IL63406A0 - Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL63406A0
IL63406A0 IL63406A IL6340681A IL63406A0 IL 63406 A0 IL63406 A0 IL 63406A0 IL 63406 A IL63406 A IL 63406A IL 6340681 A IL6340681 A IL 6340681A IL 63406 A0 IL63406 A0 IL 63406A0
Authority
IL
Israel
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
benzodiazepine derivatives
benzodiazepine
Prior art date
Application number
IL63406A
Other languages
English (en)
Original Assignee
Sparamedica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sparamedica Ag filed Critical Sparamedica Ag
Publication of IL63406A0 publication Critical patent/IL63406A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL63406A 1980-07-31 1981-07-24 Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them IL63406A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH584180 1980-07-31

Publications (1)

Publication Number Publication Date
IL63406A0 true IL63406A0 (en) 1981-10-30

Family

ID=4300189

Family Applications (1)

Application Number Title Priority Date Filing Date
IL63406A IL63406A0 (en) 1980-07-31 1981-07-24 Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them

Country Status (9)

Country Link
US (1) US4327026A (fr)
EP (1) EP0045452A3 (fr)
JP (1) JPS5758674A (fr)
AU (1) AU7339781A (fr)
CA (1) CA1157855A (fr)
DK (1) DK341181A (fr)
IL (1) IL63406A0 (fr)
PH (1) PH17045A (fr)
ZA (1) ZA815115B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3431195A1 (de) * 1984-08-24 1986-03-06 Troponwerke GmbH & Co KG, 5000 Köln Neue benzodiazepine, verfahren zu ihrer herstellung sowie ihre verwendung
US5939412A (en) * 1992-06-26 1999-08-17 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists
WO1993000095A2 (fr) * 1991-06-28 1993-01-07 Smithkline Beecham Corporation Antagonistes bicycliques de fibrinogene
US6403578B1 (en) 1993-12-21 2002-06-11 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists
MA23420A1 (fr) * 1994-01-07 1995-10-01 Smithkline Beecham Corp Antagonistes bicycliques de fibrinogene.
US6458784B1 (en) 1994-06-29 2002-10-01 Smithkline Beecham Corporation Vitronectin receptor antagonists
US5977101A (en) * 1995-06-29 1999-11-02 Smithkline Beecham Corporation Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity
US6100254A (en) * 1997-10-10 2000-08-08 Board Of Regents, The University Of Texas System Inhibitors of protein tyrosine kinases
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
WO2012075456A1 (fr) 2010-12-02 2012-06-07 Constellation Pharmaceuticals Inhibiteurs de bromodomaines et leurs utilisations
WO2012151512A2 (fr) 2011-05-04 2012-11-08 Constellation Pharmaceuticals, Inc. Inhibiteurs de bromodomaines et leurs utilisations
EP2721031B1 (fr) 2011-06-17 2016-01-20 Constellation Pharmaceuticals, Inc. Inhibiteurs à bromodomaine et leurs utilisations
TWI602820B (zh) 2012-06-06 2017-10-21 星宿藥物公司 溴域抑制劑及其用途
EP2864336B1 (fr) 2012-06-06 2016-11-23 Constellation Pharmaceuticals, Inc. Inhibiteurs de bromo-domaine de benzo[b]isoxazoloazépines et applications associées
TR201906788T4 (tr) 2014-06-20 2019-05-21 Constellation Pharmaceuticals Inc 2-((4s)-6-(4-klorofenil)-1-metil-4h-benzo[c]izoksazolo[4,5-e]azepın-4-il)asetamidin kristal formları.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL23270A (en) * 1964-04-10 1969-02-27 Hoffmann La Roche Quinazoline derivatives and process for the manufacture and conversion thereof
DE2163622A1 (de) * 1971-12-21 1973-06-28 Standard Elektrik Lorenz Ag Steuerung von wechselspannungsgeraeten
CA1114373A (fr) * 1978-08-11 1981-12-15 Albert E. Fischli Derives de benzodiazepine

Also Published As

Publication number Publication date
ZA815115B (en) 1982-08-25
US4327026A (en) 1982-04-27
EP0045452A2 (fr) 1982-02-10
AU7339781A (en) 1982-02-04
DK341181A (da) 1982-02-01
EP0045452A3 (fr) 1982-03-31
CA1157855A (fr) 1983-11-29
JPS5758674A (en) 1982-04-08
PH17045A (en) 1984-05-17

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