IL153364A0 - PROCESS FOR THE PREPARATION OS SALTS OF 5-PHENYLPENTANOYL-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-{(S)-2-[(r)-3-AMINO-2-OXOPYRROLIDIN-1-YL]PROPIONYL}-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-4-AMINOPHENYLACETAMIDE, INTERMEDIATES USED IN THE PROCESS AND PROCESS FOR THEIR PREPARATION - Google Patents

PROCESS FOR THE PREPARATION OS SALTS OF 5-PHENYLPENTANOYL-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-{(S)-2-[(r)-3-AMINO-2-OXOPYRROLIDIN-1-YL]PROPIONYL}-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-4-AMINOPHENYLACETAMIDE, INTERMEDIATES USED IN THE PROCESS AND PROCESS FOR THEIR PREPARATION

Info

Publication number: IL153364A0
Authority: IL; Israel
Prior art keywords: alanyl; arginyl; preparation; aminophenylacetamide; phenylpentanoyl
Prior art date: 2000-07-22

Application number

IL15336401A

Other languages

English (en)

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-07-22

Filing date

2001-07-18

Publication date

2003-07-06

2001-07-18 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2003-07-06 Publication of IL153364A0 publication Critical patent/IL153364A0/xx

Links

238000000034 method Methods 0.000 title 3
SPCXPAYQHPMHJI-MINGNZLKSA-N (4s)-4-[[(2s)-2-[[(2s)-2-[[(2s)-2-[(3r)-3-amino-2-oxopyrrolidin-1-yl]propanoyl]-[(2s)-2-[[(2s)-5-(diaminomethylideneamino)-2-[[(2s)-2-(5-phenylpentanoylamino)propanoyl]amino]pentanoyl]amino]propanoyl]amino]propanoyl]amino]-5-(diaminomethylideneamino)penta Chemical class N([C@@H](C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)N([C@@H](C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C)C(=O)C(C(N)=O)C=1C=CC(N)=CC=1)C(=O)[C@H](C)N1C([C@H](N)CC1)=O)C(=O)CCCCC1=CC=CC=C1 SPCXPAYQHPMHJI-MINGNZLKSA-N 0.000 title 1
239000000543 intermediate Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
- C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
- C07K14/4713—Autoimmune diseases, e.g. Insulin-dependent diabetes mellitus, multiple sclerosis, rheumathoid arthritis, systemic lupus erythematosus; Autoantigens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
- C07K14/70503—Immunoglobulin superfamily
- C07K14/70539—MHC-molecules, e.g. HLA-molecules

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Immunology (AREA)
Medicinal Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Gastroenterology & Hepatology (AREA)
Zoology (AREA)
Toxicology (AREA)
Rheumatology (AREA)
Diabetes (AREA)
Hematology (AREA)
Rehabilitation Therapy (AREA)
Cell Biology (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

IL15336401A 2000-07-22 2001-07-18 PROCESS FOR THE PREPARATION OS SALTS OF 5-PHENYLPENTANOYL-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-{(S)-2-[(r)-3-AMINO-2-OXOPYRROLIDIN-1-YL]PROPIONYL}-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-4-AMINOPHENYLACETAMIDE, INTERMEDIATES USED IN THE PROCESS AND PROCESS FOR THEIR PREPARATION IL153364A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0017979.6A GB0017979D0 (en)	2000-07-22	2000-07-22	Chemical process
PCT/GB2001/003228 WO2002008247A2 (en)	2000-07-22	2001-07-18	Process for the preparation of 5-phenylpentanoyl-ala-argl-{2-[3-amino-2-oxopyrrolidin-1-yl]propionyl}-ala-arg-ala-4-aminophenylacetamide

Publications (1)

Publication Number	Publication Date
IL153364A0 true IL153364A0 (en)	2003-07-06

Family

ID=9896124

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL15336401A IL153364A0 (en)	2000-07-22	2001-07-18	PROCESS FOR THE PREPARATION OS SALTS OF 5-PHENYLPENTANOYL-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-{(S)-2-[(r)-3-AMINO-2-OXOPYRROLIDIN-1-YL]PROPIONYL}-(S)-ALANYL-(S)-ARGINYL-(S)-ALANYL-4-AMINOPHENYLACETAMIDE, INTERMEDIATES USED IN THE PROCESS AND PROCESS FOR THEIR PREPARATION

Country Status (18)

Country	Link
US (1)	US20040101864A1 (cs)
EP (1)	EP1320538A2 (cs)
JP (1)	JP2004504405A (cs)
KR (1)	KR20030033001A (cs)
CN (1)	CN1617881A (cs)
AU (1)	AU2001270863A1 (cs)
BR (1)	BR0112652A (cs)
CA (1)	CA2412787A1 (cs)
CZ (1)	CZ2003165A3 (cs)
GB (1)	GB0017979D0 (cs)
HU (1)	HUP0400485A3 (cs)
IL (1)	IL153364A0 (cs)
MX (1)	MXPA03000607A (cs)
NO (1)	NO20030317L (cs)
NZ (1)	NZ523217A (cs)
PL (1)	PL365426A1 (cs)
WO (1)	WO2002008247A2 (cs)
ZA (1)	ZA200210247B (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0130286D0 (en) *	2001-12-19	2002-02-06	Astrazeneca Ab	Chemical process
GB0130285D0 (en) *	2001-12-19	2002-02-06	Astrazeneca Ab	Chemical process
US7923577B2 (en)	2009-04-27	2011-04-12	International Flavors & Fragrances Inc.	Menthylcarboxamides and their use as cooling agents
JP6084021B2 (ja) *	2012-12-04	2017-02-22	富士通テン株式会社	表示システム、表示装置、表示方法、及び、プログラム
CN111848433B (zh) *	2020-07-14	2023-04-28	安徽中草香料股份有限公司	4-氨基苯基乙酰胺的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1155925A (en) *	1967-02-16	1969-06-25	Miles Lab	Synthesis Of Octapeptides
US4152322A (en) *	1978-04-28	1979-05-01	Merck & Co., Inc.	Process for selective reduction of nitroarginyl peptides with titanium (iii)
GB9702377D0 (en) *	1996-02-23	1997-03-26	Zeneca Ltd	Peptide derivatives

2000
- 2000-07-22 GB GBGB0017979.6A patent/GB0017979D0/en not_active Ceased
2001
- 2001-07-18 AU AU2001270863A patent/AU2001270863A1/en not_active Abandoned
- 2001-07-18 KR KR10-2003-7000906A patent/KR20030033001A/ko not_active Withdrawn
- 2001-07-18 CN CNA018130984A patent/CN1617881A/zh active Pending
- 2001-07-18 HU HU0400485A patent/HUP0400485A3/hu unknown
- 2001-07-18 MX MXPA03000607A patent/MXPA03000607A/es not_active Application Discontinuation
- 2001-07-18 US US10/333,571 patent/US20040101864A1/en not_active Abandoned
- 2001-07-18 CZ CZ2003165A patent/CZ2003165A3/cs unknown
- 2001-07-18 BR BR0112652-0A patent/BR0112652A/pt not_active Application Discontinuation
- 2001-07-18 EP EP01949746A patent/EP1320538A2/en not_active Withdrawn
- 2001-07-18 JP JP2002514151A patent/JP2004504405A/ja active Pending
- 2001-07-18 IL IL15336401A patent/IL153364A0/xx unknown
- 2001-07-18 NZ NZ523217A patent/NZ523217A/en unknown
- 2001-07-18 PL PL01365426A patent/PL365426A1/xx unknown
- 2001-07-18 WO PCT/GB2001/003228 patent/WO2002008247A2/en not_active Ceased
- 2001-07-18 CA CA002412787A patent/CA2412787A1/en not_active Abandoned
2002
- 2002-12-18 ZA ZA200210247A patent/ZA200210247B/en unknown
2003
- 2003-01-21 NO NO20030317A patent/NO20030317L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
BR0112652A (pt)	2003-07-01
US20040101864A1 (en)	2004-05-27
WO2002008247A3 (en)	2002-10-17
JP2004504405A (ja)	2004-02-12
CN1617881A (zh)	2005-05-18
CZ2003165A3 (cs)	2003-04-16
NZ523217A (en)	2004-07-30
CA2412787A1 (en)	2002-01-31
MXPA03000607A (es)	2003-05-14
NO20030317L (no)	2003-03-14
HUP0400485A3 (en)	2005-02-28
GB0017979D0 (en)	2000-09-13
ZA200210247B (en)	2003-10-31
EP1320538A2 (en)	2003-06-25
KR20030033001A (ko)	2003-04-26
AU2001270863A1 (en)	2002-02-05
WO2002008247A2 (en)	2002-01-31
PL365426A1 (en)	2005-01-10
HUP0400485A2 (hu)	2004-06-28
NO20030317D0 (no)	2003-01-21

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