IN2014MN00841A - - Google Patents

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Publication number
IN2014MN00841A
IN2014MN00841A IN841MUN2014A IN2014MN00841A IN 2014MN00841 A IN2014MN00841 A IN 2014MN00841A IN 841MUN2014 A IN841MUN2014 A IN 841MUN2014A IN 2014MN00841 A IN2014MN00841 A IN 2014MN00841A
Authority
IN
India
Application number
Other languages
English (en)
Inventor
Jean-Claude Pascal
Original Assignee
Estetra Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48043195&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014MN00841(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Estetra Sprl filed Critical Estetra Sprl
Publication of IN2014MN00841A publication Critical patent/IN2014MN00841A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN841MUN2014 2011-10-07 2014-05-05 IN2014MN00841A (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161544591P 2011-10-07 2011-10-07
EP11184278 2011-10-07
PCT/EP2012/069761 WO2013050553A1 (en) 2011-10-07 2012-10-05 Process for the production of estetrol

Publications (1)

Publication Number Publication Date
IN2014MN00841A true IN2014MN00841A (sr) 2015-07-03

Family

ID=48043195

Family Applications (1)

Application Number Title Priority Date Filing Date
IN841MUN2014 IN2014MN00841A (sr) 2011-10-07 2014-05-05

Country Status (26)

Country Link
US (1) US8987484B2 (sr)
EP (1) EP2764008B1 (sr)
JP (1) JP6196625B2 (sr)
KR (1) KR102007874B1 (sr)
CN (1) CN103890001B (sr)
AU (1) AU2012320423C1 (sr)
BR (1) BR112014008196B8 (sr)
CA (1) CA2847813C (sr)
CL (1) CL2014000802A1 (sr)
CY (1) CY1118674T1 (sr)
DK (1) DK2764008T3 (sr)
EA (1) EA024003B1 (sr)
ES (1) ES2593316T3 (sr)
HR (1) HRP20161282T1 (sr)
HU (1) HUE028963T2 (sr)
IN (1) IN2014MN00841A (sr)
LT (1) LT2764008T (sr)
ME (1) ME02527B (sr)
MX (1) MX348917B (sr)
PL (1) PL2764008T3 (sr)
PT (1) PT2764008T (sr)
RS (1) RS55231B1 (sr)
SG (1) SG11201401282PA (sr)
SI (1) SI2764008T1 (sr)
SM (1) SMT201600375B (sr)
WO (1) WO2013050553A1 (sr)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS54880B1 (sr) 2011-06-01 2016-10-31 Estetra Sprl Postupak proizvodnje intermedijarnih proizvoda estetrola
ME02585B (me) 2011-06-01 2017-06-20 Estetra Sprl Postupak proizvodnje intermedijara estetrola
EP2383279A1 (en) 2011-07-19 2011-11-02 Pantarhei Bioscience B.V. Process for the preparation of estetrol
WO2013034780A2 (en) * 2012-12-20 2013-03-14 Crystal Pharma, S.A.U. Process for the preparation of estetrol and related compounds
ES2624667T3 (es) * 2013-09-18 2017-07-17 Crystal Pharma, S.A.U. Procedimiento para la preparación de estetrol
LT3310345T (lt) 2015-06-18 2021-06-25 Estetra Sprl Burnoje disperguojama tabletė, turinti estetrolio
MA44206B1 (fr) * 2015-06-18 2021-04-30 Estetra Sprl Comprimé orodispersible comprenant estetrol
CU24523B1 (es) 2015-06-18 2021-06-08 Estetra Sprl Unidad de dosificación orodispersable que contiene un componente estetrol
EP3701944B1 (en) 2015-06-18 2021-12-08 Estetra SRL Orodispersible dosage unit containing an estetrol component
CA3178291A1 (en) 2016-08-05 2018-04-12 Estetra Srl Method for the management of dysmenorrhea and menstrual pain
EP3781171B1 (en) 2018-04-19 2022-02-09 Estetra SRL Compounds and their uses for alleviating menopause-associated symptoms
TWI801561B (zh) 2018-04-19 2023-05-11 比利時商依思特拉私人有限責任公司 化合物及其用於緩解絕經相關症狀的用途
EP3647413A1 (en) * 2018-10-31 2020-05-06 Centro de Investigaciones Energéticas, Medioambientales y Tecnológicas O.A., M.P. (CIEMAT) Improvements for performing and facilitating the recovery after hematopoietic stem cell transplantation
HU231240B1 (hu) * 2019-09-03 2022-04-28 Richter Gedeon Nyrt. Ipari eljárás nagytisztaságú ösztetrol hatóanyag előállítására
IT201900021879A1 (it) 2019-11-22 2021-05-22 Ind Chimica Srl PROCESSO PER LA PREPARAZIONE DI (15α,16α,17β)-ESTRA-1,3,5(10)-TRIENE-3,15,16,17-TETROLO (ESTETROLO) ED INTERMEDI DI DETTO PROCESSO
DE112020004564T5 (de) 2019-09-27 2022-06-15 Industriale Chimica S.R.L. VERFAHREN ZUM HERSTELLEN VON (15α,16α,17β)-ESTRA-1,3,5(10)-TRIEN-3,15,16,17-TETROL (ESTETROL) UND ZWISCHENSTUFEN DES VERFAHRENS
IT201900017414A1 (it) 2019-09-27 2021-03-27 Ind Chimica Srl Processo per la preparazione di (15α,16α,17β)-estra-1,3,5(10)-triene-3,15,16,17-tetrolo (Estetrolo) ed intermedi di detto processo
TWI893101B (zh) 2020-04-16 2025-08-11 比利時商埃斯特拉有限責任公司 具有降低之副作用之避孕組成物
IT202100019631A1 (it) 2021-07-23 2023-01-23 Newchem S P A Metodo per produrre estetrolo e i suoi intermedi
WO2023021026A1 (en) 2021-08-17 2023-02-23 Aspen Oss B.V. A synthetic pathway to estra-1,3,5(10)-triene-3,15a,16a,17b-tetrol
HU231651B1 (hu) 2021-10-01 2025-05-28 Industriale Chimica S.R.L. Eljárás (15alfa,16alfa,17béta)-ösztra-1,3,5(10)-trién-3,15,16,17-tetrol (esztetrol) és esztetrol-monohidrát előállítására
JP2026503158A (ja) 2023-02-02 2026-01-27 インダストリアーレ キミカ エッセ.エッレ.エッレ. (15α,16α,17β)-エストラ-1,3,5(10)-トリエン-3,15,16,17-テトロール(エステトロール)一水和物の調製方法
CN121605114A (zh) * 2023-08-30 2026-03-03 埃斯特拉私人有限责任公司 雌四醇中间体的制造方法
HUP2400151A1 (hu) 2024-02-28 2025-09-28 Richter Gedeon Nyrt Ösztetrol-monohidrát kristályosítási eljárás
WO2025181200A1 (en) 2024-02-28 2025-09-04 Estetra Srl Estetrol polymorphic form and production thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW548277B (en) * 1999-07-16 2003-08-21 Akzo Nobel Nv Orally active androgens
IL149424A (en) * 1999-12-02 2007-05-15 Organon Nv Androgens are converted to methylene at positions 15,14
CN100343269C (zh) * 2002-11-08 2007-10-17 潘塔希生物科学股份有限公司 通过雌酮衍生的甾体化合物合成雌四醇
UA89964C2 (ru) * 2004-09-08 2010-03-25 Н.В. Органон 15β-ЗАМЕЩЕННЫЕ СТЕРОИДЫ, КОТОРЫЕ ИМЕЮТ СЕЛЕКТИВНУЮ ЭСТРОГЕННУЮ АКТИВНОСТЬ
ME02585B (me) 2011-06-01 2017-06-20 Estetra Sprl Postupak proizvodnje intermedijara estetrola
RS54880B1 (sr) 2011-06-01 2016-10-31 Estetra Sprl Postupak proizvodnje intermedijarnih proizvoda estetrola
EP2383279A1 (en) * 2011-07-19 2011-11-02 Pantarhei Bioscience B.V. Process for the preparation of estetrol

Also Published As

Publication number Publication date
SMT201600375B (it) 2017-01-10
CN103890001B (zh) 2016-05-04
WO2013050553A1 (en) 2013-04-11
US20140243539A1 (en) 2014-08-28
PT2764008T (pt) 2016-11-10
EP2764008A1 (en) 2014-08-13
HUE028963T2 (en) 2017-01-30
CA2847813A1 (en) 2013-04-11
SI2764008T1 (sl) 2016-10-28
CY1118674T1 (el) 2017-07-12
MX2014003723A (es) 2014-10-13
ME02527B (me) 2017-02-20
ES2593316T3 (es) 2016-12-07
SG11201401282PA (en) 2014-05-29
EA201490713A1 (ru) 2014-07-30
BR112014008196B1 (pt) 2020-10-20
LT2764008T (lt) 2016-11-10
HK1199882A1 (zh) 2015-07-24
BR112014008196B8 (pt) 2020-12-15
NZ621973A (en) 2015-08-28
KR102007874B1 (ko) 2019-08-06
AU2012320423B2 (en) 2017-02-09
AU2012320423A1 (en) 2014-03-20
JP6196625B2 (ja) 2017-09-13
CL2014000802A1 (es) 2014-11-14
MX348917B (es) 2017-07-04
US8987484B2 (en) 2015-03-24
BR112014008196A2 (pt) 2017-04-18
EA024003B1 (ru) 2016-08-31
PL2764008T3 (pl) 2017-04-28
AU2012320423C1 (en) 2018-01-25
KR20140083994A (ko) 2014-07-04
CN103890001A (zh) 2014-06-25
HRP20161282T1 (hr) 2016-11-18
JP2014528438A (ja) 2014-10-27
DK2764008T3 (en) 2016-11-07
RS55231B1 (sr) 2017-02-28
CA2847813C (en) 2018-12-11
EP2764008B1 (en) 2016-08-17

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