IL88183A0 - Intermediates for the preparation of halogenated protease inhibitors - Google Patents

Intermediates for the preparation of halogenated protease inhibitors

Info

Publication number: IL88183A0
Authority: IL; Israel
Prior art keywords: intermediates; halogenated; preparation; protease inhibitors; protease
Prior art date: 1987-10-29

Application number

IL88183A

Other languages

English (en)

Original Assignee

Searle & Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-10-29

Filing date

1988-10-27

Publication date

1989-06-30

1988-10-27 Application filed by Searle & Co filed Critical Searle & Co

1989-06-30 Publication of IL88183A0 publication Critical patent/IL88183A0/xx

Links

229940042399 direct acting antivirals protease inhibitors Drugs 0.000 title 1
239000000543 intermediate Substances 0.000 title 1
239000000137 peptide hydrolase inhibitor Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/78—Benzoic acid esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
- C07C69/716—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
- C07C69/72—Acetoacetic acid esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/02—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen
- C07C69/22—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen having three or more carbon atoms in the acid moiety

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

IL88183A 1987-10-29 1988-10-27 Intermediates for the preparation of halogenated protease inhibitors IL88183A0 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/114,186 US4803294A (en)	1987-10-29	1987-10-29	Process and intermediates for the preparation of halogenated protease inhibitors

Publications (1)

Publication Number	Publication Date
IL88183A0 true IL88183A0 (en)	1989-06-30

Family

ID=22353816

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL88183A IL88183A0 (en)	1987-10-29	1988-10-27	Intermediates for the preparation of halogenated protease inhibitors

Country Status (12)

Country	Link
US (1)	US4803294A (da)
EP (1)	EP0314126A3 (da)
JP (1)	JPH01149754A (da)
KR (1)	KR890006562A (da)
AU (1)	AU2437488A (da)
DK (1)	DK602288A (da)
FI (1)	FI884958A7 (da)
IL (1)	IL88183A0 (da)
NO (1)	NO884818L (da)
NZ (1)	NZ226749A (da)
PT (1)	PT88870B (da)
ZA (1)	ZA888113B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7063838B1 (en) *	1999-09-24	2006-06-20	Proteon Therapeutics Llc	Methods for treating an artery or vein in a human subject
US7632494B2 (en) *	1999-09-24	2009-12-15	Proteon Therapeutics, Inc.	Methods for enlarging the diameter of a biological conduit in a human subject
AU7612100A (en) *	1999-09-24	2001-04-24	Johns Hopkins University, The	Systems and methods for opening obstructed biological conduits

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4469885A (en) *	1983-05-09	1984-09-04	G. D. Searle & Co.	Halogenated protease inhibitors
US4499295A (en) *	1983-05-09	1985-02-12	G. D. Searle & Co.	Protease inhibitors
US4501895A (en) *	1983-05-09	1985-02-26	G.D. Searle & Co.	[Halo-4-(4,5-dihydro-4,4-dimethyl-2-oxazolyl)-phenyl]octadecan-ols and -ones

1987
- 1987-10-29 US US07/114,186 patent/US4803294A/en not_active Expired - Lifetime
1988
- 1988-10-27 IL IL88183A patent/IL88183A0/xx unknown
- 1988-10-27 AU AU24374/88A patent/AU2437488A/en not_active Withdrawn
- 1988-10-27 PT PT88870A patent/PT88870B/pt not_active IP Right Cessation
- 1988-10-27 KR KR1019880014026A patent/KR890006562A/ko not_active Withdrawn
- 1988-10-27 EP EP88117897A patent/EP0314126A3/en not_active Ceased
- 1988-10-27 NZ NZ226749A patent/NZ226749A/xx unknown
- 1988-10-27 FI FI884958A patent/FI884958A7/fi not_active IP Right Cessation
- 1988-10-28 DK DK602288A patent/DK602288A/da not_active Application Discontinuation
- 1988-10-28 JP JP63271108A patent/JPH01149754A/ja active Pending
- 1988-10-28 ZA ZA888113A patent/ZA888113B/xx unknown
- 1988-10-28 NO NO88884818A patent/NO884818L/no unknown

Also Published As

Publication number	Publication date
EP0314126A2 (en)	1989-05-03
FI884958A7 (fi)	1989-04-30
EP0314126A3 (en)	1990-01-31
JPH01149754A (ja)	1989-06-12
AU2437488A (en)	1989-05-04
NO884818L (no)	1989-05-02
PT88870B (pt)	1993-01-29
NZ226749A (en)	1989-10-27
FI884958A0 (fi)	1988-10-27
DK602288A (da)	1989-04-30
KR890006562A (ko)	1989-06-14
DK602288D0 (da)	1988-10-28
ZA888113B (en)	1989-12-27
US4803294A (en)	1989-02-07
NO884818D0 (no)	1988-10-28

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