IL136738A0 - Inhibition of p38 kinase activity using substituted heterocyclic ureas - Google Patents

Inhibition of p38 kinase activity using substituted heterocyclic ureas

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Publication number
IL136738A0
IL136738A0 IL13673898A IL13673898A IL136738A0 IL 136738 A0 IL136738 A0 IL 136738A0 IL 13673898 A IL13673898 A IL 13673898A IL 13673898 A IL13673898 A IL 13673898A IL 136738 A0 IL136738 A0 IL 136738A0
Authority
IL
Israel
Prior art keywords
inhibition
kinase activity
substituted heterocyclic
heterocyclic ureas
ureas
Prior art date
Application number
IL13673898A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of IL136738A0 publication Critical patent/IL136738A0/xx

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
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    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
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    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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IL13673898A 1997-12-22 1998-12-22 Inhibition of p38 kinase activity using substituted heterocyclic ureas IL136738A0 (en)

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IL136738A IL136738A (en) 1997-12-22 2000-06-12 USE OF SUBSTITUTED HETEROCYCLIC UREAS FOR THE PREPARATION OF MEDICAMENTS FOR TREATING A DISEASE MEDIATED BY p38 OTHER THAN CANCER
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IL170201A IL170201A (en) 1997-12-22 2005-08-10 Sustituted heterocyclic ureas and pharmaceutical compositions comprising them

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AU739642B2 (en) 2001-10-18
IL170201A (en) 2006-12-31
JP2001526223A (ja) 2001-12-18
EP1041982A4 (fr) 2006-06-14
DE1041982T1 (de) 2001-06-07
IL136738A (en) 2007-06-17
ATE529109T1 (de) 2011-11-15
CA2315720A1 (fr) 1999-07-01
MXPA00006233A (es) 2002-09-18
JP4403482B2 (ja) 2010-01-27
EP1041982B1 (fr) 2011-10-19
WO1999032111A1 (fr) 1999-07-01
ES2154253T1 (es) 2001-04-01
ES2154253T3 (es) 2012-01-27
EP1041982A1 (fr) 2000-10-11
AU1997199A (en) 1999-07-12

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