508907A (ja)	1999-08-03
AR003966A1 (es)	1998-09-30
NO980109D0 (no)	1998-01-09

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Legal Events

Date	Code	Title
2001-03-19	FF	Patent granted
2001-06-14	KB	Patent renewed
2002-08-14	KB	Patent renewed
2007-05-21	MM9K	Patent not in force due to non-payment of renewal fees