IL94943A - Preparation of penem compounds - Google Patents

Preparation of penem compounds

Info

Publication number
IL94943A
IL94943A IL9494390A IL9494390A IL94943A IL 94943 A IL94943 A IL 94943A IL 9494390 A IL9494390 A IL 9494390A IL 9494390 A IL9494390 A IL 9494390A IL 94943 A IL94943 A IL 94943A
Authority
IL
Israel
Prior art keywords
compound
formula
group
halogen atom
hydroxy group
Prior art date
Application number
IL9494390A
Other languages
English (en)
Other versions
IL94943A0 (en
Inventor
Ettore Perrone
Marco Alpegiani
Franco Zarini
Giuseppe Mazzini
Giovanni Franceschi
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of IL94943A0 publication Critical patent/IL94943A0/xx
Publication of IL94943A publication Critical patent/IL94943A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/32—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D317/34—Oxygen atoms
    • C07D317/40—Vinylene carbonate; Substituted vinylene carbonates
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Glass Compositions (AREA)
  • Electric Double-Layer Capacitors Or The Like (AREA)
  • Medicinal Preparation (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
  • Magnetic Resonance Imaging Apparatus (AREA)
  • Measurement And Recording Of Electrical Phenomena And Electrical Characteristics Of The Living Body (AREA)
  • Pens And Brushes (AREA)
IL9494390A 1989-07-05 1990-07-02 Preparation of penem compounds IL94943A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898915392A GB8915392D0 (en) 1989-07-05 1989-07-05 Process for penems

Publications (2)

Publication Number Publication Date
IL94943A0 IL94943A0 (en) 1991-06-10
IL94943A true IL94943A (en) 1994-11-11

Family

ID=10659566

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9494390A IL94943A (en) 1989-07-05 1990-07-02 Preparation of penem compounds

Country Status (21)

Country Link
EP (2) EP0433425A1 (de)
JP (1) JPH05500210A (de)
KR (1) KR920701212A (de)
AT (1) ATE131483T1 (de)
AU (1) AU644805B2 (de)
CA (1) CA2035434A1 (de)
DD (1) DD299304A5 (de)
DE (1) DE69024114T2 (de)
DK (1) DK0406790T3 (de)
ES (1) ES2083401T3 (de)
FI (1) FI911081A7 (de)
GB (1) GB8915392D0 (de)
HU (1) HU209924B (de)
IE (1) IE902423A1 (de)
IL (1) IL94943A (de)
MY (1) MY105720A (de)
NZ (1) NZ234329A (de)
PT (1) PT94589A (de)
RU (1) RU2049786C1 (de)
WO (1) WO1991000283A1 (de)
ZA (1) ZA905198B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8818789D0 (en) * 1988-08-08 1988-09-07 Erba Carlo Spa Crystalline(5r 6s)-2-carbamoyloxymethyl-6-((1r)-hydroxyethyl)-2-penem-carboxylic acid & pharmaceutical formulation
GB9006114D0 (en) * 1990-03-19 1990-05-16 Erba Carlo Spa Process for preparing penem esters
IT1286558B1 (it) * 1996-02-27 1998-07-15 Menarini Farma Ind Processo per la preparazione di 2-alogenometil-penems e loro uso per la preparazione di penems antibatterici

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5835190A (ja) * 1981-08-25 1983-03-01 Sankyo Co Ltd ペネム−３−カルボン酸誘導体
JPS59212488A (ja) * 1983-05-18 1984-12-01 Kyoto Yakuhin Kogyo Kk ジオキソ−ル誘導体
JPH075463B2 (ja) * 1985-03-09 1995-01-25 サントリー株式会社 抗菌剤
GB8713515D0 (en) * 1987-06-10 1987-07-15 Erba Farmitalia Methoxymethyl compounds
GB8716679D0 (en) * 1987-07-15 1987-08-19 Erba Farmitalia Penem derivatives

Also Published As

Publication number Publication date
ATE131483T1 (de) 1995-12-15
HU209924B (en) 1994-12-28
EP0406790A1 (de) 1991-01-09
DE69024114T2 (de) 1996-05-09
IE902423A1 (en) 1991-06-19
IL94943A0 (en) 1991-06-10
WO1991000283A1 (en) 1991-01-10
DD299304A5 (de) 1992-04-09
HU905471D0 (en) 1991-06-28
EP0406790B1 (de) 1995-12-13
AU644805B2 (en) 1993-12-23
EP0433425A1 (de) 1991-06-26
JPH05500210A (ja) 1993-01-21
DE69024114D1 (de) 1996-01-25
AU6031890A (en) 1991-01-17
RU2049786C1 (ru) 1995-12-10
PT94589A (pt) 1991-03-20
ES2083401T3 (es) 1996-04-16
FI911081A0 (fi) 1991-03-04
KR920701212A (ko) 1992-08-11
DK0406790T3 (da) 1996-01-29
FI911081A7 (fi) 1991-03-04
GB8915392D0 (en) 1989-08-23
NZ234329A (en) 1992-03-26
MY105720A (en) 1994-11-30
HUT56374A (en) 1991-08-28
ZA905198B (en) 1991-04-24
CA2035434A1 (en) 1991-01-06

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Legal Events

Date Code Title Description
RH Patent void