NO980109L - Difenylmetylen-piperidin-derivater - Google Patents

Difenylmetylen-piperidin-derivater

Info

Publication number: NO980109L
Authority: NO; Norway
Prior art keywords: piperidine derivatives; diphenylmethylene piperidine; diphenylmethylene; derivatives; piperidine
Prior art date: 1995-07-12

Application number

NO980109A

Other languages

English (en)

Other versions

NO309765B1 (no

NO980109D0 (no

Inventor

Duncan Robertson Rae

David Robert Jaap

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-07-12

Filing date

1998-01-09

Publication date

1998-01-09

1998-01-09 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

1998-01-09 Publication of NO980109L publication Critical patent/NO980109L/no

1998-01-09 Publication of NO980109D0 publication Critical patent/NO980109D0/no

2001-03-26 Publication of NO309765B1 publication Critical patent/NO309765B1/no

Links

ZFDDWBKSMIWSBN-UHFFFAOYSA-N 2-benzhydrylidenepiperidine Chemical class N1CCCCC1=C(C=1C=CC=CC=1)C1=CC=CC=C1 ZFDDWBKSMIWSBN-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)

NO980109A 1995-07-12 1998-01-09 Difenylmetylen-piperidin-derivater, anvendelse av og farmasöytiske blandinger inneholdende dem og fremgangsmåte for fremstilling derav NO309765B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP95201910		1995-07-12
PCT/EP1996/003099 WO1997003065A1 (en)	1995-07-12	1996-07-09	Diphenylmethylene piperidine derivatives

Publications (3)

Publication Number	Publication Date
NO980109L true NO980109L (no)	1998-01-09
NO980109D0 NO980109D0 (no)	1998-01-09
NO309765B1 NO309765B1 (no)	2001-03-26

Family

ID=8220478

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO980109A NO309765B1 (no)	1995-07-12	1998-01-09	Difenylmetylen-piperidin-derivater, anvendelse av og farmasöytiske blandinger inneholdende dem og fremgangsmåte for fremstilling derav

Country Status (26)

Country	Link
US (1)	US5935974A (no)
EP (1)	EP0842170B1 (no)
JP (1)	JPH11508907A (no)
KR (1)	KR19990028807A (no)
CN (1)	CN1091108C (no)
AR (1)	AR003966A1 (no)
AT (1)	ATE199150T1 (no)
AU (1)	AU699370B2 (no)
BR (1)	BR9609330A (no)
CA (1)	CA2226851A1 (no)
CZ (1)	CZ288909B6 (no)
DE (1)	DE69611788T2 (no)
DK (1)	DK0842170T3 (no)
ES (1)	ES2156287T3 (no)
GR (1)	GR3035849T3 (no)
HU (1)	HUP9802762A3 (no)
IL (1)	IL118768A (no)
NO (1)	NO309765B1 (no)
NZ (1)	NZ315318A (no)
PL (1)	PL183837B1 (no)
PT (1)	PT842170E (no)
RU (1)	RU2162846C2 (no)
TR (1)	TR199800027T1 (no)
TW (1)	TW419477B (no)
WO (1)	WO1997003065A1 (no)
ZA (1)	ZA965691B (no)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1021440A2 (en) *	1997-10-07	2000-07-26	Akzo Nobel N.V.	Antipsychotic substituted piperidine derivatives
AU2517499A (en) *	1998-01-09	1999-07-26	Akzo Nobel N.V.	Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of movement disorders
WO1999034801A1 (en) *	1998-01-09	1999-07-15	Akzo Nobel N.V.	Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of depression
WO2000076513A1 (en)	1999-06-11	2000-12-21	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
US6472410B1 (en)	1999-06-11	2002-10-29	Merck & Co., Inc.	N-cyclopentyl modulators of chemokine receptor activity
AU5600100A (en)	1999-06-11	2001-01-02	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
US6500844B1 (en)	1999-06-11	2002-12-31	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
AU5469400A (en)	1999-06-11	2001-01-02	Merck & Co., Inc.	Cyclopentyl modulators of chemokine receptor activity
US6358979B1 (en)	1999-06-11	2002-03-19	Merck & Co., Inc.	N-cyclopentyl modulators of chemokine receptor activity
KR20010113007A (ko) *	2000-06-15	2001-12-24	주정호	항암제로서 유용한 ｎ-치환된 피페리디닐우레아 유도체 및그의 제조방법
TW200303304A (en) *	2002-02-18	2003-09-01	Astrazeneca Ab	Chemical compounds
US6770659B2 (en) *	2002-08-26	2004-08-03	Sk Corporation	Benzoyl piperidine compounds
BR0317324A (pt) *	2002-12-18	2005-11-16	Fmc Corp	N-(arilmetil substituìdo)-4-(metil dissubstituìdo) piperidinas e piridinas
SE0400208D0 (sv) *	2004-02-02	2004-02-02	Astrazeneca Ab	Chemical compounds
TW200812582A (en) *	2006-04-06	2008-03-16	Astrazeneca Ab	Medicaments
BR112017003658B1 (pt)	2014-08-28	2022-12-06	Asceneuron Sa	Composto, mistura, método para inibição de uma glicosidase, e, composição farmacêutica
US10913733B2 (en)	2015-12-18	2021-02-09	Alectos Therapeutics Inc.	Substituted piperidines thiazolyl acetamides as glycosidase inhibitors and uses thereof
EP3419976B1 (en)	2016-02-25	2021-04-07	Asceneuron SA	Acid addition salts of piperazine derivatives
EP3585783A2 (en)	2016-02-25	2020-01-01	Asceneuron SA	Sulfoximine glycosidase inhibitors
AU2017222964B2 (en)	2016-02-25	2020-01-02	Asceneuron S. A.	Glycosidase inhibitors
US11612599B2 (en)	2016-02-25	2023-03-28	Asceneuron Sa	Glycosidase inhibitors
EP3672959A1 (en)	2017-08-24	2020-07-01	Asceneuron SA	Linear glycosidase inhibitors
WO2020039028A1 (en)	2018-08-22	2020-02-27	Asceneuron S. A.	Tetrahydro-benzoazepine glycosidase inhibitors
US11731972B2 (en)	2018-08-22	2023-08-22	Asceneuron Sa	Spiro compounds as glycosidase inhibitors
US12016852B2 (en)	2018-08-22	2024-06-25	Asceneuron Sa	Pyrrolidine glycosidase inhibitors
EP3841093B1 (en)	2018-08-22	2023-06-21	Asceneuron SA	Succinate and fumarate acid addition salts of piperazine derivatives useful as glycosidase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US450780A (en) *		1891-04-21		Steam-engine
US4180583A (en) *	1972-01-28	1979-12-25	Richardson-Merrell Inc.	Olefinic 4-substituted piperidino derivatives as therapeutics
US3922276A (en) *	1974-12-11	1975-11-25	Robins Co Inc A H	1-Substituted-4-benzylidenepiperidines
US4540780A (en) *	1983-06-02	1985-09-10	Warner-Lambert Company	Diphenylmethylene piperidines
US4666905A (en) *	1983-06-02	1987-05-19	Warner-Lambert Company	Diphenylmethylene piperidines compositions and methods for their use
MX173362B (es) *	1987-03-02	1994-02-23	Pfizer	Compuestos de piperazinil heterociclicos y procedimiento para su preparacion

1996
- 1996-07-01 IL IL11876896A patent/IL118768A/xx not_active IP Right Cessation
- 1996-07-04 ZA ZA965691A patent/ZA965691B/xx unknown
- 1996-07-09 PT PT96927006T patent/PT842170E/pt unknown
- 1996-07-09 WO PCT/EP1996/003099 patent/WO1997003065A1/en not_active Ceased
- 1996-07-09 RU RU98102392/04A patent/RU2162846C2/ru not_active IP Right Cessation
- 1996-07-09 DK DK96927006T patent/DK0842170T3/da active
- 1996-07-09 HU HU9802762A patent/HUP9802762A3/hu unknown
- 1996-07-09 CA CA002226851A patent/CA2226851A1/en not_active Abandoned
- 1996-07-09 PL PL96324451A patent/PL183837B1/pl unknown
- 1996-07-09 DE DE69611788T patent/DE69611788T2/de not_active Expired - Fee Related
- 1996-07-09 TR TR1998/00027T patent/TR199800027T1/xx unknown
- 1996-07-09 AU AU66993/96A patent/AU699370B2/en not_active Ceased
- 1996-07-09 ES ES96927006T patent/ES2156287T3/es not_active Expired - Lifetime
- 1996-07-09 CN CN96195461A patent/CN1091108C/zh not_active Expired - Fee Related
- 1996-07-09 CZ CZ199883A patent/CZ288909B6/cs not_active IP Right Cessation
- 1996-07-09 US US08/983,059 patent/US5935974A/en not_active Expired - Fee Related
- 1996-07-09 EP EP96927006A patent/EP0842170B1/en not_active Expired - Lifetime
- 1996-07-09 BR BR9609330A patent/BR9609330A/pt active Search and Examination
- 1996-07-09 AT AT96927006T patent/ATE199150T1/de not_active IP Right Cessation
- 1996-07-09 JP JP9505516A patent/JPH11508907A/ja active Pending
- 1996-07-09 NZ NZ315318A patent/NZ315318A/en unknown
- 1996-07-09 KR KR1019980700107A patent/KR19990028807A/ko not_active Ceased
- 1996-07-12 AR ARP960103567A patent/AR003966A1/es active IP Right Grant
- 1996-07-29 TW TW085109218A patent/TW419477B/zh not_active IP Right Cessation
1998
- 1998-01-09 NO NO980109A patent/NO309765B1/no unknown
2001
- 2001-05-11 GR GR20010400699T patent/GR3035849T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR19990028807A (ko)	1999-04-15
CA2226851A1 (en)	1997-01-30
GR3035849T3 (en)	2001-08-31
HK1010818A1 (en)	1999-07-02
PL183837B1 (pl)	2002-07-31
TW419477B (en)	2001-01-21
ATE199150T1 (de)	2001-02-15
DE69611788D1 (de)	2001-03-22
IL118768A (en)	2000-10-31
BR9609330A (pt)	1999-05-25
EP0842170A1 (en)	1998-05-20
US5935974A (en)	1999-08-10
JPH11508907A (ja)	1999-08-03
AR003966A1 (es)	1998-09-30
IL118768A0 (en)	1996-10-31
NO309765B1 (no)	2001-03-26
NZ315318A (en)	1999-10-28
RU2162846C2 (ru)	2001-02-10
AU6699396A (en)	1997-02-10
MX9800368A (es)	1998-03-31
AU699370B2 (en)	1998-12-03
WO1997003065A1 (en)	1997-01-30
PL324451A1 (en)	1998-05-25
CZ288909B6 (cs)	2001-09-12
ES2156287T3 (es)	2001-06-16
NO980109D0 (no)	1998-01-09
EP0842170B1 (en)	2001-02-14
CN1091108C (zh)	2002-09-18
HUP9802762A2 (hu)	1999-10-28
CN1190965A (zh)	1998-08-19
CZ8398A3 (cs)	1998-06-17
HUP9802762A3 (en)	2002-10-28
TR199800027T1 (xx)	1998-05-21
PT842170E (pt)	2001-06-29
DK0842170T3 (da)	2001-06-18
DE69611788T2 (de)	2001-08-02
ZA965691B (en)	1997-01-24

Publication	Publication Date	Title
NO980109D0 (no)	1998-01-09	Difenylmetylen-piperidin-derivater
DE69522717D1 (de)	2001-10-18	Chinazolinderivate
DE69611361D1 (de)	2001-02-01	Chinazolin-derivate
NO974103D0 (no)	1997-09-05	Arylsulfonylaminohydroksamsyre-derivater
DE69610698D1 (de)	2000-11-23	Chinazolin-derivate
FI941022L (fi)	1994-09-05	Spirosykliset piperidiinijohdannaiset
FI943976A7 (fi)	1995-03-01	5-aryyli-indolijohdannaiset
ATE278695T1 (de)	2004-10-15	Piperidinderivate
NO964667D0 (no)	1996-11-05	Purin-6-on-derivater
FI942444A7 (fi)	1994-11-28	Terahydropyraanijohdannaisia
FI943885L (fi)	1995-02-25	Penaami-johdannaiset
ATA100695A (de)	1998-03-15	Prothrombin-derivate
DE69627830D1 (de)	2003-06-05	Pyrazol-derivate
DE69628200D1 (de)	2003-06-18	Diarylalkenylamin-derivate
DE69635580D1 (de)	2006-01-19	Impulsgeber
NO992302D0 (no)	1999-05-12	Piperidin-derivater
NO961404D0 (no)	1996-04-09	4-indolylpiperazinyl-derivater
DK0846683T3 (da)	2001-11-05	4-hydroxypiperidinderivater
DK0723963T3 (da)	2001-09-24	4-Amino-benzoylguanidin-derivater
DE59610106D1 (de)	2003-03-13	Fluorbenzylether-Derivate
ATE177102T1 (de)	1999-03-15	Chromanderivate
DK0843675T3 (da)	2003-02-10	Aza-anthracyclinonderivater
DE59407726D1 (de)	1999-03-11	3-Aryl-4-hydroxy-3-dihydrofuranon-Derivate
DE59607055D1 (de)	2001-07-19	4-Mercapto-benzoylguanidin-Derivate
DE69620514D1 (de)	2002-05-16	5-aminoflavon-derivate